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Title : Conjugates of Methylene Blue with Cycloalkaneindoles as New Multifunctional Agents for Potential Treatment of Neurodegenerative Disease - Bachurin_2022_Int.J.Mol.Sci_23_ |
Author(s) : Bachurin SO , Shevtsova EF , Makhaeva GF , Aksinenko AY , Grigoriev VV , Goreva TV , Epishina TA , Kovaleva NV , Boltneva NP , Lushchekina SV , Rudakova EV , Vinogradova DV , Shevtsov PN , Pushkareva EA , Dubova LG , Serkova TP , Veselov IM , Fisenko VP , Richardson RJ |
Ref : Int J Mol Sci , 23 : , 2022 |
Abstract : Bachurin_2022_Int.J.Mol.Sci_23_ |
ESTHER : Bachurin_2022_Int.J.Mol.Sci_23_ |
PubMedSearch : Bachurin_2022_Int.J.Mol.Sci_23_ |
PubMedID: 36430413 |
Title : Conjugation of Aminoadamantane and gamma-Carboline Pharmacophores Gives Rise to Unexpected Properties of Multifunctional Ligands - Bachurin_2021_Molecules_26_ |
Author(s) : Bachurin SO , Makhaeva GF , Shevtsova EF , Aksinenko AY , Grigoriev VV , Shevtsov PN , Goreva TV , Epishina TA , Kovaleva NV , Pushkareva EA , Boltneva NP , Lushchekina SV , Gabrelyan AV , Zamoyski VL , Dubova LG , Rudakova EV , Fisenko VP , Bovina EV , Richardson RJ |
Ref : Molecules , 26 : , 2021 |
Abstract : Bachurin_2021_Molecules_26_ |
ESTHER : Bachurin_2021_Molecules_26_ |
PubMedSearch : Bachurin_2021_Molecules_26_ |
PubMedID: 34576998 |
Title : Conjugates of methylene blue with gamma-carboline derivatives as new multifunctional agents for the treatment of neurodegenerative diseases - Bachurin_2019_Sci.Rep_9_4873 |
Author(s) : Bachurin SO , Makhaeva GF , Shevtsova EF , Boltneva NP , Kovaleva NV , Lushchekina SV , Rudakova EV , Dubova LG , Vinogradova DV , Sokolov VB , Aksinenko AY , Fisenko VP , Richardson RJ , Aliev G |
Ref : Sci Rep , 9 :4873 , 2019 |
Abstract : Bachurin_2019_Sci.Rep_9_4873 |
ESTHER : Bachurin_2019_Sci.Rep_9_4873 |
PubMedSearch : Bachurin_2019_Sci.Rep_9_4873 |
PubMedID: 30890752 |
Title : Novel conjugates of aminoadamantanes with carbazole derivatives as potential multitarget agents for AD treatment - Bachurin_2017_Sci.Rep_7_45627 |
Author(s) : Bachurin SO , Shevtsova EF , Makhaeva GF , Grigoriev VV , Boltneva NP , Kovaleva NV , Lushchekina SV , Shevtsov PN , Neganova ME , Redkozubova OM , Bovina EV , Gabrelyan AV , Fisenko VP , Sokolov VB , Aksinenko AY , Echeverria V , Barreto GE , Aliev G |
Ref : Sci Rep , 7 :45627 , 2017 |
Abstract : Bachurin_2017_Sci.Rep_7_45627 |
ESTHER : Bachurin_2017_Sci.Rep_7_45627 |
PubMedSearch : Bachurin_2017_Sci.Rep_7_45627 |
PubMedID: 28358144 |
Title : Esterase profiles of organophosphorus compounds in vitro predict their behavior in vivo - Makhaeva_2016_Chem.Biol.Interact_259_332 |
Author(s) : Makhaeva GF , Rudakova EV , Serebryakova OG , Aksinenko AY , Lushchekina SV , Bachurin SO , Richardson RJ |
Ref : Chemico-Biological Interactions , 259 :332 , 2016 |
Abstract : Makhaeva_2016_Chem.Biol.Interact_259_332 |
ESTHER : Makhaeva_2016_Chem.Biol.Interact_259_332 |
PubMedSearch : Makhaeva_2016_Chem.Biol.Interact_259_332 |
PubMedID: 27154493 |
Title : Conjugates of gamma-Carbolines and Phenothiazine as new selective inhibitors of butyrylcholinesterase and blockers of NMDA receptors for Alzheimer Disease - Makhaeva_2015_Sci.Rep_5_13164 |
Author(s) : Makhaeva GF , Lushchekina SV , Boltneva NP , Sokolov VB , Grigoriev VV , Serebryakova OG , Vikhareva EA , Aksinenko AY , Barreto GE , Aliev G , Bachurin SO |
Ref : Sci Rep , 5 :13164 , 2015 |
Abstract : Makhaeva_2015_Sci.Rep_5_13164 |
ESTHER : Makhaeva_2015_Sci.Rep_5_13164 |
PubMedSearch : Makhaeva_2015_Sci.Rep_5_13164 |
PubMedID: 26281952 |
Title : Organophosphorus compound esterase profiles as predictors of therapeutic and toxic effects - Makhaeva_2013_Chem.Biol.Interact_203_231 |
Author(s) : Makhaeva GF , Radchenko EV , Palyulin VA , Rudakova EV , Aksinenko AY , Sokolov VB , Zefirov NS , Richardson RJ |
Ref : Chemico-Biological Interactions , 203 :231 , 2013 |
