Report for Melchiorre C

General

Full name : Melchiorre Carlo

First name : Carlo

Mail : Department of Pharmacy and Biotechnology, Alma Mater Studiorum-University of Bologna, Via Belmeloro 6, 40126, Bologna

Zip Code :

City :

Country : Italy

Email :

Phone :

Fax :

Website :

Directory :

References (37)

Title : Multi-target Design Strategies in the Context of Alzheimer's Disease: Acetylcholinesterase Inhibition and NMDA Receptor Antagonism as the Driving Forces - Rosini_2014_Neurochem.Res_39_1914
Author(s) : Rosini M , Simoni E , Minarini A , Melchiorre C
Ref : Neurochem Res , 39 :1914 , 2014
Abstract : Rosini_2014_Neurochem.Res_39_1914
ESTHER : Rosini_2014_Neurochem.Res_39_1914
PubMedSearch : Rosini_2014_Neurochem.Res_39_1914
PubMedID: 24493627

Title : Combining galantamine and memantine in multitargeted, new chemical entities potentially useful in Alzheimer's disease - Simoni_2012_J.Med.Chem_55_9708
Author(s) : Simoni E , Daniele S , Bottegoni G , Pizzirani D , Trincavelli ML , Goldoni L , Tarozzo G , Reggiani A , Martini C , Piomelli D , Melchiorre C , Rosini M , Cavalli A
Ref : Journal of Medicinal Chemistry , 55 :9708 , 2012
Abstract : Simoni_2012_J.Med.Chem_55_9708
ESTHER : Simoni_2012_J.Med.Chem_55_9708
PubMedSearch : Simoni_2012_J.Med.Chem_55_9708
PubMedID: 23033965

Title : Exploiting the lipoic acid structure in the search for novel multitarget ligands against Alzheimer's disease - Rosini_2011_Eur.J.Med.Chem_46_5435
Author(s) : Rosini M , Simoni E , Bartolini M , Tarozzi A , Matera R , Milelli A , Hrelia P , Andrisano V , Bolognesi ML , Melchiorre C
Ref : Eur Journal of Medicinal Chemistry , 46 :5435 , 2011
Abstract : Rosini_2011_Eur.J.Med.Chem_46_5435
ESTHER : Rosini_2011_Eur.J.Med.Chem_46_5435
PubMedSearch : Rosini_2011_Eur.J.Med.Chem_46_5435
PubMedID: 21924801

Title : Tacrine derivatives and Alzheimer's disease - Tumiatti_2010_Curr.Med.Chem_17_1825
Author(s) : Tumiatti V , Minarini A , Bolognesi ML , Milelli A , Rosini M , Melchiorre C
Ref : Curr Med Chem , 17 :1825 , 2010
Abstract : Tumiatti_2010_Curr.Med.Chem_17_1825
ESTHER : Tumiatti_2010_Curr.Med.Chem_17_1825
PubMedSearch : Tumiatti_2010_Curr.Med.Chem_17_1825
PubMedID: 20345341

Title : Structure-activity relationships of memoquin: Influence of the chain chirality in the multi-target mechanism of action - Bolognesi_2009_Bioorg.Med.Chem.Lett_19_4312
Author(s) : Bolognesi ML , Bartolini M , Rosini M , Andrisano V , Melchiorre C
Ref : Bioorganic & Medicinal Chemistry Lett , 19 :4312 , 2009
Abstract : Bolognesi_2009_Bioorg.Med.Chem.Lett_19_4312
ESTHER : Bolognesi_2009_Bioorg.Med.Chem.Lett_19_4312
PubMedSearch : Bolognesi_2009_Bioorg.Med.Chem.Lett_19_4312
PubMedID: 19505825

Title : MTDL design strategy in the context of Alzheimer's disease: from lipocrine to memoquin and beyond - Bolognesi_2009_Curr.Pharm.Des_15_601
Author(s) : Bolognesi ML , Rosini M , Andrisano V , Bartolini M , Minarini A , Tumiatti V , Melchiorre C
Ref : Curr Pharm Des , 15 :601 , 2009
Abstract : Bolognesi_2009_Curr.Pharm.Des_15_601
ESTHER : Bolognesi_2009_Curr.Pharm.Des_15_601
PubMedSearch : Bolognesi_2009_Curr.Pharm.Des_15_601
PubMedID: 19199985

