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| Title : meso-Transdiene analogs inhibit vesicular monoamine transporter-2 function and methamphetamine-evoked dopamine release - Horton_2011_J.Pharmacol.Exp.Ther_336_940 |
| Author(s) : Horton DB , Siripurapu KB , Norrholm SD , Culver JP , Hojahmat M , Beckmann JS , Harrod SB , Deaciuc AG , Bardo MT , Crooks PA , Dwoskin LP |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 336 :940 , 2011 |
| Abstract : Horton_2011_J.Pharmacol.Exp.Ther_336_940 |
| ESTHER : Horton_2011_J.Pharmacol.Exp.Ther_336_940 |
| PubMedSearch : Horton_2011_J.Pharmacol.Exp.Ther_336_940 |
| PubMedID: 21177475 |
| Title : Novel bis-, tris-, and tetrakis-tertiary amino analogs as antagonists at neuronal nicotinic receptors that mediate nicotine-evoked dopamine release - Zhang_2011_Bioorg.Med.Chem.Lett_21_88 |
| Author(s) : Zhang Z , Zheng G , Pivavarchyk M , Deaciuc AG , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 21 :88 , 2011 |
| Abstract : Zhang_2011_Bioorg.Med.Chem.Lett_21_88 |
| ESTHER : Zhang_2011_Bioorg.Med.Chem.Lett_21_88 |
| PubMedSearch : Zhang_2011_Bioorg.Med.Chem.Lett_21_88 |
| PubMedID: 21147530 |
| Title : Phenyl ring-substituted lobelane analogs: inhibition of [(3)H]dopamine uptake at the vesicular monoamine transporter-2 - Nickell_2011_J.Pharmacol.Exp.Ther_336_724 |
| Author(s) : Nickell JR , Zheng G , Deaciuc AG , Crooks PA , Dwoskin LP |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 336 :724 , 2011 |
| Abstract : Nickell_2011_J.Pharmacol.Exp.Ther_336_724 |
| ESTHER : Nickell_2011_J.Pharmacol.Exp.Ther_336_724 |
| PubMedSearch : Nickell_2011_J.Pharmacol.Exp.Ther_336_724 |
| PubMedID: 20876747 |
| Title : Novel bis-2,2,6,6-tetramethylpiperidine (bis-TMP) and bis-mecamylamine antagonists at neuronal nicotinic receptors mediating nicotine-evoked dopamine release - Zhang_2010_Bioorg.Med.Chem.Lett_20_1420 |
| Author(s) : Zhang Z , Pivavarchyk M , Subramanian KL , Deaciuc AG , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 20 :1420 , 2010 |
| Abstract : Zhang_2010_Bioorg.Med.Chem.Lett_20_1420 |
| ESTHER : Zhang_2010_Bioorg.Med.Chem.Lett_20_1420 |
| PubMedSearch : Zhang_2010_Bioorg.Med.Chem.Lett_20_1420 |
| PubMedID: 20079634 |
| Title : Lobeline esters as novel ligands for neuronal nicotinic acetylcholine receptors and neurotransmitter transporters - Hojahmat_2010_Bioorg.Med.Chem_18_640 |
| Author(s) : Hojahmat M , Horton DB , Norrholm SD , Miller DK , Grinevich VP , Deaciuc AG , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry , 18 :640 , 2010 |
| Abstract : Hojahmat_2010_Bioorg.Med.Chem_18_640 |
| ESTHER : Hojahmat_2010_Bioorg.Med.Chem_18_640 |
| PubMedSearch : Hojahmat_2010_Bioorg.Med.Chem_18_640 |
| PubMedID: 20036131 |
| Title : Computational neural network analysis of the affinity of N-n-alkylnicotinium salts for the alpha4beta2* nicotinic acetylcholine receptor - Zheng_2009_J.Enzyme.Inhib.Med.Chem_24_157 |
| Author(s) : Zheng F , Zheng G , Deaciuc AG , Zhan CG , Dwoskin LP , Crooks PA |
| Ref : J Enzyme Inhib Med Chem , 24 :157 , 2009 |
| Abstract : Zheng_2009_J.Enzyme.Inhib.Med.Chem_24_157 |
| ESTHER : Zheng_2009_J.Enzyme.Inhib.Med.Chem_24_157 |
| PubMedSearch : Zheng_2009_J.Enzyme.Inhib.Med.Chem_24_157 |
| PubMedID: 18629679 |
| Title : Tetrakis-azaaromatic quaternary ammonium salts: novel subtype-selective antagonists at neuronal nicotinic receptors that mediate nicotine-evoked dopamine release - Zhang_2008_Bioorg.Med.Chem.Lett_18_5753 |
| Author(s) : Zhang Z , Zheng G , Pivavarchyk M , Deaciuc AG , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 18 :5753 , 2008 |
