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| Title : Diethoxyphosphoryloxy-oleanolic acid is a nanomolar-inhibitor of butyrylcholinesterase - Petrova_2024_Chem.Biol.Drug.Des_103_e14506 |
| Author(s) : Petrova AV , Poptsov AI , Heise NV , Csuk R , Kazakova OB |
| Ref : Chemical Biology Drug Des , 103 :e14506 , 2024 |
| Abstract : Petrova_2024_Chem.Biol.Drug.Des_103_e14506 |
| ESTHER : Petrova_2024_Chem.Biol.Drug.Des_103_e14506 |
| PubMedSearch : Petrova_2024_Chem.Biol.Drug.Des_103_e14506 |
| PubMedID: 38480508 |
| Title : Acetylcholinesterase inhibitory activity of modified lupane, oleanane, and ursane A-seco-triterpenoids - Petrova_2023_Chem.Biodivers__e202300185 |
| Author(s) : Petrova A , Kazakova OB , Nazarov IS , Csuk R , Heise NV |
| Ref : Chem Biodivers , :e202300185 , 2023 |
| Abstract : Petrova_2023_Chem.Biodivers__e202300185 |
| ESTHER : Petrova_2023_Chem.Biodivers__e202300185 |
| PubMedSearch : Petrova_2023_Chem.Biodivers__e202300185 |
| PubMedID: 36960660 |
| Title : Inhibitory properties of quinopimaric acid derivatives towards cholinesterases - Tretyakova_2023_Nat.Prod.Res__1 |
| Author(s) : Tretyakova E , Heise NV , Csuk R , Kazakova O |
| Ref : Nat Prod Res , :1 , 2023 |
| Abstract : Tretyakova_2023_Nat.Prod.Res__1 |
| ESTHER : Tretyakova_2023_Nat.Prod.Res__1 |
| PubMedSearch : Tretyakova_2023_Nat.Prod.Res__1 |
| PubMedID: 37812150 |
| Title : Substrate-like novel inhibitors of prolyl specific oligo peptidase for neurodegenerative disorders - Khan_2023_J.Biomol.Struct.Dyn__1 |
| Author(s) : Khan M , Halim SA , Waqas M , Golmohammadi F , Balalaie S , Csuk R , Uddin J , Khan A , Al-Harrasi A |
| Ref : J Biomol Struct Dyn , :1 , 2023 |
| Abstract : Khan_2023_J.Biomol.Struct.Dyn__1 |
| ESTHER : Khan_2023_J.Biomol.Struct.Dyn__1 |
| PubMedSearch : Khan_2023_J.Biomol.Struct.Dyn__1 |
| PubMedID: 37608559 |
| Gene_locus related to this paper: pig-ppce |
| Title : Synthesis and Exploitation of the Biological Profile of Novel Guanidino Xylofuranose Derivatives - Fortuna_2022_ChemMedChem__ |
| Author(s) : Fortuna A , Goncalves-Pereira R , Costa PJ , Jorda R , Vojackova V , Gonzalez G , Heise NV , Csuk R , Oliveira MC , Xavier NM |
| Ref : ChemMedChem , : , 2022 |
| Abstract : Fortuna_2022_ChemMedChem__ |
| ESTHER : Fortuna_2022_ChemMedChem__ |
| PubMedSearch : Fortuna_2022_ChemMedChem__ |
| PubMedID: 35576106 |
| Title : New amides derived from sclareolide as anticholinesterase agents - Silva_2022_Bioorg.Chem_130_106249 |
| Author(s) : Silva JG , Borgati TF , Lopes SMG , Heise N , Hoenke S , Csuk R , Barbosa LCA |
| Ref : Bioorg Chem , 130 :106249 , 2022 |
| Abstract : Silva_2022_Bioorg.Chem_130_106249 |
| ESTHER : Silva_2022_Bioorg.Chem_130_106249 |
| PubMedSearch : Silva_2022_Bioorg.Chem_130_106249 |
| PubMedID: 36356369 |
| Title : Cytotoxic Potential of a-Azepano- and 3-Amino-3,4-SeCo-Triterpenoids - Kazakova_2021_Int.J.Mol.Sci_22_ |
| Author(s) : Kazakova O , Smirnova I , Tret'yakova E , Csuk R , Hoenke S , Fischer L |
| Ref : Int J Mol Sci , 22 : , 2021 |
| Abstract : Kazakova_2021_Int.J.Mol.Sci_22_ |
| ESTHER : Kazakova_2021_Int.J.Mol.Sci_22_ |
| PubMedSearch : Kazakova_2021_Int.J.Mol.Sci_22_ |
| PubMedID: 33567783 |