Title : Toward a rational design of multitarget-directed antioxidants: merging memoquin and lipoic acid molecular frameworks - Bolognesi_2009_J.Med.Chem_52_7883
Author(s) : Bolognesi ML , Cavalli A , Bergamini C , Fato R , Lenaz G , Rosini M , Bartolini M , Andrisano V , Melchiorre C
Ref : Journal of Medicinal Chemistry , 52 :7883 , 2009
Abstract : Bolognesi_2009_J.Med.Chem_52_7883
ESTHER : Bolognesi_2009_J.Med.Chem_52_7883
PubMedSearch : Bolognesi_2009_J.Med.Chem_52_7883
PubMedID: 19813747

Title : Inhibition of acetylcholinesterase, beta-amyloid aggregation, and NMDA receptors in Alzheimer's disease: a promising direction for the multi-target-directed ligands gold rush - Rosini_2008_J.Med.Chem_51_4381
Author(s) : Rosini M , Simoni E , Bartolini M , Cavalli A , Ceccarini L , Pascu N , McClymont DW , Tarozzi A , Bolognesi ML , Minarini A , Tumiatti V , Andrisano V , Mellor IR , Melchiorre C
Ref : Journal of Medicinal Chemistry , 51 :4381 , 2008
Abstract : Rosini_2008_J.Med.Chem_51_4381
ESTHER : Rosini_2008_J.Med.Chem_51_4381
PubMedSearch : Rosini_2008_J.Med.Chem_51_4381
PubMedID: 18605718

Title : Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 4. Further investigation on the inner spacer - Tumiatti_2008_J.Med.Chem_51_7308
Author(s) : Tumiatti V , Milelli A , Minarini A , Rosini M , Bolognesi ML , Micco M , Andrisano V , Bartolini M , Mancini F , Recanatini M , Cavalli A , Melchiorre C
Ref : Journal of Medicinal Chemistry , 51 :7308 , 2008
Abstract : Tumiatti_2008_J.Med.Chem_51_7308
ESTHER : Tumiatti_2008_J.Med.Chem_51_7308
PubMedSearch : Tumiatti_2008_J.Med.Chem_51_7308
PubMedID: 18954037

Title : From dual binding site acetylcholinesterase inhibitors to multi-target-directed ligands (MTDLs): a step forward in the treatment of Alzheimer's disease - Bolognesi_2008_Mini.Rev.Med.Chem_8_960
Author(s) : Bolognesi ML , Minarini A , Rosini M , Tumiatti V , Melchiorre C
Ref : Mini Rev Med Chem , 8 :960 , 2008
Abstract : Bolognesi_2008_Mini.Rev.Med.Chem_8_960
ESTHER : Bolognesi_2008_Mini.Rev.Med.Chem_8_960
PubMedSearch : Bolognesi_2008_Mini.Rev.Med.Chem_8_960
PubMedID: 18782050

Title : Multi-target-directed drug design strategy: from a dual binding site acetylcholinesterase inhibitor to a trifunctional compound against Alzheimer's disease - Bolognesi_2007_J.Med.Chem_50_6446
Author(s) : Bolognesi ML , Cavalli A , Valgimigli L , Bartolini M , Rosini M , Andrisano V , Recanatini M , Melchiorre C
Ref : Journal of Medicinal Chemistry , 50 :6446 , 2007
Abstract : Bolognesi_2007_J.Med.Chem_50_6446
ESTHER : Bolognesi_2007_J.Med.Chem_50_6446
PubMedSearch : Bolognesi_2007_J.Med.Chem_50_6446
PubMedID: 18047264

Title : Rational approach to discover multipotent anti-Alzheimer drugs - Rosini_2005_J.Med.Chem_48_360
Author(s) : Rosini M , Andrisano V , Bartolini M , Bolognesi ML , Hrelia P , Minarini A , Tarozzi A , Melchiorre C
Ref : Journal of Medicinal Chemistry , 48 :360 , 2005
Abstract : Rosini_2005_J.Med.Chem_48_360
ESTHER : Rosini_2005_J.Med.Chem_48_360
PubMedSearch : Rosini_2005_J.Med.Chem_48_360
PubMedID: 15658850