| Abstract : Zhang_2008_Bioorg.Med.Chem.Lett_18_5753 |
| ESTHER : Zhang_2008_Bioorg.Med.Chem.Lett_18_5753 |
| PubMedSearch : Zhang_2008_Bioorg.Med.Chem.Lett_18_5753 |
| PubMedID: 18851914 |
| Title : N,N'-Alkane-diyl-bis-3-picoliniums as nicotinic receptor antagonists: inhibition of nicotine-evoked dopamine release and hyperactivity - Dwoskin_2008_J.Pharmacol.Exp.Ther_326_563 |
| Author(s) : Dwoskin LP , Wooters TE , Sumithran SP , Siripurapu KB , Joyce BM , Lockman PR , Manda VK , Ayers JT , Zhang Z , Deaciuc AG , McIntosh JM , Crooks PA , Bardo MT |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 326 :563 , 2008 |
| Abstract : Dwoskin_2008_J.Pharmacol.Exp.Ther_326_563 |
| ESTHER : Dwoskin_2008_J.Pharmacol.Exp.Ther_326_563 |
| PubMedSearch : Dwoskin_2008_J.Pharmacol.Exp.Ther_326_563 |
| PubMedID: 18460644 |
| Title : Computational neural network analysis of the affinity of lobeline and tetrabenazine analogs for the vesicular monoamine transporter-2 - Zheng_2007_Bioorg.Med.Chem_15_2975 |
| Author(s) : Zheng F , Zheng G , Deaciuc AG , Zhan CG , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry , 15 :2975 , 2007 |
| Abstract : Zheng_2007_Bioorg.Med.Chem_15_2975 |
| ESTHER : Zheng_2007_Bioorg.Med.Chem_15_2975 |
| PubMedSearch : Zheng_2007_Bioorg.Med.Chem_15_2975 |
| PubMedID: 17331733 |
| Title : Tris-azaaromatic quaternary ammonium salts: Novel templates as antagonists at nicotinic receptors mediating nicotine-evoked dopamine release - Zheng_2007_Bioorg.Med.Chem.Lett_17_6701 |
| Author(s) : Zheng G , Sumithran SP , Deaciuc AG , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :6701 , 2007 |
| Abstract : Zheng_2007_Bioorg.Med.Chem.Lett_17_6701 |
| ESTHER : Zheng_2007_Bioorg.Med.Chem.Lett_17_6701 |
| PubMedSearch : Zheng_2007_Bioorg.Med.Chem.Lett_17_6701 |
| PubMedID: 17977723 |
| Title : Bis-azaaromatic quaternary ammonium salts as antagonists at nicotinic receptors mediating nicotine-evoked dopamine release: An investigation of binding conformation - Zheng_2007_Bioorg.Med.Chem.Lett_17_6734 |
| Author(s) : Zheng G , Zhang Z , Pivavarchyk M , Deaciuc AG , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 17 :6734 , 2007 |
| Abstract : Zheng_2007_Bioorg.Med.Chem.Lett_17_6734 |
| ESTHER : Zheng_2007_Bioorg.Med.Chem.Lett_17_6734 |
| PubMedSearch : Zheng_2007_Bioorg.Med.Chem.Lett_17_6734 |
| PubMedID: 18029180 |
| Title : Des-keto lobeline analogs with increased potency and selectivity at dopamine and serotonin transporters - Zheng_2006_Bioorg.Med.Chem.Lett_16_5018 |
| Author(s) : Zheng G , Horton DB , Deaciuc AG , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 16 :5018 , 2006 |
| Abstract : Zheng_2006_Bioorg.Med.Chem.Lett_16_5018 |
| ESTHER : Zheng_2006_Bioorg.Med.Chem.Lett_16_5018 |
| PubMedSearch : Zheng_2006_Bioorg.Med.Chem.Lett_16_5018 |
| PubMedID: 16905316 |
| Title : N, N -disubstituted piperazines and homopiperazines: synthesis and affinities at alpha4beta2* and alpha7* neuronal nicotinic acetylcholine receptors - Chen_2006_J.Enzyme.Inhib.Med.Chem_21_667 |
| Author(s) : Chen J , Deaciuc AG , Dwoskin LP , Crooks PA , Bai D |
| Ref : J Enzyme Inhib Med Chem , 21 :667 , 2006 |
| Abstract : Chen_2006_J.Enzyme.Inhib.Med.Chem_21_667 |
| ESTHER : Chen_2006_J.Enzyme.Inhib.Med.Chem_21_667 |
| PubMedSearch : Chen_2006_J.Enzyme.Inhib.Med.Chem_21_667 |
| PubMedID: 17252939 |
| Title : Identification and synthesis of novel alkaloids from the root system of Nicotiana tabacum: affinity for neuronal nicotinic acetylcholine receptors - Wei_2005_Life.Sci_78_495 |
| Author(s) : Wei X , Sumithran SP , Deaciuc AG , Burton HR , Bush LP , Dwoskin LP , Crooks PA |
