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| Title : Novel multifunctional tacrine-donepezil hybrids against Alzheimer's disease: Design synthesis and bioactivity studies - Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575 |
| Author(s) : Bayraktar G , Bartolini M , Bolognesi ML , Erdogan MA , Armagan G , Bayir E , Sendemir A , Bagetta D , Alcaro S , Alptuzun V |
| Ref : Arch Pharm (Weinheim) , :e2300575 , 2024 |
| Abstract : Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575 |
| ESTHER : Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575 |
| PubMedSearch : Bayraktar_2024_Arch.Pharm.(Weinheim)__e2300575 |
| PubMedID: 38593283 |
| Title : Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease - Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
| Author(s) : Moutayakine A , Marques C , Lopez O , Bagetta D , Leitzbach L , Hagenow S , Carreiro EP , Stark H , Alcaro S , Fernandez-Bolanos JG , Burke AJ |
| Ref : Bioorganic & Medicinal Chemistry , 68 :116807 , 2022 |
| Abstract : Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
| ESTHER : Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
| PubMedSearch : Moutayakine_2022_Bioorg.Med.Chem_68_116807 |
| PubMedID: 35653868 |
| Title : Design, Synthesis, and In Vitro, In Silico and In Cellulo Evaluation of New Pyrimidine and Pyridine Amide and Carbamate Derivatives as Multi-Functional Cholinesterase Inhibitors - Bortolami_2022_Pharmaceuticals.(Basel)_15_ |
| Author(s) : Bortolami M , Pandolfi F , Tudino V , Messore A , Madia VN , De Vita D , Di Santo R , Costi R , Romeo I , Alcaro S , Colone M , Stringaro A , Espargaro A , Sabate R , Scipione L |
| Ref : Pharmaceuticals (Basel) , 15 : , 2022 |
| Abstract : Bortolami_2022_Pharmaceuticals.(Basel)_15_ |
| ESTHER : Bortolami_2022_Pharmaceuticals.(Basel)_15_ |
| PubMedSearch : Bortolami_2022_Pharmaceuticals.(Basel)_15_ |
| PubMedID: 35745594 |
| Title : Novel propargylamine-based inhibitors of cholinesterases and monoamine oxidases: Synthesis, biological evaluation and docking study - Kratky_2021_Bioorg.Chem_116_105301 |
| Author(s) : Kratky M , Vu QA , Stepankova S , Maruca A , Silva TB , Ambroz M , Pflegr V , Rocca R , Svrckova K , Alcaro S , Borges F , Vinsova J |
| Ref : Bioorg Chem , 116 :105301 , 2021 |
| Abstract : Kratky_2021_Bioorg.Chem_116_105301 |
| ESTHER : Kratky_2021_Bioorg.Chem_116_105301 |
| PubMedSearch : Kratky_2021_Bioorg.Chem_116_105301 |
| PubMedID: 34492558 |
| Title : New Pyrimidine and Pyridine Derivatives as Multitarget Cholinesterase Inhibitors: Design, Synthesis, and In Vitro and In Cellulo Evaluation - Bortolami_2021_ACS.Chem.Neurosci__ |
| Author(s) : Bortolami M , Pandolfi F , Tudino V , Messore A , Madia VN , De Vita D , Di Santo R , Costi R , Romeo I , Alcaro S , Colone M , Stringaro A , Espargaro A , Sabate R , Scipione L |
| Ref : ACS Chem Neurosci , : , 2021 |
| Abstract : Bortolami_2021_ACS.Chem.Neurosci__ |
| ESTHER : Bortolami_2021_ACS.Chem.Neurosci__ |
| PubMedSearch : Bortolami_2021_ACS.Chem.Neurosci__ |
| PubMedID: 34652128 |
| Title : N-1,2,3-triazole-isatin derivatives for cholinesterase and beta-amyloid aggregation inhibition: A comprehensive bioassay study - Marques_2020_Bioorg.Chem_98_103753 |
| Author(s) : Marques CS , Lopez O , Bagetta D , Carreiro EP , Petralla S , Bartolini M , Hoffmann M , Alcaro S , Monti B , Bolognesi ML , Decker M , Fernandez-Bolanos JG , Burke AJ |
