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Title : (3,3-Difluoro-pyrrolidin-1-yl)-[(2S,4S)-(4-(4-pyrimidin-2-yl-piperazin-1-yl)-pyrr olidin-2-yl]-methanone: a potent, selective, orally active dipeptidyl peptidase IV inhibitor - Ammirati_2009_Bioorg.Med.Chem.Lett_19_1991 |
Author(s) : Ammirati MJ , Andrews KM , Boyer DD , Brodeur AM , Danley DE , Doran SD , Hulin B , Liu S , McPherson RK , Orena SJ , Parker JC , Polivkova J , Qiu X , Soglia CB , Treadway JL , VanVolkenburg MA , Wilder DC , Piotrowski DW |
Ref : Bioorganic & Medicinal Chemistry Lett , 19 :1991 , 2009 |
Abstract : Ammirati_2009_Bioorg.Med.Chem.Lett_19_1991 |
ESTHER : Ammirati_2009_Bioorg.Med.Chem.Lett_19_1991 |
PubMedSearch : Ammirati_2009_Bioorg.Med.Chem.Lett_19_1991 |
PubMedID: 19275964 |
Gene_locus related to this paper: human-DPP4 |