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Title : Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer's disease therapy - Pachon-Angona_2019_J.Enzyme.Inhib.Med.Chem_34_479 |
Author(s) : Pachon-Angona I , Refouvelet B , Andrys R , Martin H , Luzet V , Iriepa I , Moraleda I , Diez-Iriepa D , Oset-Gasque MJ , Marco-Contelles J , Musilek K , Ismaili L |
Ref : J Enzyme Inhib Med Chem , 34 :479 , 2019 |
Abstract : Pachon-Angona_2019_J.Enzyme.Inhib.Med.Chem_34_479 |
ESTHER : Pachon-Angona_2019_J.Enzyme.Inhib.Med.Chem_34_479 |
PubMedSearch : Pachon-Angona_2019_J.Enzyme.Inhib.Med.Chem_34_479 |
PubMedID: 30712420 |
Title : Tetrahydropyranodiquinolin-8-amines as new, non hepatotoxic, antioxidant, and acetylcholinesterase inhibitors for Alzheimer's disease therapy - Dgachi_2016_Eur.J.Med.Chem_126_576 |
Author(s) : Dgachi Y , Sokolov O , Luzet V , Godyn J , Panek D , Bonet A , Martin H , Iriepa I , Moraleda I , Garcia-Iriepa C , Janockova J , Richert L , Soukup O , Malawska B , Chabchoub F , Marco-Contelles J , Ismaili L |
Ref : Eur Journal of Medicinal Chemistry , 126 :576 , 2016 |
Abstract : Dgachi_2016_Eur.J.Med.Chem_126_576 |
ESTHER : Dgachi_2016_Eur.J.Med.Chem_126_576 |
PubMedSearch : Dgachi_2016_Eur.J.Med.Chem_126_576 |
PubMedID: 27918993 |
Title : Synthesis and Biological Assessment of Racemic Benzochromenopyrimidinimines as Antioxidant, Cholinesterase, and Abeta1-42 Aggregation Inhibitors for Alzheimer's Disease Therapy - Dgachi_2016_ChemMedChem_11_1318 |
Author(s) : Dgachi Y , Ismaili L , Knez D , Benchekroun M , Martin H , Szalaj N , Wehle S , Bautista-Aguilera OM , Luzet V , Bonnet A , Malawska B , Gobec S , Chioua M , Decker M , Chabchoub F , Marco-Contelles J |
Ref : ChemMedChem , 11 :1318 , 2016 |
Abstract : Dgachi_2016_ChemMedChem_11_1318 |
ESTHER : Dgachi_2016_ChemMedChem_11_1318 |
PubMedSearch : Dgachi_2016_ChemMedChem_11_1318 |
PubMedID: 26804623 |
Title : Donepezil-ferulic acid hybrids as anti-Alzheimer drugs - Benchekroun_2015_Future.Med.Chem_7_15 |
Author(s) : Benchekroun M , Ismaili L , Pudlo M , Luzet V , Gharbi T , Refouvelet B , Marco-Contelles J |
Ref : Future Med Chem , 7 :15 , 2015 |
Abstract : Benchekroun_2015_Future.Med.Chem_7_15 |
ESTHER : Benchekroun_2015_Future.Med.Chem_7_15 |
PubMedSearch : Benchekroun_2015_Future.Med.Chem_7_15 |
PubMedID: 25582330 |
Title : Novel tacrine-grafted ugi adducts as multipotent anti-Alzheimer drugs: a synthetic renewal in tacrine-ferulic Acid hybrids - Benchekroun_2015_ChemMedChem_10_523 |
Author(s) : Benchekroun M , Bartolini M , Egea J , Romero A , Soriano E , Pudlo M , Luzet V , Andrisano V , Jimeno ML , Lopez MG , Wehle S , Gharbi T , Refouvelet B , de Andres L , Herrera-Arozamena C , Monti B , Bolognesi ML , Rodriguez-Franco MI , Decker M , Marco-Contelles J , Ismaili L |
Ref : ChemMedChem , 10 :523 , 2015 |
Abstract : Benchekroun_2015_ChemMedChem_10_523 |
ESTHER : Benchekroun_2015_ChemMedChem_10_523 |
PubMedSearch : Benchekroun_2015_ChemMedChem_10_523 |
PubMedID: 25537267 |
Title : Quinolone-benzylpiperidine derivatives as novel acetylcholinesterase inhibitor and antioxidant hybrids for Alzheimer Disease - Pudlo_2014_Bioorg.Med.Chem_22_2496 |
Author(s) : Pudlo M , Luzet V , Ismaili L , Tomassoli I , Iutzeler A , Refouvelet B |
Ref : Bioorganic & Medicinal Chemistry , 22 :2496 , 2014 |
Abstract : Pudlo_2014_Bioorg.Med.Chem_22_2496 |
ESTHER : Pudlo_2014_Bioorg.Med.Chem_22_2496 |
PubMedSearch : Pudlo_2014_Bioorg.Med.Chem_22_2496 |
PubMedID: 24657052 |