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| Title : 1-((3S,4S)-4-amino-1-(4-substituted-1,3,5-triazin-2-yl) pyrrolidin-3-yl)-5,5-difluoropiperidin-2-one inhibitors of DPP-4 for the treatment of type 2 diabetes - Andrews_2011_Bioorg.Med.Chem.Lett_21_1810 |
| Author(s) : Andrews KM , Beebe DA , Benbow JW , Boyer DA , Doran SD , Hui Y , Liu S , McPherson RK , Neagu C , Parker JC , Piotrowski DW , Schneider SR , Treadway JL , VanVolkenberg MA , Zembrowski WJ |
| Ref : Bioorganic & Medicinal Chemistry Lett , 21 :1810 , 2011 |
| Abstract : Andrews_2011_Bioorg.Med.Chem.Lett_21_1810 |
| ESTHER : Andrews_2011_Bioorg.Med.Chem.Lett_21_1810 |
| PubMedSearch : Andrews_2011_Bioorg.Med.Chem.Lett_21_1810 |
| PubMedID: 21324688 |
| Title : (3,3-Difluoro-pyrrolidin-1-yl)-[(2S,4S)-(4-(4-pyrimidin-2-yl-piperazin-1-yl)-pyrr olidin-2-yl]-methanone: a potent, selective, orally active dipeptidyl peptidase IV inhibitor - Ammirati_2009_Bioorg.Med.Chem.Lett_19_1991 |
| Author(s) : Ammirati MJ , Andrews KM , Boyer DD , Brodeur AM , Danley DE , Doran SD , Hulin B , Liu S , McPherson RK , Orena SJ , Parker JC , Polivkova J , Qiu X , Soglia CB , Treadway JL , VanVolkenburg MA , Wilder DC , Piotrowski DW |
| Ref : Bioorganic & Medicinal Chemistry Lett , 19 :1991 , 2009 |
| Abstract : Ammirati_2009_Bioorg.Med.Chem.Lett_19_1991 |
| ESTHER : Ammirati_2009_Bioorg.Med.Chem.Lett_19_1991 |
| PubMedSearch : Ammirati_2009_Bioorg.Med.Chem.Lett_19_1991 |
| PubMedID: 19275964 |
| Gene_locus related to this paper: human-DPP4 |
| Title : (3R,4S)-4-(2,4,5-Trifluorophenyl)-pyrrolidin-3-ylamine inhibitors of dipeptidyl peptidase IV: synthesis, in vitro, in vivo, and X-ray crystallographic characterization - Wright_2007_Bioorg.Med.Chem.Lett_17_5638 |
| Author(s) : Wright SW , Ammirati MJ , Andrews KM , Brodeur AM , Danley DE , Doran SD , Lillquist JS , Liu S , McClure LD , McPherson RK , Olson TV , Orena SJ , Parker JC , Rocke BN , Soeller WC , Soglia CB , Treadway JL , VanVolkenburg MA , Zhao Z , Cox ED |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :5638 , 2007 |
| Abstract : Wright_2007_Bioorg.Med.Chem.Lett_17_5638 |
| ESTHER : Wright_2007_Bioorg.Med.Chem.Lett_17_5638 |
| PubMedSearch : Wright_2007_Bioorg.Med.Chem.Lett_17_5638 |
| PubMedID: 17822893 |
| Gene_locus related to this paper: human-DPP4 |
| Title : cis-2,5-dicyanopyrrolidine inhibitors of dipeptidyl peptidase IV: synthesis and in vitro, in vivo, and X-ray crystallographic characterization - Wright_2006_J.Med.Chem_49_3068 |
| Author(s) : Wright SW , Ammirati MJ , Andrews KM , Brodeur AM , Danley DE , Doran SD , Lillquist JS , McClure LD , McPherson RK , Orena SJ , Parker JC , Polivkova J , Qiu X , Soeller WC , Soglia CB , Treadway JL , VanVolkenburg MA , Wang H , Wilder DC , Olson TV |
| Ref : Journal of Medicinal Chemistry , 49 :3068 , 2006 |
| Abstract : Wright_2006_J.Med.Chem_49_3068 |
| ESTHER : Wright_2006_J.Med.Chem_49_3068 |
| PubMedSearch : Wright_2006_J.Med.Chem_49_3068 |
| PubMedID: 16722626 |
| Title : New fluorinated pyrrolidine and azetidine amides as dipeptidyl peptidase IV inhibitors - Hulin_2005_Bioorg.Med.Chem.Lett_15_4770 |
| Author(s) : Hulin B , Cabral S , Lopaze MG , Van Volkenburg MA , Andrews KM , Parker JC |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :4770 , 2005 |
| Abstract : Hulin_2005_Bioorg.Med.Chem.Lett_15_4770 |
| ESTHER : Hulin_2005_Bioorg.Med.Chem.Lett_15_4770 |
| PubMedSearch : Hulin_2005_Bioorg.Med.Chem.Lett_15_4770 |
| PubMedID: 16115768 |