7ZXS

Name : Crystal structure of DPP9 in complex with a 4-oxo-b-lactam based inhibitor, A295

Revelation date : 28-Sep-2022

Family : DPP4N_Peptidase_S9

Gene_locus : human-DPP9

PDB file : ESTHER: header of PDB entry RCSB: Full entry

Comment
Ross, B.,Huber, R.

Ligand :

References (1)

Title : Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9 - Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498
Author(s) : Carvalho LAR , Ross B , Fehr L , Bolgi O , Wohrle S , Lum KM , Podlesainski D , Vieira AC , Kiefersauer R , Felix R , Rodrigues T , Lucas SD , Gross O , Geiss-Friedlander R , Cravatt BF , Huber R , Kaiser M , Moreira R
Ref : Angew Chem Int Ed Engl , : , 2022
Abstract : Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498
ESTHER : Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498
PubMedSearch : Carvalho_2022_Angew.Chem.Int.Ed.Engl_61_e202210498
PubMedID: 36089535
Gene_locus related to this paper: human-DPP8 , human-DPP9

Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server

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