| Title : N-methylated diazabicyclo[3.2.2]nonane substituted triterpenoic acids are excellent, hyperbolic and selective inhibitors for butyrylcholinesterase - Heise_2021_Eur.J.Med.Chem_227_113947 |
| Author(s) : Heise N , Friedrich S , Temml V , Schuster D , Siewert B , Csuk R |
| Ref : Eur Journal of Medicinal Chemistry , 227 :113947 , 2021 |
| Abstract : Heise_2021_Eur.J.Med.Chem_227_113947 |
| ESTHER : Heise_2021_Eur.J.Med.Chem_227_113947 |
| PubMedSearch : Heise_2021_Eur.J.Med.Chem_227_113947 |
| PubMedID: 34731766 |
| Title : 4-Benzyloxylonchocarpin and Muracatanes A-C from Ranunculus muricatus L. and Their Biological Effects - Hussain_2020_Biomolecules_10_ |
| Author(s) : Hussain H , Ali I , Wang D , Mamadalieva NZ , Hussain W , Csuk R , Loesche A , Fischer L , Staerk D , Anam S , AlZain MN , Mushtaq M , Ul-Haq Z , Ullah R , Noman OM , Abbas G , Green IR |
| Ref : Biomolecules , 10 : , 2020 |
| Abstract : Hussain_2020_Biomolecules_10_ |
| ESTHER : Hussain_2020_Biomolecules_10_ |
| PubMedSearch : Hussain_2020_Biomolecules_10_ |
| PubMedID: 33212893 |
| Title : Synthesis and cholinesterase inhibiting potential of A-ring azepano- and 3-amino-3,4-seco-triterpenoids - Kazakova_2020_Bioorg.Chem_101_104001 |
| Author(s) : Kazakova O , Smirnova I , Lopatina T , Giniyatullina G , Petrova A , Khusnutdinova E , Csuk R , Serbian I , Loesche A |
| Ref : Bioorg Chem , 101 :104001 , 2020 |
| Abstract : Kazakova_2020_Bioorg.Chem_101_104001 |
| ESTHER : Kazakova_2020_Bioorg.Chem_101_104001 |
| PubMedSearch : Kazakova_2020_Bioorg.Chem_101_104001 |
| PubMedID: 32683137 |
| Title : Caffeic acid phenethyl ester (CAPE)-derivatives act as selective inhibitors of acetylcholinesterase - Giessel_2019_Eur.J.Med.Chem_177_259 |
| Author(s) : Giessel JM , Loesche A , Csuk R |
| Ref : Eur Journal of Medicinal Chemistry , 177 :259 , 2019 |
| Abstract : Giessel_2019_Eur.J.Med.Chem_177_259 |
| ESTHER : Giessel_2019_Eur.J.Med.Chem_177_259 |
| PubMedSearch : Giessel_2019_Eur.J.Med.Chem_177_259 |
| PubMedID: 31158743 |
| Title : Novel 12-hydroxydehydroabietylamine derivatives act as potent and selective butyrylcholinesterase inhibitors - Loesche_2019_Bioorg.Chem_90_103092 |
| Author(s) : Loesche A , Wiemann J , Rohmer M , Brandt W , Csuk R |
| Ref : Bioorg Chem , 90 :103092 , 2019 |
| Abstract : Loesche_2019_Bioorg.Chem_90_103092 |
| ESTHER : Loesche_2019_Bioorg.Chem_90_103092 |
| PubMedSearch : Loesche_2019_Bioorg.Chem_90_103092 |
| PubMedID: 31280014 |
| Title : Triterpene-Based Carboxamides Act as Good Inhibitors of Butyrylcholinesterase - Loesche_2019_Molecules_24_ |
| Author(s) : Loesche A , Kahnt M , Serbian I , Brandt W , Csuk R |
| Ref : Molecules , 24 : , 2019 |
| Abstract : Loesche_2019_Molecules_24_ |
| ESTHER : Loesche_2019_Molecules_24_ |
| PubMedSearch : Loesche_2019_Molecules_24_ |
| PubMedID: 30866589 |
| Title : Synthesis and Biological Evaluation of Structurally Varied 5'-\/6'-Isonucleosides and Theobromine-Containing N-Isonucleosidyl Derivatives - Xavier_2019_Pharmaceuticals.(Basel)_12_ |
| Author(s) : Xavier NM , De Sousa EC , Pereira MP , Loesche A , Serbian I , Csuk R , Oliveira MC |
| Ref : Pharmaceuticals (Basel) , 12 : , 2019 |
| Abstract : Xavier_2019_Pharmaceuticals.(Basel)_12_ |
