Full name : DeLapp Neil W
First name : Neil W
Mail : Retired from Cardiovascular Research, Eli Lilly and Company, Indianapolis, Indiana
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Country : USA
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| Title : M1 muscarinic receptor signaling in mouse hippocampus and cortex - Porter_2002_Brain.Res_944_82 |
| Author(s) : Porter AC , Bymaster FP , DeLapp NW , Yamada M , Wess J , Hamilton SE , Nathanson NM , Felder CC |
| Ref : Brain Research , 944 :82 , 2002 |
| Abstract : Porter_2002_Brain.Res_944_82 |
| ESTHER : Porter_2002_Brain.Res_944_82 |
| PubMedSearch : Porter_2002_Brain.Res_944_82 |
| PubMedID: 12106668 |
| Title : Potent antagonism of 5-HT(3) and 5-HT(6) receptors by olanzapine - Bymaster_2001_Eur.J.Pharmacol_430_341 |
| Author(s) : Bymaster FP , Falcone JF , Bauzon D , Kennedy JS , Schenck K , DeLapp NW , Cohen ML |
| Ref : European Journal of Pharmacology , 430 :341 , 2001 |
| Abstract : Bymaster_2001_Eur.J.Pharmacol_430_341 |
| ESTHER : Bymaster_2001_Eur.J.Pharmacol_430_341 |
| PubMedSearch : Bymaster_2001_Eur.J.Pharmacol_430_341 |
| PubMedID: 11711053 |
| Title : The muscarinic receptor agonist BuTAC, a novel potential antipsychotic, does not impair learning and memory in mouse passive avoidance - Rasmussen_2001_Schizophr.Res_49_193 |
| Author(s) : Rasmussen T , Fink-Jensen A , Sauerberg P , Swedberg MD , Thomsen C , Sheardown MJ , Jeppesen L , Calligaro DO , DeLapp NW , Whitesitt CA , Ward JS , Shannon HE , Bymaster FP |
| Ref : Schizophr Res , 49 :193 , 2001 |
| Abstract : Rasmussen_2001_Schizophr.Res_49_193 |
| ESTHER : Rasmussen_2001_Schizophr.Res_49_193 |
| PubMedSearch : Rasmussen_2001_Schizophr.Res_49_193 |
| PubMedID: 11343877 |
| Title : Poster: The M1 muscarinic receptor subtype mediates Gq coupling in mouse hippocampus and pre-frontal cortex - |
| Author(s) : Porter AC , Bymaster FP , Nathanson NM , Hamilton SE , Carter PA , DeLapp NW , Felder CC |
| Ref : Life Sciences , 68 :2624 , 2001 |
| PubMedID: |
| Title : Receptor reserve of phosphoinositide-coupled muscarinic receptors in mouse hippocampus in vivo - Bymaster_2001_Brain.Res_916_165 |
| Author(s) : Bymaster FP , Carter PA , DeLapp NW , Calligaro DO , Felder CC |
| Ref : Brain Research , 916 :165 , 2001 |
| Abstract : Bymaster_2001_Brain.Res_916_165 |
| ESTHER : Bymaster_2001_Brain.Res_916_165 |
| PubMedSearch : Bymaster_2001_Brain.Res_916_165 |
| PubMedID: 11597604 |
| Title : Muscarinic receptor agonists decrease cocaine self-administration rates in drug-naive mice - Rasmussen_2000_Eur.J.Pharmacol_402_241 |
| Author(s) : Rasmussen T , Sauerberg P , Nielsen EB , Swedberg MD , Thomsen C , Sheardown MJ , Jeppesen L , Calligaro DO , DeLapp NW , Whitesitt CA , Ward JS , Shannon HE , Bymaster FP , Fink-Jensen A |
| Ref : European Journal of Pharmacology , 402 :241 , 2000 |
| Abstract : Rasmussen_2000_Eur.J.Pharmacol_402_241 |
| ESTHER : Rasmussen_2000_Eur.J.Pharmacol_402_241 |
| PubMedSearch : Rasmussen_2000_Eur.J.Pharmacol_402_241 |
| PubMedID: 10958890 |
| Title : Poster: A study of M1 receptor coupling to inhibitory G proteins in CHO cells via GTPS binding determined with anti-G protein antibodies - |
| Author(s) : DeLapp NW , McClure D , McKinzie J , Silbernagel A , Sawyer BD , Felder CC |
| Ref : Life Sciences , 64 :569 , 1999 |
| PubMedID: |
