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| Title : Discovery of a Selective Covalent Inhibitor of Lysophospholipase-like 1 (LYPLAL1) as a Tool to Evaluate the Role of this Serine Hydrolase in Metabolism - Ahn_2016_ACS.Chem.Biol_11_2529 |
| Author(s) : Ahn K , Boehm M , Brown MF , Calloway J , Che Y , Chen J , Fennell KF , Geoghegan KF , Gilbert AM , Gutierrez JA , Kalgutkar AS , Lanba A , Limberakis C , Magee TV , O'Doherty I , Oliver R , Pabst B , Pandit J , Parris K , Pfefferkorn JA , Rolph TP , Patel R , Schuff B , Shanmugasundaram V , Starr JT , Varghese AH , Vera NB , Vernochet C , Yan J |
| Ref : ACS Chemical Biology , 11 :2529 , 2016 |
| Abstract : Ahn_2016_ACS.Chem.Biol_11_2529 |
| ESTHER : Ahn_2016_ACS.Chem.Biol_11_2529 |
| PubMedSearch : Ahn_2016_ACS.Chem.Biol_11_2529 |
| PubMedID: 27391855 |
| Gene_locus related to this paper: human-LYPLAL1 |
| Title : Insights into the Novel Hydrolytic Mechanism of a Diethyl 2-Phenyl-2-(2-arylacetoxy)methyl Malonate Ester-Based Microsomal Triglyceride Transfer Protein (MTP) Inhibitor - Ryder_2012_Chem.Res.Toxicol_25_2138 |
| Author(s) : Ryder T , Walker GS , Goosen TC , Ruggeri RB , Conn EL , Rocke BN , Lapham K , Steppan CM , Hepworth D , Kalgutkar AS |
| Ref : Chemical Research in Toxicology , 25 :2138 , 2012 |
| Abstract : Ryder_2012_Chem.Res.Toxicol_25_2138 |
| ESTHER : Ryder_2012_Chem.Res.Toxicol_25_2138 |
| PubMedSearch : Ryder_2012_Chem.Res.Toxicol_25_2138 |
| PubMedID: 22989032 |
| Title : Utility of the carboxylesterase inhibitor bis-para-nitrophenylphosphate (BNPP) in the plasma unbound fraction determination for a hydrolytically unstable amide derivative and agonist of the TGR5 receptor - Eng_2010_Xenobiotica_40_369 |
| Author(s) : Eng H , Niosi M , McDonald TS , Wolford A , Chen Y , Simila ST , Bauman JN , Warmus J , Kalgutkar AS |
| Ref : Xenobiotica , 40 :369 , 2010 |
| Abstract : Eng_2010_Xenobiotica_40_369 |
| ESTHER : Eng_2010_Xenobiotica_40_369 |
| PubMedSearch : Eng_2010_Xenobiotica_40_369 |
| PubMedID: 20297923 |
| Title : Discovery of N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]furo[2,3-c]pyridine-5-carboxamide, an agonist of the alpha7 nicotinic acetylcholine receptor, for the potential treatment of cognitive deficits in schizophrenia: synthesis and structure--activity relationship - Wishka_2006_J.Med.Chem_49_4425 |
| Author(s) : Wishka DG , Walker DP , Yates KM , Reitz SC , Jia S , Myers JK , Olson KL , Jacobsen EJ , Wolfe ML , Groppi VE , Hanchar AJ , Thornburgh BA , Cortes-Burgos LA , Wong EH , Staton BA , Raub TJ , Higdon NR , Wall TM , Hurst RS , Walters RR , Hoffmann WE , Hajos M , Franklin S , Carey G , Gold LH , Cook KK , Sands SB , Zhao SX , Soglia JR , Kalgutkar AS , Arneric SP , Rogers BN |
| Ref : Journal of Medicinal Chemistry , 49 :4425 , 2006 |
| Abstract : Wishka_2006_J.Med.Chem_49_4425 |
| ESTHER : Wishka_2006_J.Med.Chem_49_4425 |
| PubMedSearch : Wishka_2006_J.Med.Chem_49_4425 |
| PubMedID: 16821801 |