Title : Propidium-based polyamine ligands as potent inhibitors of acetylcholinesterase and acetylcholinesterase-induced amyloid-beta aggregation - Bolognesi_2005_J.Med.Chem_48_24
Author(s) : Bolognesi ML , Andrisano V , Bartolini M , Banzi R , Melchiorre C
Ref : Journal of Medicinal Chemistry , 48 :24 , 2005
Abstract : Bolognesi_2005_J.Med.Chem_48_24
ESTHER : Bolognesi_2005_J.Med.Chem_48_24
PubMedSearch : Bolognesi_2005_J.Med.Chem_48_24
PubMedID: 15633997

Title : Heterocyclic inhibitors of AChE acylation and peripheral sites - Bolognesi_2005_Farmaco_60_465
Author(s) : Bolognesi ML , Andrisano V , Bartolini M , Cavalli A , Minarini A , Recanatini M , Rosini M , Tumiatti V , Melchiorre C
Ref : Farmaco , 60 :465 , 2005
Abstract : Bolognesi_2005_Farmaco_60_465
ESTHER : Bolognesi_2005_Farmaco_60_465
PubMedSearch : Bolognesi_2005_Farmaco_60_465
PubMedID: 15878569

Title : Design, synthesis, and biological evaluation of conformationally restricted rivastigmine analogues - Bolognesi_2004_J.Med.Chem_47_5945
Author(s) : Bolognesi ML , Bartolini M , Cavalli A , Andrisano V , Rosini M , Minarini A , Melchiorre C
Ref : Journal of Medicinal Chemistry , 47 :5945 , 2004
Abstract : Bolognesi_2004_J.Med.Chem_47_5945
ESTHER : Bolognesi_2004_J.Med.Chem_47_5945
PubMedSearch : Bolognesi_2004_J.Med.Chem_47_5945
PubMedID: 15537349

Title : Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 3. Effect of replacing the inner polymethylene chain with cyclic moieties - Tumiatti_2004_J.Med.Chem_47_6490
Author(s) : Tumiatti V , Andrisano V , Banzi R , Bartolini M , Minarini A , Rosini M , Melchiorre C
Ref : Journal of Medicinal Chemistry , 47 :6490 , 2004
Abstract : Tumiatti_2004_J.Med.Chem_47_6490
ESTHER : Tumiatti_2004_J.Med.Chem_47_6490
PubMedSearch : Tumiatti_2004_J.Med.Chem_47_6490
PubMedID: 15588084

Title : Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 2. Role of the substituents on the phenyl ring and nitrogen atoms of caproctamine - Tumiatti_2003_J.Med.Chem_46_954
Author(s) : Tumiatti V , Rosini M , Bartolini M , Cavalli A , Marucci G , Andrisano V , Angeli P , Banzi R , Minarini A , Recanatini M , Melchiorre C
Ref : Journal of Medicinal Chemistry , 46 :954 , 2003
Abstract : Tumiatti_2003_J.Med.Chem_46_954
ESTHER : Tumiatti_2003_J.Med.Chem_46_954
PubMedSearch : Tumiatti_2003_J.Med.Chem_46_954
PubMedID: 12620072

Title : Polymethylene tetraamine backbone as template for the development of biologically active polyamines - Melchiorre_2003_Med.Res.Rev_23_200
Author(s) : Melchiorre C , Antonello A , Banzi R , Bolognesi ML , Minarini A , Rosini M , Tumiatti V
Ref : Med Res Rev , 23 :200 , 2003
Abstract : Melchiorre_2003_Med.Res.Rev_23_200
ESTHER : Melchiorre_2003_Med.Res.Rev_23_200
PubMedSearch : Melchiorre_2003_Med.Res.Rev_23_200
PubMedID: 12500289

