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Title : Identification of Reversible Small Molecule Inhibitors of Endothelial Lipase (EL) That Demonstrate HDL-C Increase In Vivo - Tora_2020_J.Med.Chem_63_1660 |
Author(s) : Tora G , Kim SH , Pi Z , Johnson JA , Jiang J , Phillips M , Lloyd J , Abell LM , Lu H , Locke G , Adam LP , Taylor DS , Yin X , Behnia K , Zhao L , Yang R , Basso M , Caporuscio C , Chen AY , Liu E , Kirshgessner T , Onorato JM , Ryan C , Traeger SC , Gordon D , Wexler RR , Finlay HJ |
Ref : Journal of Medicinal Chemistry , 63 :1660 , 2020 |
Abstract : Tora_2020_J.Med.Chem_63_1660 |
ESTHER : Tora_2020_J.Med.Chem_63_1660 |
PubMedSearch : Tora_2020_J.Med.Chem_63_1660 |
PubMedID: 31990537 |
Title : Sulfonylated Benzothiazoles as Inhibitors of Endothelial Lipase - Johnson_2018_ACS.Med.Chem.Lett_9_1263 |
Author(s) : Johnson JA , Tora G , Pi Z , Phillips M , Yin X , Yang R , Zhao L , Chen AY , Taylor DS , Basso M , Rose A , Behnia K , Onorato J , Chen XQ , Abell LM , Lu H , Locke G , Caporuscio C , Galella M , Adam LP , Gordon D , Wexler RR , Finlay HJ |
Ref : ACS Med Chem Lett , 9 :1263 , 2018 |
Abstract : Johnson_2018_ACS.Med.Chem.Lett_9_1263 |
ESTHER : Johnson_2018_ACS.Med.Chem.Lett_9_1263 |
PubMedSearch : Johnson_2018_ACS.Med.Chem.Lett_9_1263 |
PubMedID: 30613337 |
Gene_locus related to this paper: human-LIPG |