Abstract : Makhaeva_2013_Chem.Biol.Interact_203_231 |
ESTHER : Makhaeva_2013_Chem.Biol.Interact_203_231 |
PubMedSearch : Makhaeva_2013_Chem.Biol.Interact_203_231 |
PubMedID: 23123251 |
Title : A new selective inhibitor of mouse blood plasma carboxylesterase - |
Author(s) : Rudakova EV , Makhaeva GF , Galenko TG , Aksinenko AY , Sokolov VB , Martynov IV |
Ref : Dokl Biochem Biophys , 449 :87 , 2013 |
PubMedID: 23657654 |
Title : Kinetics and mechanism of inhibition of serine esterases by fluorinated carbethoxy 1-aminophosphonates - |
Author(s) : Makhaeva GF , Lushchekina SV , Serebryakova OG , Aksinenko AY , Goreva TV , Richardson RJ , Martynov IV |
Ref : Dokl Biochem Biophys , 451 :203 , 2013 |
PubMedID: 23975401 |
Title : Esterase profile of O-phosphorylated ethyltrifluorolactates in prediction of their therapeutic and toxic effects - |
Author(s) : Rudakova EV , Makhaeva GF , Galenko TG , Aksinenko AY , Sokolov VB , Richardson RJ , Martynov IV |
Ref : Dokl Biochem Biophys , 443 :81 , 2012 |
PubMedID: 22562631 |
Title : Kinetics and mechanism of inhibition of serine esterases by fluorinated aminophosphonates - Makhaeva_2010_Chem.Biol.Interact_187_177 |
Author(s) : Makhaeva GF , Aksinenko AY , Sokolov VB , Baskin, II , Palyulin VA , Zefirov NS , Hein ND , Kampf JW , Wijeyesakere SJ , Richardson RJ |
Ref : Chemico-Biological Interactions , 187 :177 , 2010 |
Abstract : Makhaeva_2010_Chem.Biol.Interact_187_177 |
ESTHER : Makhaeva_2010_Chem.Biol.Interact_187_177 |
PubMedSearch : Makhaeva_2010_Chem.Biol.Interact_187_177 |
PubMedID: 20035729 |
Title : Synthesis of organophosphates with fluorine-containing leaving groups as serine esterase inhibitors with potential for Alzheimer disease therapeutics - Makhaeva_2009_Bioorg.Med.Chem.Lett_19_5528 |
Author(s) : Makhaeva GF , Aksinenko AY , Sokolov VB , Serebryakova OG , Richardson RJ |
Ref : Bioorganic & Medicinal Chemistry Lett , 19 :5528 , 2009 |
Abstract : Makhaeva_2009_Bioorg.Med.Chem.Lett_19_5528 |
ESTHER : Makhaeva_2009_Bioorg.Med.Chem.Lett_19_5528 |
PubMedSearch : Makhaeva_2009_Bioorg.Med.Chem.Lett_19_5528 |
PubMedID: 19717305 |
Title : Diethyl [2,2,2-trifluoro-1-phenyl-sulfonyl-amino-1-(trifluoro-meth-yl)eth-yl]phospho-nate - Wijeyesakere_2008_Acta.Crystallogr.Sect.E.Struct.Rep.Online_64_o1425 |
Author(s) : Wijeyesakere SJ , Nasser FA , Kampf JW , Aksinenko AY , Sokolov VB , Malygin VV , Makhaeva GF , Richardson RJ |
Ref : Acta Crystallographica Sect E Struct Rep Online , 64 :o1425 , 2008 |
Abstract : Wijeyesakere_2008_Acta.Crystallogr.Sect.E.Struct.Rep.Online_64_o1425 |
ESTHER : Wijeyesakere_2008_Acta.Crystallogr.Sect.E.Struct.Rep.Online_64_o1425 |
PubMedSearch : Wijeyesakere_2008_Acta.Crystallogr.Sect.E.Struct.Rep.Online_64_o1425 |
PubMedID: 19079747 |
Title : Esterase profile and analysis of structure-inhibitor selectivity relationships for homologous phosphorylated 1-hydroperfluoroisopropanols - |
Author(s) : Makhaeva GF , Serebryakova OG , Boltneva NP , Galenko TG , Aksinenko AY , Sokolov VB , Martynov IV |
Ref : Dokl Biochem Biophys , 423 :352 , 2008 |
PubMedID: 19230387 |
Title : Fluorinated alpha-aminophosphonates--a new type of irreversible inhibitors of serine hydrolases - |
Author(s) : Makhaeva GF , Malygin VV , Aksinenko AY , Sokolov VB , Strakhova NN , Rasdolsky AN , Richardson RJ , Martynov IV |
Ref : Dokl Biochem Biophys , 400 :92 , 2005 |
PubMedID: 15846994 |
Title : Poster: The fluorocontaining derivatives of alpha-aminoalkylphosphonates a new type of cholinesterase inhibitors - |
Author(s) : Kuusk VV , Agabekian RS , Morozova IV , Kovaleva NV , Rasdolsky AN , Sokolov VB , Aksinenko AY , Fetisov VI , Martynov IV |
Ref : In: Cholinesterases: Structure, Function, Mechanism, Genetics, and Cell Biology , (Massoulie J, Barnard EA, Chatonnet A, Bacou F, Doctor BP, Quinn DM) American Chemical Society, Washington, DC :293 , 1991 |
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