Title : Structure-activity relationships of methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists. 3. Effect of inserting the tetraamine backbone into a macrocyclic structure - Bolognesi_2002_J.Med.Chem_45_3286
Author(s) : Bolognesi ML , Bixel MG , Marucci G , Bartolini M , Krauss M , Angeli P , Antonello A , Rosini M , Tumiatti V , Hucho F , Melchiorre C
Ref : Journal of Medicinal Chemistry , 45 :3286 , 2002
Abstract : Bolognesi_2002_J.Med.Chem_45_3286
ESTHER : Bolognesi_2002_J.Med.Chem_45_3286
PubMedSearch : Bolognesi_2002_J.Med.Chem_45_3286
PubMedID: 12109912

Title : Hexahydrochromeno[4,3-b]pyrrole derivatives as acetylcholinesterase inhibitors - Bolognesi_2001_J.Med.Chem_44_105
Author(s) : Bolognesi ML , Andrisano V , Bartolini M , Minarini A , Rosini M , Tumiatti V , Melchiorre C
Ref : Journal of Medicinal Chemistry , 44 :105 , 2001
Abstract : Bolognesi_2001_J.Med.Chem_44_105
ESTHER : Bolognesi_2001_J.Med.Chem_44_105
PubMedSearch : Bolognesi_2001_J.Med.Chem_44_105
PubMedID: 11141093

Title : Prejunctional muscarinic inhibitory control of acetylcholine release in the human isolated detrusor: involvement of the M4 receptor subtype - D'Agostino_2000_Br.J.Pharmacol_129_493
Author(s) : D'Agostino G , Bolognesi ML , Lucchelli A , Vicini D , Balestra B , Spelta V , Melchiorre C , Tonini M
Ref : British Journal of Pharmacology , 129 :493 , 2000
Abstract : D'Agostino_2000_Br.J.Pharmacol_129_493
ESTHER : D'Agostino_2000_Br.J.Pharmacol_129_493
PubMedSearch : D'Agostino_2000_Br.J.Pharmacol_129_493
PubMedID: 10711347

Title : [4-[[N-(3-chlorophenyl)carbamoyl]oxy]-2-butynyl]-trimethylammonium (McN-A-343)-related compounds. Effect of the butynyl chain inclusion into an aromatic unit on the potency for muscarinic receptors - Tumiatti_2000_Bioorg.Med.Chem_8_681
Author(s) : Tumiatti V , Angeli P , Andrisano V , Bolognesi ML , Cavalli A , Marucci G , Minarini A , Recanatini M , Rosini M , Melchiorre C
Ref : Bioorganic & Medicinal Chemistry , 8 :681 , 2000
Abstract : Tumiatti_2000_Bioorg.Med.Chem_8_681
ESTHER : Tumiatti_2000_Bioorg.Med.Chem_8_681
PubMedSearch : Tumiatti_2000_Bioorg.Med.Chem_8_681
PubMedID: 10819156

Title : Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists - Rosini_1999_J.Med.Chem_42_5212
Author(s) : Rosini M , Budriesi R , Bixel MG , Bolognesi ML , Chiarini A , Hucho F , Krogsgaard-Larsen P , Mellor IR , Minarini A , Tumiatti V , Usherwood PN , Melchiorre C
Ref : Journal of Medicinal Chemistry , 42 :5212 , 1999
Abstract : Rosini_1999_J.Med.Chem_42_5212
ESTHER : Rosini_1999_J.Med.Chem_42_5212
PubMedSearch : Rosini_1999_J.Med.Chem_42_5212
PubMedID: 10602706

Title : Universal template approach to drug design: polyamines as selective muscarinic receptor antagonists - Bolognesi_1998_J.Med.Chem_41_4150
Author(s) : Bolognesi ML , Minarini A , Budriesi R , Cacciaguerra S , Chiarini A , Spampinato S , Tumiatti V , Melchiorre C
Ref : Journal of Medicinal Chemistry , 41 :4150 , 1998
Abstract : Bolognesi_1998_J.Med.Chem_41_4150
ESTHER : Bolognesi_1998_J.Med.Chem_41_4150
PubMedSearch : Bolognesi_1998_J.Med.Chem_41_4150
PubMedID: 9767650

