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Author Report for: Joossens J

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    Title: Extended structure-activity relationship and pharmacokinetic investigation of (4-quinolinoyl)glycyl-2-cyanopyrrolidine inhibitors of fibroblast activation protein (FAP)
    Jansen K, Heirbaut L, Verkerk R, Cheng JD, Joossens J, Cos P, Maes L, Lambeir AM, De Meester I and Van der Veken P <1 more author(s)>
    Ref: Journal of Medicinal Chemistry, 57:3053, 2014 : PubMed

            

    Title: Selective Inhibitors of Fibroblast Activation Protein (FAP) with a (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine Scaffold
    Jansen K, Heirbaut L, Cheng JD, Joossens J, Ryabtsova O, Cos P, Maes L, Lambeir AM, De Meester I and Van der Veken P <1 more author(s)>
    Ref: ACS Med Chem Lett, 4:491, 2013 : PubMed

            

    Title: Acylated Gly-(2-cyano)pyrrolidines as inhibitors of fibroblast activation protein (FAP) and the issue of FAP/prolyl oligopeptidase (PREP)-selectivity
    Ryabtsova O, Jansen K, Van Goethem S, Joossens J, Cheng JD, Lambeir AM, De Meester I, Augustyns K, Van der Veken P
    Ref: Bioorganic & Medicinal Chemistry Lett, 22:3412, 2012 : PubMed

            

    Title: P2-substituted N-acylprolylpyrrolidine inhibitors of prolyl oligopeptidase: biochemical evaluation, binding mode determination, and assessment in a cellular model of synucleinopathy
    Van der Veken P, Fulop V, Rea D, Gerard M, Van Elzen R, Joossens J, Cheng JD, Baekelandt V, De Meester I and Augustyns K <1 more author(s)>
    Ref: Journal of Medicinal Chemistry, 55:9856, 2012 : PubMed

            

    Title: Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal?
    Van Goethem S, Matheeussen V, Joossens J, Lambeir AM, Chen X, De Meester I, Haemers A, Augustyns K, Van der Veken P
    Ref: Journal of Medicinal Chemistry, 54:5737, 2011 : PubMed

            

    Title: Inhibition of dipeptidyl-peptidase IV catalyzed peptide truncation by Vildagliptin ((2S)-{[(3-hydroxyadamantan-1-yl)amino]acetyl}-pyrrolidine-2-carbonitrile)
    Brandt I, Joossens J, Chen X, Maes MB, Scharpe S, De Meester I, Lambeir AM
    Ref: Biochemical Pharmacology, 70:134, 2005 : PubMed

            


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