Report for Brogi S

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References (7)

Title : Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization - Butini_2024_J.Med.Chem__
Author(s) : Butini S , Grether U , Jung KM , Ligresti A , Allara M , Postmus AGJ , Maramai S , Brogi S , Papa A , Carullo G , Sykes D , Veprintsev D , Federico S , Grillo A , Di Guglielmo B , Ramunno A , Stevens AF , Heer D , Lamponi S , Gemma S , Benz J , Di Marzo V , van der Stelt M , Piomelli D , Campiani G
Ref : Journal of Medicinal Chemistry , : , 2024
Abstract : Butini_2024_J.Med.Chem__
ESTHER : Butini_2024_J.Med.Chem__
PubMedSearch : Butini_2024_J.Med.Chem__
PubMedID: 38241614
Gene_locus related to this paper: human-MGLL

Title : MicroRNA-Based Multitarget Approach for Alzheimer's Disease: Discovery of the First-In-Class Dual Inhibitor of Acetylcholinesterase and MicroRNA-15b Biogenesis - Gabr_2020_J.Med.Chem_63_9695
Author(s) : Gabr MT , Brogi S
Ref : Journal of Medicinal Chemistry , 63 :9695 , 2020
Abstract : Gabr_2020_J.Med.Chem_63_9695
ESTHER : Gabr_2020_J.Med.Chem_63_9695
PubMedSearch : Gabr_2020_J.Med.Chem_63_9695
PubMedID: 32787143

Title : Multitarget compounds bearing tacrine- and donepezil-like structural and functional motifs for the potential treatment of Alzheimer's disease - Ismaili_2017_Prog.Neurobiol_151_4
Author(s) : Ismaili L , Refouvelet B , Benchekroun M , Brogi S , Brindisi M , Gemma S , Campiani G , Filipic S , Agbaba D , Esteban G , Unzeta M , Nikolic K , Butini S , Marco-Contelles J
Ref : Prog Neurobiol , 151 :4 , 2017
Abstract : Ismaili_2017_Prog.Neurobiol_151_4
ESTHER : Ismaili_2017_Prog.Neurobiol_151_4
PubMedSearch : Ismaili_2017_Prog.Neurobiol_151_4
PubMedID: 26797191

Title : Donepezil-like multifunctional agents: Design, synthesis, molecular modeling and biological evaluation - Wu_2016_Eur.J.Med.Chem_121_864
Author(s) : Wu MY , Esteban G , Brogi S , Shionoya M , Wang L , Campiani G , Unzeta M , Inokuchi T , Butini S , Marco-Contelles J
Ref : Eur Journal of Medicinal Chemistry , 121 :864 , 2016
Abstract : Wu_2016_Eur.J.Med.Chem_121_864
ESTHER : Wu_2016_Eur.J.Med.Chem_121_864
PubMedSearch : Wu_2016_Eur.J.Med.Chem_121_864
PubMedID: 26471320

Title : Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain - Brindisi_2016_J.Med.Chem_59_2612
Author(s) : Brindisi M , Maramai S , Gemma S , Brogi S , Grillo A , Di Cesare Mannelli L , Gabellieri E , Lamponi S , Saponara S , Gorelli B , Tedesco D , Bonfiglio T , Landry C , Jung KM , Armirotti A , Luongo L , Ligresti A , Piscitelli F , Bertucci C , Dehouck MP , Campiani G , Maione S , Ghelardini C , Pittaluga A , Piomelli D , Di Marzo V , Butini S
Ref : Journal of Medicinal Chemistry , 59 :2612 , 2016
Abstract : Brindisi_2016_J.Med.Chem_59_2612
ESTHER : Brindisi_2016_J.Med.Chem_59_2612
PubMedSearch : Brindisi_2016_J.Med.Chem_59_2612
PubMedID: 26888301

Title : Disease-Modifying Anti-Alzheimer's Drugs: Inhibitors of Human Cholinesterases Interfering with beta-Amyloid Aggregation - Brogi_2014_CNS.Neurosci.Ther_20_624
Author(s) : Brogi S , Butini S , Maramai S , Colombo R , Verga L , Lanni C , De Lorenzi E , Lamponi S , Andreassi M , Bartolini M , Andrisano V , Novellino E , Campiani G , Brindisi M , Gemma S
Ref : CNS Neurosci Ther , 20 :624 , 2014
Abstract : Brogi_2014_CNS.Neurosci.Ther_20_624
ESTHER : Brogi_2014_CNS.Neurosci.Ther_20_624
PubMedSearch : Brogi_2014_CNS.Neurosci.Ther_20_624
PubMedID: 24935788

Title : Multifunctional cholinesterase and amyloid Beta fibrillization modulators. Synthesis and biological investigation - Butini_2013_ACS.Med.Chem.Lett_4_1178
Author(s) : Butini S , Brindisi M , Brogi S , Maramai S , Guarino E , Panico A , Saxena A , Chauhan V , Colombo R , Verga L , De Lorenzi E , Bartolini M , Andrisano V , Novellino E , Campiani G , Gemma S
Ref : ACS Med Chem Lett , 4 :1178 , 2013
Abstract : Butini_2013_ACS.Med.Chem.Lett_4_1178
ESTHER : Butini_2013_ACS.Med.Chem.Lett_4_1178
PubMedSearch : Butini_2013_ACS.Med.Chem.Lett_4_1178
PubMedID: 24900626