| Ref : Life Sciences , 78 :495 , 2005 |
| Abstract : Wei_2005_Life.Sci_78_495 |
| ESTHER : Wei_2005_Life.Sci_78_495 |
| PubMedSearch : Wei_2005_Life.Sci_78_495 |
| PubMedID: 16197964 |
| Title : Synthesis and evaluation of a series of tropane analogues as novel vesicular monoamine transporter-2 ligands - Zheng_2005_Bioorg.Med.Chem.Lett_15_4463 |
| Author(s) : Zheng G , Dwoskin LP , Deaciuc AG , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :4463 , 2005 |
| Abstract : Zheng_2005_Bioorg.Med.Chem.Lett_15_4463 |
| ESTHER : Zheng_2005_Bioorg.Med.Chem.Lett_15_4463 |
| PubMedSearch : Zheng_2005_Bioorg.Med.Chem.Lett_15_4463 |
| PubMedID: 16112864 |
| Title : Defunctionalized lobeline analogues: structure-activity of novel ligands for the vesicular monoamine transporter - Zheng_2005_J.Med.Chem_48_5551 |
| Author(s) : Zheng G , Dwoskin LP , Deaciuc AG , Norrholm SD , Crooks PA |
| Ref : Journal of Medicinal Chemistry , 48 :5551 , 2005 |
| Abstract : Zheng_2005_J.Med.Chem_48_5551 |
| ESTHER : Zheng_2005_J.Med.Chem_48_5551 |
| PubMedSearch : Zheng_2005_J.Med.Chem_48_5551 |
| PubMedID: 16107155 |
| Title : Lobelane analogues as novel ligands for the vesicular monoamine transporter-2 - Zheng_2005_Bioorg.Med.Chem_13_3899 |
| Author(s) : Zheng G , Dwoskin LP , Deaciuc AG , Zhu J , Jones MD , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry , 13 :3899 , 2005 |
| Abstract : Zheng_2005_Bioorg.Med.Chem_13_3899 |
| ESTHER : Zheng_2005_Bioorg.Med.Chem_13_3899 |
| PubMedSearch : Zheng_2005_Bioorg.Med.Chem_13_3899 |
| PubMedID: 15911306 |
| Title : Introduction of unsaturation into the N-n-alkyl chain of the nicotinic receptor antagonists, NONI and NDNI: effect on affinity and selectivity - Sumithran_2005_AAPS.J_7_E201 |
| Author(s) : Sumithran SP , Crooks PA , Xu R , Zhu J , Deaciuc AG , Wilkins LH , Dwoskin LP |
| Ref : AAPS J , 7 :E201 , 2005 |
| Abstract : Sumithran_2005_AAPS.J_7_E201 |
| ESTHER : Sumithran_2005_AAPS.J_7_E201 |
| PubMedSearch : Sumithran_2005_AAPS.J_7_E201 |
| PubMedID: 16146341 |
| Title : Development of subtype-selective ligands as antagonists at nicotinic receptors mediating nicotine-evoked dopamine release - Crooks_2004_Bioorg.Med.Chem.Lett_14_1869 |
| Author(s) : Crooks PA , Ayers JT , Xu R , Sumithran SP , Grinevich VP , Wilkins LH , Deaciuc AG , Allen DD , Dwoskin LP |
| Ref : Bioorganic & Medicinal Chemistry Lett , 14 :1869 , 2004 |
| Abstract : Crooks_2004_Bioorg.Med.Chem.Lett_14_1869 |
| ESTHER : Crooks_2004_Bioorg.Med.Chem.Lett_14_1869 |
| PubMedSearch : Crooks_2004_Bioorg.Med.Chem.Lett_14_1869 |
| PubMedID: 15050618 |
| Title : Subtype-selective nicotinic receptor antagonists: potential as tobacco use cessation agents - Dwoskin_2004_Bioorg.Med.Chem.Lett_14_1863 |
| Author(s) : Dwoskin LP , Sumithran SP , Zhu J , Deaciuc AG , Ayers JT , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 14 :1863 , 2004 |
| Abstract : Dwoskin_2004_Bioorg.Med.Chem.Lett_14_1863 |
| ESTHER : Dwoskin_2004_Bioorg.Med.Chem.Lett_14_1863 |
| PubMedSearch : Dwoskin_2004_Bioorg.Med.Chem.Lett_14_1863 |
| PubMedID: 15050617 |
| Title : bis-Azaaromatic quaternary ammonium analogues: ligands for alpha4beta2* and alpha7* subtypes of neuronal nicotinic receptors - Ayers_2002_Bioorg.Med.Chem.Lett_12_3067 |
| Author(s) : Ayers JT , Dwoskin LP , Deaciuc AG , Grinevich VP , Zhu J , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 12 :3067 , 2002 |
| Abstract : Ayers_2002_Bioorg.Med.Chem.Lett_12_3067 |
| ESTHER : Ayers_2002_Bioorg.Med.Chem.Lett_12_3067 |
| PubMedSearch : Ayers_2002_Bioorg.Med.Chem.Lett_12_3067 |
| PubMedID: 12372503 |