| Title : Poster: Muscarinic receptor characterization and neurochemical effects of the antipsychotic-like muscarinic agonist PTAC - |
| Author(s) : Bymaster FP , Shannon HE , DeLapp NW , Calligaro DO , Perry KW , Zhang W , Rasmussen K , Ward JS , Fink-Jensen A , Olesen PH , Rasmussen T , Sheardown M , Swedberg MD , Jeppesen L , Sauerberg P |
| Ref : Life Sciences , 64 :579 , 1999 |
| PubMedID: |
| Title : Poster: Behavioral and electrophysiological effects of the antipsychotic-like muscarinic agonist PTAC - |
| Author(s) : Shannon HE , Bymaster FP , Rasmussen K , DeLapp NW , Calligaro DO , Perry KW , Mitch CH , Ward JS , Fink-Jensen A , Olesen PH , Rasmussen T , Sheardown M , Swedberg MD , Jeppesen L , Sauerberg P |
| Ref : Life Sciences , 64 :587 , 1999 |
| PubMedID: |
| Title : Potential role of muscarinic receptors in schizophrenia - Bymaster_1999_Life.Sci_64(6-7)_527 |
| Author(s) : Bymaster FP , Shannon HE , Rasmussen K , DeLapp NW , Ward JS , Calligaro DO , Mitch CH , Whitesitt CA , Ludvigsen TS , Sheardown MJ , Swedberg MD , Rasmussen T , Olesen PH , Jeppesen L , Sauerberg P , Fink-Jensen A |
| Ref : Life Sciences , 64 :527 , 1999 |
| Abstract : Bymaster_1999_Life.Sci_64(6-7)_527 |
| ESTHER : Bymaster_1999_Life.Sci_64(6-7)_527 |
| PubMedSearch : Bymaster_1999_Life.Sci_64(6-7)_527 |
| PubMedID: 10069519 |
| Title : Poster: An anti-G protein scintillation proximity assay for M1-M5 receptor-mediated GTPS binding - |
| Author(s) : McKinzie JH , Sawyer BD , Felder CC , Falcone J , Silbernagel A , McClure D , DeLapp NW |
| Ref : Life Sciences , 64 :570 , 1999 |
| PubMedID: |
| Title : Muscarinic receptor agonists, like dopamine receptor antagonist antipsychotics, inhibit conditioned avoidance response in rats - Shannon_1999_J.Pharmacol.Exp.Ther_290_901 |
| Author(s) : Shannon HE , Hart JC , Bymaster FP , Calligaro DO , DeLapp NW , Mitch CH , Ward JS , Fink-Jensen A , Sauerberg P , Jeppesen L , Sheardown MJ , Swedberg MD |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 290 :901 , 1999 |
| Abstract : Shannon_1999_J.Pharmacol.Exp.Ther_290_901 |
| ESTHER : Shannon_1999_J.Pharmacol.Exp.Ther_290_901 |
| PubMedSearch : Shannon_1999_J.Pharmacol.Exp.Ther_290_901 |
| PubMedID: 10411607 |
| Title : Poster: Muscarinic agonists with antipsychotic-like activity. Structure activity-relationships of 1,2,5-thiadiazole analogues with functioally dopamine antagonist activity - |
| Author(s) : Sauerberg P , Jeppesen L , Olesen PH , Rasmussen T , Swedberg MD , Sheardown MJ , Fink-Jensen A , Thomsen C , Thogersen H , Ward JS , Calligaro DO , DeLapp NW , Bymaster FP , Shannon HE |
| Ref : Life Sciences , 64 :555 , 1999 |
| PubMedID: |
| Title : 1-(1,2,5-Thiadiazol-4-yl)-4-azatricyclo[2.2.1.0(2,6)]heptanes as new potent muscarinic M1 agonists: structure-activity relationship for 3-aryl-2-propyn-1-yloxy and 3-aryl-2-propyn-1-ylthio derivatives - Jeppesen_1999_J.Med.Chem_42_1999 |
| Author(s) : Jeppesen L , Olesen PH , Hansen L , Sheardown MJ , Thomsen C , Rasmussen T , Jensen AF , Christensen MS , Rimvall K , Ward JS , Whitesitt CA , Calligaro DO , Bymaster FP , DeLapp NW , Felder CC , Shannon HE , Sauerberg P |
| Ref : Journal of Medicinal Chemistry , 42 :1999 , 1999 |
| Abstract : Jeppesen_1999_J.Med.Chem_42_1999 |
| ESTHER : Jeppesen_1999_J.Med.Chem_42_1999 |
| PubMedSearch : Jeppesen_1999_J.Med.Chem_42_1999 |