| ESTHER : Xavier_2019_Pharmaceuticals.(Basel)_12_ |
| PubMedSearch : Xavier_2019_Pharmaceuticals.(Basel)_12_ |
| PubMedID: 31269639 |
| Title : Substituted cinnamic anhydrides act as selective inhibitors of acetylcholinesterase - Giessel_2019_Bioorg.Chem_90_103058 |
| Author(s) : Giessel JM , Serbian I , Loesche A , Csuk R |
| Ref : Bioorg Chem , 90 :103058 , 2019 |
| Abstract : Giessel_2019_Bioorg.Chem_90_103058 |
| ESTHER : Giessel_2019_Bioorg.Chem_90_103058 |
| PubMedSearch : Giessel_2019_Bioorg.Chem_90_103058 |
| PubMedID: 31212181 |
| Title : Ursolic and oleanolic acid derivatives with cholinesterase inhibiting potential - Loesche_2018_Bioorg.Chem_85_23 |
| Author(s) : Loesche A , Kowitsch A , Lucas SD , Al-Halabi Z , Sippl W , Al-Harrasi A , Csuk R |
| Ref : Bioorg Chem , 85 :23 , 2018 |
| Abstract : Loesche_2018_Bioorg.Chem_85_23 |
| ESTHER : Loesche_2018_Bioorg.Chem_85_23 |
| PubMedSearch : Loesche_2018_Bioorg.Chem_85_23 |
| PubMedID: 30599410 |
| Title : Unexpected AChE inhibitory activity of (2E)alpha,beta-unsaturated fatty acids - Loesche_2018_Bioorg.Med.Chem.Lett_28_3315 |
| Author(s) : Loesche A , Wiemann J , Al Halabi Z , Karasch J , Sippl W , Csuk R |
| Ref : Bioorganic & Medicinal Chemistry Lett , 28 :3315 , 2018 |
| Abstract : Loesche_2018_Bioorg.Med.Chem.Lett_28_3315 |
| ESTHER : Loesche_2018_Bioorg.Med.Chem.Lett_28_3315 |
| PubMedSearch : Loesche_2018_Bioorg.Med.Chem.Lett_28_3315 |
| PubMedID: 30220607 |
| Title : Piperlongumine B and analogs are promising and selective inhibitors for acetylcholinesterase - Wiemann_2017_Eur.J.Med.Chem_139_222 |
| Author(s) : Wiemann J , Karasch J , Loesche A , Heller L , Brandt W , Csuk R |
| Ref : Eur Journal of Medicinal Chemistry , 139 :222 , 2017 |
| Abstract : Wiemann_2017_Eur.J.Med.Chem_139_222 |
| ESTHER : Wiemann_2017_Eur.J.Med.Chem_139_222 |
| PubMedSearch : Wiemann_2017_Eur.J.Med.Chem_139_222 |
| PubMedID: 28802122 |
| Title : Novel dehydroabietylamine derivatives as potent inhibitors of acetylcholinesterase - Wiemann_2017_Bioorg.Chem_74_145 |
| Author(s) : Wiemann J , Loesche A , Csuk R |
| Ref : Bioorg Chem , 74 :145 , 2017 |
| Abstract : Wiemann_2017_Bioorg.Chem_74_145 |
| ESTHER : Wiemann_2017_Bioorg.Chem_74_145 |
| PubMedSearch : Wiemann_2017_Bioorg.Chem_74_145 |
| PubMedID: 28797788 |
| Title : Amino derivatives of platanic acid act as selective and potent inhibitors of butyrylcholinesterase - Heller_2016_Eur.J.Med.Chem_126_652 |
| Author(s) : Heller L , Kahnt M , Loesche A , Grabandt P , Schwarz S , Brandt W , Csuk R |
| Ref : Eur Journal of Medicinal Chemistry , 126 :652 , 2016 |
| Abstract : Heller_2016_Eur.J.Med.Chem_126_652 |
| ESTHER : Heller_2016_Eur.J.Med.Chem_126_652 |
| PubMedSearch : Heller_2016_Eur.J.Med.Chem_126_652 |
| PubMedID: 27936444 |
| Title : Repurposing N,N'-bis-(arylamidino)-1,4-piperazinedicarboxamidines: An unexpected class of potent inhibitors of cholinesterases - Loesche_2016_Eur.J.Med.Chem_125_430 |
| Author(s) : Loesche A , Wiese J , Sommerwerk S , Simon V , Brandt W , Csuk R |
| Ref : Eur Journal of Medicinal Chemistry , 125 :430 , 2016 |
| Abstract : Loesche_2016_Eur.J.Med.Chem_125_430 |
| ESTHER : Loesche_2016_Eur.J.Med.Chem_125_430 |