| Ref : Bioorg Chem , 98 :103753 , 2020 |
| Abstract : Marques_2020_Bioorg.Chem_98_103753 |
| ESTHER : Marques_2020_Bioorg.Chem_98_103753 |
| PubMedSearch : Marques_2020_Bioorg.Chem_98_103753 |
| PubMedID: 32200328 |
| Title : New deferiprone derivatives as multi-functional cholinesterase inhibitors: design, synthesis and in vitro evaluation - Bortolami_2020_Eur.J.Med.Chem_198_112350 |
| Author(s) : Bortolami M , Pandolfi F , De Vita D , Carafa C , Messore A , Di Santo R , Feroci M , Costi R , Chiarotto I , Bagetta D , Alcaro S , Colone M , Stringaro A , Scipione L |
| Ref : Eur Journal of Medicinal Chemistry , 198 :112350 , 2020 |
| Abstract : Bortolami_2020_Eur.J.Med.Chem_198_112350 |
| ESTHER : Bortolami_2020_Eur.J.Med.Chem_198_112350 |
| PubMedSearch : Bortolami_2020_Eur.J.Med.Chem_198_112350 |
| PubMedID: 32380385 |
| Title : Benzoic acid-derived nitrones: A new class of potential acetylcholinesterase inhibitors and neuroprotective agents - Oliveira_2019_Eur.J.Med.Chem_174_116 |
| Author(s) : Oliveira C , Bagetta D , Cagide F , Teixeira J , Amorim R , Silva T , Garrido J , Remiao F , Uriarte E , Oliveira PJ , Alcaro S , Ortuso F , Borges F |
| Ref : Eur Journal of Medicinal Chemistry , 174 :116 , 2019 |
| Abstract : Oliveira_2019_Eur.J.Med.Chem_174_116 |
| ESTHER : Oliveira_2019_Eur.J.Med.Chem_174_116 |
| PubMedSearch : Oliveira_2019_Eur.J.Med.Chem_174_116 |
| PubMedID: 31029943 |
| Title : The chemistry toolbox of multitarget-directed ligands for Alzheimer's disease - Mesiti_2019_Eur.J.Med.Chem_181_111572 |
| Author(s) : Mesiti F , Chavarria D , Gaspar A , Alcaro S , Borges F |
| Ref : Eur Journal of Medicinal Chemistry , 181 :111572 , 2019 |
| Abstract : Mesiti_2019_Eur.J.Med.Chem_181_111572 |
| ESTHER : Mesiti_2019_Eur.J.Med.Chem_181_111572 |
| PubMedSearch : Mesiti_2019_Eur.J.Med.Chem_181_111572 |
| PubMedID: 31404859 |
| Title : 4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis - Secci_2019_J.Enzyme.Inhib.Med.Chem_34_597 |
| Author(s) : Secci D , Carradori S , Petzer A , Guglielmi P , D'Ascenzio M , Chimenti P , Bagetta D , Alcaro S , Zengin G , Petzer JP , Ortuso F |
| Ref : J Enzyme Inhib Med Chem , 34 :597 , 2019 |
| Abstract : Secci_2019_J.Enzyme.Inhib.Med.Chem_34_597 |
| ESTHER : Secci_2019_J.Enzyme.Inhib.Med.Chem_34_597 |
| PubMedSearch : Secci_2019_J.Enzyme.Inhib.Med.Chem_34_597 |
| PubMedID: 30727777 |
| Title : Multi-target-directed ligands for Alzheimer's disease: Discovery of chromone-based monoamine oxidase\/cholinesterase inhibitors - Reis_2018_Eur.J.Med.Chem_158_781 |
| Author(s) : Reis J , Cagide F , Valencia ME , Teixeira J , Bagetta D , Perez C , Uriarte E , Oliveira PJ , Ortuso F , Alcaro S , Rodriguez-Franco MI , Borges F |
| Ref : Eur Journal of Medicinal Chemistry , 158 :781 , 2018 |
| Abstract : Reis_2018_Eur.J.Med.Chem_158_781 |
| ESTHER : Reis_2018_Eur.J.Med.Chem_158_781 |
| PubMedSearch : Reis_2018_Eur.J.Med.Chem_158_781 |
| PubMedID: 30245401 |
| Title : Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents - Carradori_2018_Eur.J.Med.Chem_143_1543 |
| Author(s) : Carradori S , Ortuso F , Petzer A , Bagetta D , De Monte C , Secci D , De Vita D , Guglielmi P , Zengin G , Aktumsek A , Alcaro S , Petzer JP |
| Ref : Eur Journal of Medicinal Chemistry , 143 :1543 , 2018 |
| Abstract : Carradori_2018_Eur.J.Med.Chem_143_1543 |
| ESTHER : Carradori_2018_Eur.J.Med.Chem_143_1543 |
| PubMedSearch : Carradori_2018_Eur.J.Med.Chem_143_1543 |