| PubMedID: 10354408 |
| Title : Poster: New potent muscarinic 1,2,5-thiadiazole-azacycles and dimers hereof - |
| Author(s) : Jeppesen L , Sauerberg P , Olesen PH , Sheardown MJ , Thomsen C , Rasmussen T , Fink-Jensen A , Christensen MS , Ward JS , Whitesitt C , Calligaro DO , Bymaster FP , DeLapp NW , Felder CC , Shannon HE |
| Ref : Life Sciences , 64 :555 , 1999 |
| PubMedID: |
| Title : Poster: Reversal of pertussis toxin-induced thermal allodynia by muscarinic cholinergic agonists in mice - |
| Author(s) : Zhang L , Shannon HE , Bymaster FP , DeLapp NW , Womer DE , Mitch CH , Ward JS , Olesen PH , Sheardown M , Swedberg MD , Jeppesen L , Sauerberg P |
| Ref : Life Sciences , 64 :587 , 1999 |
| PubMedID: |
| Title : Poster: Comparison of GTP-gamma-35S and 3H-NMS binding in CHO cells stably expressing human M1-M5 muscarinic receptors using scintillation proximity assays - |
| Author(s) : Sawyer BD , Silbernagel A , McKinzie JB , Falcone J , DeLapp NW , Felder CC |
| Ref : Life Sciences , 64 :568 , 1999 |
| PubMedID: |
| Title : Muscarinic agonists with antipsychotic-like activity: structure-activity relationships of 1,2,5-thiadiazole analogues with functional dopamine antagonist activity - Sauerberg_1998_J.Med.Chem_41_4378 |
| Author(s) : Sauerberg P , Jeppesen L , Olesen PH , Rasmussen T , Swedberg MD , Sheardown MJ , Fink-Jensen A , Thomsen C , Thogersen H , Rimvall K , Ward JS , Calligaro DO , DeLapp NW , Bymaster FP , Shannon HE |
| Ref : Journal of Medicinal Chemistry , 41 :4378 , 1998 |
| Abstract : Sauerberg_1998_J.Med.Chem_41_4378 |
| ESTHER : Sauerberg_1998_J.Med.Chem_41_4378 |
| PubMedSearch : Sauerberg_1998_J.Med.Chem_41_4378 |
| PubMedID: 9784113 |
| Title : Identification of side chains on 1,2,5-thiadiazole-azacycles optimal for muscarinic m1 receptor activation - Sauerberg_1998_Bioorg.Med.Chem.Lett_8_2897 |
| Author(s) : Sauerberg P , Jeppesen L , Olesen PH , Sheardown MJ , Fink-Jensen A , Rasmussen T , Rimvall K , Shannon HE , Bymaster FP , DeLapp NW , Calligaro DO , Ward JS , Whitesitt CA , Thomsen C |
| Ref : Bioorganic & Medicinal Chemistry Lett , 8 :2897 , 1998 |
| Abstract : Sauerberg_1998_Bioorg.Med.Chem.Lett_8_2897 |
| ESTHER : Sauerberg_1998_Bioorg.Med.Chem.Lett_8_2897 |
| PubMedSearch : Sauerberg_1998_Bioorg.Med.Chem.Lett_8_2897 |
| PubMedID: 9873644 |
| Title : Conformationally constrained analogues of the muscarinic agonist 3-(4-(methylthio)-1,2,5-thiadiazol-3-yl)-1,2,5,6-tetrahydro-1-methylpyr idine. Synthesis, receptor affinity, and antinociceptive activity - Sauerberg_1998_J.Med.Chem_41_109 |
| Author(s) : Sauerberg P , Olesen PH , Sheardown MJ , Rimvall K , Thogersen H , Shannon HE , Sawyer BD , Ward JS , Bymaster FP , DeLapp NW , Calligaro DO , Swedberg MD |
| Ref : Journal of Medicinal Chemistry , 41 :109 , 1998 |
| Abstract : Sauerberg_1998_J.Med.Chem_41_109 |
| ESTHER : Sauerberg_1998_J.Med.Chem_41_109 |
| PubMedSearch : Sauerberg_1998_J.Med.Chem_41_109 |
| PubMedID: 9438027 |
| Title : Unexpected antipsychotic-like activity with the muscarinic receptor ligand (5R,6R)6-(3-propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[3.2.1]octane - Bymaster_1998_Eur.J.Pharmacol_356_109 |
| Author(s) : Bymaster FP , Shannon HE , Rasmussen K , DeLapp NW , Mitch CH , Ward JS , Calligaro DO , Ludvigsen TS , Sheardown MJ , Olesen PH , Swedberg MD , Sauerberg P , Fink-Jensen A |
