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References (11)

Title : Characterization of a Selective, Reversible Inhibitor of Lysophospholipase 2 (LYPLA2) - Adibekian_2013_Probe.Report__4
Author(s) : Adibekian A , Martin BR , Chang JW , Hsu KL , Tsuboi K , Bachovchin DA , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H
Ref : Probe Report , : , 2013
Abstract : Adibekian_2013_Probe.Report__4
ESTHER : Adibekian_2013_Probe.Report__4
PubMedSearch : Adibekian_2013_Probe.Report__4
PubMedID: 24624468

Title : Characterization of a Selective, Reversible Inhibitor of Lysophospholipase 1 (LYPLA1) - Adibekian_2013_Probe.Report__3
Author(s) : Adibekian A , Martin BR , Chang JW , Hsu KL , Tsuboi K , Bachovchin DA , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H
Ref : Probe Report , : , 2013
Abstract : Adibekian_2013_Probe.Report__3
ESTHER : Adibekian_2013_Probe.Report__3
PubMedSearch : Adibekian_2013_Probe.Report__3
PubMedID: 24624465

Title : Selective inhibitors and tailored activity probes for lipoprotein-associated phospholipase A(2) - Nagano_2013_Bioorg.Med.Chem.Lett_23_839
Author(s) : Nagano JM , Hsu KL , Whitby LR , Niphakis MJ , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Hodder P , Srinivasan P , Gonzalez TD , Rosen H , Bahnson BJ , Cravatt BF
Ref : Bioorganic & Medicinal Chemistry Lett , 23 :839 , 2013
Abstract : Nagano_2013_Bioorg.Med.Chem.Lett_23_839
ESTHER : Nagano_2013_Bioorg.Med.Chem.Lett_23_839
PubMedSearch : Nagano_2013_Bioorg.Med.Chem.Lett_23_839
PubMedID: 23260346

Title : Optimization and characterization of a triazole urea inhibitor for diacylglycerol lipase beta (DAGL-beta) - Hsu_2012_Probe.Report__
Author(s) : Hsu KL , Tsuboi K , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H
Ref : Probe Report , : , 2012
Abstract : Hsu_2012_Probe.Report__
ESTHER : Hsu_2012_Probe.Report__
PubMedSearch : Hsu_2012_Probe.Report__
PubMedID: 23658950
Gene_locus related to this paper: human-ABHD6

Title : Confirming target engagement for reversible inhibitors in vivo by kinetically tuned activity-based probes - Adibekian_2012_J.Am.Chem.Soc_134_10345
Author(s) : Adibekian A , Martin BR , Chang JW , Hsu KL , Tsuboi K , Bachovchin DA , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Hodder PS , Rosen H , Cravatt BF
Ref : J Am Chem Soc , 134 :10345 , 2012
Abstract : Adibekian_2012_J.Am.Chem.Soc_134_10345
ESTHER : Adibekian_2012_J.Am.Chem.Soc_134_10345
PubMedSearch : Adibekian_2012_J.Am.Chem.Soc_134_10345
PubMedID: 22690931

Title : Optimization and characterization of a triazole urea inhibitor for alpha\/beta hydrolase domain-containing protein 11 (ABHD11): anti-probe for LYPLA1\/LYPLA2 dual inhibitor ML211 - Adibekian_2011_Probe.Report__1
Author(s) : Adibekian A , Hsu KL , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H
Ref : Probe Report , : , 2011
Abstract : Adibekian_2011_Probe.Report__1
ESTHER : Adibekian_2011_Probe.Report__1
PubMedSearch : Adibekian_2011_Probe.Report__1
PubMedID: 23658953

Title : Optimization and characterization of a triazole urea dual inhibitor for lysophospholipase 1 (LYPLA1) and lysophospholipase 2 (LYPLA2) - Adibekian_2011_Probe.Report__5
Author(s) : Adibekian A , Martin BR , Speers AE , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Cravatt BF , Hodder P , Rosen H
Ref : Probe Report , : , 2011
Abstract : Adibekian_2011_Probe.Report__5
ESTHER : Adibekian_2011_Probe.Report__5
PubMedSearch : Adibekian_2011_Probe.Report__5
PubMedID: 23658947

Title : Optimization and characterization of a triazole urea inhibitor for platelet-activating factor acetylhydrolase type 2 (PAFAH2) - Adibekian_2011_Probe.Report__2
Author(s) : Adibekian A , Hsu KL , Speers AE , Monillas ES , Brown SJ , Spicer T , Fernandez-Vega V , Ferguson J , Bahnson BJ , Cravatt BF , Hodder P , Rosen H
Ref : Probe Report , : , 2011
Abstract : Adibekian_2011_Probe.Report__2
ESTHER : Adibekian_2011_Probe.Report__2
PubMedSearch : Adibekian_2011_Probe.Report__2
PubMedID: 23658960

Title : Probe Report for RBBP9 Inhibitors - Probe 2 - Bachovchin_2010_Probe.Report.1__
Author(s) : Bachovchin DA , Speers AE , Brown SJ , Cravatt BF , Spicer T , Mercer BA , Ferguson J , Hodder P , Rosen HR
Ref : Probe Report , : , 2010
Abstract : Bachovchin_2010_Probe.Report.1__
ESTHER : Bachovchin_2010_Probe.Report.1__
PubMedSearch : Bachovchin_2010_Probe.Report.1__
PubMedID: 21433382
Gene_locus related to this paper: human-RBBP9

Title : Probe Development Efforts to Identify Novel Inhibitors of Protein Phosphatase Methylesterase-1 (PME-1) - Bachovchin_2010_Probe.Report__1
Author(s) : Bachovchin DA , Speers AE , Brown SJ , Spicer TP , Fernandez V , Ferguson J , Mohr JT , Murphy J , Fu GC , Cravatt BF , Hodder PS , Rosen H
Ref : Probe Report , : , 2010
Abstract : Bachovchin_2010_Probe.Report__1
ESTHER : Bachovchin_2010_Probe.Report__1
PubMedSearch : Bachovchin_2010_Probe.Report__1
PubMedID: 22834039

Title : Probe Report for PME-1 Inhibitors - Bachovchin_2010_Probe.Report__2
Author(s) : Bachovchin DA , Speers AE , Zuhl AM , Brown SJ , Cravatt BF , Fernandez V , Spicer T , Mercer BA , Ferguson J , Hodder P , Rosen HR
Ref : Probe Report , : , 2010
Abstract : Bachovchin_2010_Probe.Report__2
ESTHER : Bachovchin_2010_Probe.Report__2
PubMedSearch : Bachovchin_2010_Probe.Report__2
PubMedID: 21433379