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Title : Extended structure-activity relationship and pharmacokinetic investigation of (4-quinolinoyl)glycyl-2-cyanopyrrolidine inhibitors of fibroblast activation protein (FAP) - Jansen_2014_J.Med.Chem_57_3053 |
Author(s) : Jansen K , Heirbaut L , Verkerk R , Cheng JD , Joossens J , Cos P , Maes L , Lambeir AM , De Meester I , Augustyns K , Van der Veken P |
Ref : Journal of Medicinal Chemistry , 57 :3053 , 2014 |
Abstract : Jansen_2014_J.Med.Chem_57_3053 |
ESTHER : Jansen_2014_J.Med.Chem_57_3053 |
PubMedSearch : Jansen_2014_J.Med.Chem_57_3053 |
PubMedID: 24617858 |
Title : Selective Inhibitors of Fibroblast Activation Protein (FAP) with a (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine Scaffold - Jansen_2013_ACS.Med.Chem.Lett_4_491 |
Author(s) : Jansen K , Heirbaut L , Cheng JD , Joossens J , Ryabtsova O , Cos P , Maes L , Lambeir AM , De Meester I , Augustyns K , Van der Veken P |
Ref : ACS Med Chem Lett , 4 :491 , 2013 |
Abstract : Jansen_2013_ACS.Med.Chem.Lett_4_491 |
ESTHER : Jansen_2013_ACS.Med.Chem.Lett_4_491 |
PubMedSearch : Jansen_2013_ACS.Med.Chem.Lett_4_491 |
PubMedID: 24900696 |