| PubMedID: 29126727 |
| Title : (Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies - D'Ascenzio_2015_J.Enzyme.Inhib.Med.Chem_30_908 |
| Author(s) : D'Ascenzio M , Chimenti P , Gidaro MC , De Monte C , De Vita D , Granese A , Scipione L , Di Santo R , Costa G , Alcaro S , Yanez M , Carradori S |
| Ref : J Enzyme Inhib Med Chem , 30 :908 , 2015 |
| Abstract : D'Ascenzio_2015_J.Enzyme.Inhib.Med.Chem_30_908 |
| ESTHER : D'Ascenzio_2015_J.Enzyme.Inhib.Med.Chem_30_908 |
| PubMedSearch : D'Ascenzio_2015_J.Enzyme.Inhib.Med.Chem_30_908 |
| PubMedID: 25807300 |
| Title : N-Methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2- yl)methyl)prop-2-yn-1-amine, a new cholinesterase and monoamine oxidase dual inhibitor - Bautista-Aguilera_2014_J.Med.Chem_57_10455 |
| Author(s) : Bautista-Aguilera OM , Samadi A , Chioua M , Nikolic K , Filipic S , Agbaba D , Soriano E , de Andres L , Rodriguez-Franco MI , Alcaro S , Ramsay RR , Ortuso F , Yanez M , Marco-Contelles J |
| Ref : Journal of Medicinal Chemistry , 57 :10455 , 2014 |
| Abstract : Bautista-Aguilera_2014_J.Med.Chem_57_10455 |
| ESTHER : Bautista-Aguilera_2014_J.Med.Chem_57_10455 |
| PubMedSearch : Bautista-Aguilera_2014_J.Med.Chem_57_10455 |
| PubMedID: 25418133 |
| Title : Molecular modelling and enzymatic studies of acetylcholinesterase and butyrylcholinesterase recognition with paraquat and related compounds - Alcaro_2007_SAR.QSAR.Environ.Res_18_595 |
| Author(s) : Alcaro S , Arcone R , Vecchio I , Ortuso F , Gallelli A , Pasceri R , Procopio A , Iannone M |
| Ref : SAR QSAR Environ Research , 18 :595 , 2007 |
| Abstract : Alcaro_2007_SAR.QSAR.Environ.Res_18_595 |
| ESTHER : Alcaro_2007_SAR.QSAR.Environ.Res_18_595 |
| PubMedSearch : Alcaro_2007_SAR.QSAR.Environ.Res_18_595 |
| PubMedID: 17654339 |
| Title : An approach to address Candida rugosa lipase regioselectivity in the acylation reactions of trytilated glucosides - Palocci_2007_J.Biotechnol_128_908 |
| Author(s) : Palocci C , Falconi M , Alcaro S , Tafi A , Puglisi R , Ortuso F , Botta M , Alberghina L , Cernia E |
| Ref : J Biotechnol , 128 :908 , 2007 |
| Abstract : Palocci_2007_J.Biotechnol_128_908 |
| ESTHER : Palocci_2007_J.Biotechnol_128_908 |
| PubMedSearch : Palocci_2007_J.Biotechnol_128_908 |
| PubMedID: 17321623 |
| Title : Further studies on the interaction of the 5-hydroxytryptamine3 (5-HT3) receptor with arylpiperazine ligands. development of a new 5-HT3 receptor ligand showing potent acetylcholinesterase inhibitory properties - Cappelli_2005_J.Med.Chem_48_3564 |
| Author(s) : Cappelli A , Gallelli A , Manini M , Anzini M , Mennuni L , Makovec F , Menziani MC , Alcaro S , Ortuso F , Vomero S |
| Ref : Journal of Medicinal Chemistry , 48 :3564 , 2005 |
| Abstract : Cappelli_2005_J.Med.Chem_48_3564 |
| ESTHER : Cappelli_2005_J.Med.Chem_48_3564 |
| PubMedSearch : Cappelli_2005_J.Med.Chem_48_3564 |
| PubMedID: 15887964 |
| Title : Molecular modeling and enzymatic studies of the interaction of a choline analogue and acetylcholinesterase - Alcaro_2002_Bioorg.Med.Chem.Lett_12_2899 |
| Author(s) : Alcaro S , Scipione L , Ortuso F , Posca S , Rispoli V , Rotiroti D |
| Ref : Bioorganic & Medicinal Chemistry Lett , 12 :2899 , 2002 |
| Abstract : Alcaro_2002_Bioorg.Med.Chem.Lett_12_2899 |
| ESTHER : Alcaro_2002_Bioorg.Med.Chem.Lett_12_2899 |
| PubMedSearch : Alcaro_2002_Bioorg.Med.Chem.Lett_12_2899 |
| PubMedID: 12270172 |