| PubMedSearch : Loesche_2016_Eur.J.Med.Chem_125_430 |
| PubMedID: 27689726 |
| Title : Nizwaside: a new anticancer pregnane glycoside from the sap of Desmidorchis flava - Hussain_2015_Arch.Pharm.Res_38_2137 |
| Author(s) : Hussain H , Raees MA , Rehman NU , Al-Rawahi A , Csuk R , Khan HY , Abbas G , Al-Broumi MA , Green IR , Elyassi A , Mahmood T , Al-Harrasi A |
| Ref : Arch Pharm Res , 38 :2137 , 2015 |
| Abstract : Hussain_2015_Arch.Pharm.Res_38_2137 |
| ESTHER : Hussain_2015_Arch.Pharm.Res_38_2137 |
| PubMedSearch : Hussain_2015_Arch.Pharm.Res_38_2137 |
| PubMedID: 26335549 |
| Title : Converting maslinic acid into an effective inhibitor of acylcholinesterases - Schwarz_2015_Eur.J.Med.Chem_103_438 |
| Author(s) : Schwarz S , Loesche A , Lucas SD , Sommerwerk S , Serbian I , Siewert B , Pianowski E , Csuk R |
| Ref : Eur Journal of Medicinal Chemistry , 103 :438 , 2015 |
| Abstract : Schwarz_2015_Eur.J.Med.Chem_103_438 |
| ESTHER : Schwarz_2015_Eur.J.Med.Chem_103_438 |
| PubMedSearch : Schwarz_2015_Eur.J.Med.Chem_103_438 |
| PubMedID: 26383128 |
| Title : Allobetulin derived seco-oleananedicarboxylates act as inhibitors of acetylcholinesterase - Heller_2015_Bioorg.Med.Chem.Lett_25_2654 |
| Author(s) : Heller L , Schwarz S , Obernauer A , Csuk R |
| Ref : Bioorganic & Medicinal Chemistry Lett , 25 :2654 , 2015 |
| Abstract : Heller_2015_Bioorg.Med.Chem.Lett_25_2654 |
| ESTHER : Heller_2015_Bioorg.Med.Chem.Lett_25_2654 |
| PubMedSearch : Heller_2015_Bioorg.Med.Chem.Lett_25_2654 |
| PubMedID: 25980913 |
| Title : Microwave-assisted synthesis of novel purine nucleosides as selective cholinesterase inhibitors - Schwarz_2014_Org.Biomol.Chem_12_2446 |
| Author(s) : Schwarz S , Csuk R , Rauter AP |
| Ref : Org Biomol Chem , 12 :2446 , 2014 |
| Abstract : Schwarz_2014_Org.Biomol.Chem_12_2446 |
| ESTHER : Schwarz_2014_Org.Biomol.Chem_12_2446 |
| PubMedSearch : Schwarz_2014_Org.Biomol.Chem_12_2446 |
| PubMedID: 24604285 |
| Title : Amino derivatives of glycyrrhetinic acid as potential inhibitors of cholinesterases - Schwarz_2014_Bioorg.Med.Chem_22_3370 |
| Author(s) : Schwarz S , Lucas SD , Sommerwerk S , Csuk R |
| Ref : Bioorganic & Medicinal Chemistry , 22 :3370 , 2014 |
| Abstract : Schwarz_2014_Bioorg.Med.Chem_22_3370 |
| ESTHER : Schwarz_2014_Bioorg.Med.Chem_22_3370 |
| PubMedSearch : Schwarz_2014_Bioorg.Med.Chem_22_3370 |
| PubMedID: 24853320 |
| Title : Gypsogenin derivatives: an unexpected class of inhibitors of cholinesterases - Heller_2014_Arch.Pharm.(Weinheim)_347_707 |
| Author(s) : Heller L , Schwarz S , Weber BA , Csuk R |
| Ref : Arch Pharm (Weinheim) , 347 :707 , 2014 |
| Abstract : Heller_2014_Arch.Pharm.(Weinheim)_347_707 |
| ESTHER : Heller_2014_Arch.Pharm.(Weinheim)_347_707 |
| PubMedSearch : Heller_2014_Arch.Pharm.(Weinheim)_347_707 |
| PubMedID: 25042600 |
| Title : Resveratrol derived butyrylcholinesterase inhibitors - Csuk_2013_Arch.Pharm.(Weinheim)_346_499 |
| Author(s) : Csuk R , Albert S , Kluge R , Strohl D |
| Ref : Arch Pharm (Weinheim) , 346 :499 , 2013 |
| Abstract : Csuk_2013_Arch.Pharm.(Weinheim)_346_499 |
| ESTHER : Csuk_2013_Arch.Pharm.(Weinheim)_346_499 |
| PubMedSearch : Csuk_2013_Arch.Pharm.(Weinheim)_346_499 |
| PubMedID: 23722618 |