| Ref : European Journal of Pharmacology , 356 :109 , 1998 |
| Abstract : Bymaster_1998_Eur.J.Pharmacol_356_109 |
| ESTHER : Bymaster_1998_Eur.J.Pharmacol_356_109 |
| PubMedSearch : Bymaster_1998_Eur.J.Pharmacol_356_109 |
| PubMedID: 9774240 |
| Title : Muscarinic agonists exhibit functional dopamine antagonism in unilaterally 6-OHDA lesioned rats - Fink-Jensen_1998_Neuroreport_9_3481 |
| Author(s) : Fink-Jensen A , Kristensen P , Shannon HE , Calligaro DO , DeLapp NW , Whitesitt CA , Ward JS , Thomsen C , Rasmusseen T , Sheardown MJ , Jeppesen L , Sauerberg P , Bymaster FP |
| Ref : Neuroreport , 9 :3481 , 1998 |
| Abstract : Fink-Jensen_1998_Neuroreport_9_3481 |
| ESTHER : Fink-Jensen_1998_Neuroreport_9_3481 |
| PubMedSearch : Fink-Jensen_1998_Neuroreport_9_3481 |
| PubMedID: 9855303 |
| Title : Poster: An immunoblot assay for PTX ADP-ribosylation of brain and spinal cord Gi\/0 proteins - |
| Author(s) : DeLapp NW , Womer DE , Shannon HE |
| Ref : Life Sciences , 60 :1179 , 1997 |
| PubMedID: |
| Title : Pharmacology of butylthio[2.2.2] (LY297802\/NNC11-1053): a novel analgesic with mixed muscarinic receptor agonist and antagonist activity - Shannon_1997_J.Pharmacol.Exp.Ther_281_884 |
| Author(s) : Shannon HE , Sheardown MJ , Bymaster FP , Calligaro DO , DeLapp NW , Gidda J , Mitch CH , Sawyer BD , Stengel PW , Ward JS , Wong DT , Olesen PH , Suzdak PD , Sauerberg P , Swedberg MD |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 281 :884 , 1997 |
| Abstract : Shannon_1997_J.Pharmacol.Exp.Ther_281_884 |
| ESTHER : Shannon_1997_J.Pharmacol.Exp.Ther_281_884 |
| PubMedSearch : Shannon_1997_J.Pharmacol.Exp.Ther_281_884 |
| PubMedID: 9152398 |
| Title : Butylthio[2.2.2] (NNC 11-1053\/LY297802): an orally active muscarinic agonist analgesic - Swedberg_1997_J.Pharmacol.Exp.Ther_281_876 |
| Author(s) : Swedberg MD , Sheardown MJ , Sauerberg P , Olesen PH , Suzdak PD , Hansen KT , Bymaster FP , Ward JS , Mitch CH , Calligaro DO , DeLapp NW , Shannon HE |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 281 :876 , 1997 |
| Abstract : Swedberg_1997_J.Pharmacol.Exp.Ther_281_876 |
| ESTHER : Swedberg_1997_J.Pharmacol.Exp.Ther_281_876 |
| PubMedSearch : Swedberg_1997_J.Pharmacol.Exp.Ther_281_876 |
| PubMedID: 9152397 |
| Title : Muscarinic agonist inhibition of rat striatal adenylate cyclase is enhanced by dopamine stimulation - DeLapp_1996_Life.Sci_59_565 |
| Author(s) : DeLapp NW , Eckols K , Shannon HE |
| Ref : Life Sciences , 59 :565 , 1996 |
| Abstract : DeLapp_1996_Life.Sci_59_565 |
| ESTHER : DeLapp_1996_Life.Sci_59_565 |
| PubMedSearch : DeLapp_1996_Life.Sci_59_565 |
| PubMedID: 8761345 |
| Title : The muscarinic M1 agonist xanomeline increases soluble amyloid precursor protein release from Chinese hamster ovary-m1 cells - Eckols_1995_Life.Sci_57_1183 |
| Author(s) : Eckols K , Bymaster FP , Mitch CH , Shannon HE , Ward JS , DeLapp NW |
| Ref : Life Sciences , 57 :1183 , 1995 |
| Abstract : Eckols_1995_Life.Sci_57_1183 |
| ESTHER : Eckols_1995_Life.Sci_57_1183 |
| PubMedSearch : Eckols_1995_Life.Sci_57_1183 |
| PubMedID: 7674807 |
| Title : Poster: The M1 agonist xanomeline potently stimulates APPs release from CHO-m1 cells - |
| Author(s) : DeLapp NW , Eckols K , Bymaster FP , Mitch CH , Shannon HE , Ward JS |
| Ref : Life Sciences , 56(11-12) :1024 , 1995 |
| PubMedID: |