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Title : Identification and Optimization of Novel Inhibitors of the Polyketide Synthase 13 Thioesterase Domain with Antitubercular Activity - Green_2023_J.Med.Chem__ |
Author(s) : Green SR , Wilson C , Eadsforth TC , Punekar AS , Tamaki FK , Wood G , Caldwell N , Forte B , Norcross NR , Kiczun M , Post JM , Lopez-Roman EM , Engelhart CA , Lukac I , Zuccotto F , Epemolu O , Boshoff HIM , Schnappinger D , Walpole C , Gilbert IH , Read KD , Wyatt PG , Baragana B |
Ref : Journal of Medicinal Chemistry , : , 2023 |
Abstract : Green_2023_J.Med.Chem__ |
ESTHER : Green_2023_J.Med.Chem__ |
PubMedSearch : Green_2023_J.Med.Chem__ |
PubMedID: 37948640 |
Gene_locus related to this paper: myctu-PKS13 |
Title : Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13\; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target - Wilson_2022_J.Med.Chem_65_409 |
Author(s) : Wilson C , Ray P , Zuccotto F , Hernandez J , Aggarwal A , Mackenzie C , Caldwell N , Taylor M , Huggett M , Mathieson M , Murugesan D , Smith A , Davis S , Cocco M , Parai MK , Acharya A , Tamaki F , Scullion P , Epemolu O , Riley J , Stojanovski L , Lopez-Roman EM , Torres-Gomez PA , Toledo AM , Guijarro-Lopez L , Camino I , Engelhart CA , Schnappinger D , Massoudi LM , Lenaerts A , Robertson GT , Walpole C , Matthews D , Floyd D , Sacchettini JC , Read KD , Encinas L , Bates RH , Green SR , Wyatt PG |
Ref : Journal of Medicinal Chemistry , 65 :409 , 2022 |
Abstract : Wilson_2022_J.Med.Chem_65_409 |
ESTHER : Wilson_2022_J.Med.Chem_65_409 |
PubMedSearch : Wilson_2022_J.Med.Chem_65_409 |
PubMedID: 34910486 |
Gene_locus related to this paper: myctu-PKS13 |