Title : Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone for Potential Use against Alzheimer's Disease -
Author(s) : Melchiorre C , Andrisano V , Bolognesi ML , Budriesi R , Cavalli A , Cavrini V , Rosini M , Tumiatti V , Recanatini M
Ref : Journal of Medicinal Chemistry , 41 :4186 , 1998
PubMedID: 9784091

Title : The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists - Melchiorre_1995_Life.Sci_56(11-12)_837
Author(s) : Melchiorre C , Minarini A , Budriesi R , Chiarini A , Spampinato S , Tumiatti V
Ref : Life Sciences , 56(11-12) :837 , 1995
Abstract : Melchiorre_1995_Life.Sci_56(11-12)_837
ESTHER : Melchiorre_1995_Life.Sci_56(11-12)_837
PubMedSearch : Melchiorre_1995_Life.Sci_56(11-12)_837
PubMedID: 10188783

Title : Poster: Tripitramine: Further pharmacological evaluation in pithed rat -
Author(s) : Cantalamessa F , Angeli P , Melchiorre C
Ref : Life Sciences , 56(11-12) :1012 , 1995
PubMedID:

Title : Binding profile of benextramine at neuropeptide Y receptor subtypes in rat brain areas - Melchiorre_1994_Eur.J.Pharmacol_265_93
Author(s) : Melchiorre C , Romualdi P , Bolognesi ML , Donatini A , Ferri S
Ref : European Journal of Pharmacology , 265 :93 , 1994
Abstract : Melchiorre_1994_Eur.J.Pharmacol_265_93
ESTHER : Melchiorre_1994_Eur.J.Pharmacol_265_93
PubMedSearch : Melchiorre_1994_Eur.J.Pharmacol_265_93
PubMedID: 7883034

Title : Polymethylene tetraamines: a novel class of cardioselective M2-antagonists -
Author(s) : Melchiorre C
Ref : Med Res Rev , 10 :327 , 1990
PubMedID: 2196404

Title : Selective antagonists provide evidence that M1 muscarinic receptors may mediate carbachol-induced drinking in the rat - Polidori_1990_Eur.J.Pharmacol_179_159
Author(s) : Polidori C , Massi M , Lambrecht G , Mutschler E , Tacke R , Melchiorre C
Ref : European Journal of Pharmacology , 179 :159 , 1990
Abstract : Polidori_1990_Eur.J.Pharmacol_179_159
ESTHER : Polidori_1990_Eur.J.Pharmacol_179_159
PubMedSearch : Polidori_1990_Eur.J.Pharmacol_179_159
PubMedID: 2364977

Title : Polymethylene tetraamines as muscarinic receptor probes - Melchiorre_1989_Trends.Pharmacol.Sci_Suppl_55
Author(s) : Melchiorre C , Minarini A , Angeli P , Giardina D , Gulini U , Quaglia W
Ref : Trends in Pharmacological Sciences , Suppl :55 , 1989
Abstract : Melchiorre_1989_Trends.Pharmacol.Sci_Suppl_55
ESTHER : Melchiorre_1989_Trends.Pharmacol.Sci_Suppl_55
PubMedSearch : Melchiorre_1989_Trends.Pharmacol.Sci_Suppl_55
PubMedID: 2694524

Title : Different muscarine receptors mediate the prejunctional inhibition of [3H]-noradrenaline release in rat or guinea-pig iris and the contraction of the rabbit iris sphincter muscle - Fuder_1989_Naunyn.Schmiedebergs.Arch.Pharmacol_340_597
Author(s) : Fuder H , Schopf J , Unckell J , Wesner MT , Melchiorre C , Tacke R , Mutschler E , Lambrecht G
Ref : Naunyn Schmiedebergs Arch Pharmacol , 340 :597 , 1989
Abstract : Fuder_1989_Naunyn.Schmiedebergs.Arch.Pharmacol_340_597
ESTHER : Fuder_1989_Naunyn.Schmiedebergs.Arch.Pharmacol_340_597
PubMedSearch : Fuder_1989_Naunyn.Schmiedebergs.Arch.Pharmacol_340_597
PubMedID: 2615852

Title : Binding and functional characterization of the cardioselective muscarinic antagonist methoctramine - Giraldo_1988_J.Pharmacol.Exp.Ther_244_1016
Author(s) : Giraldo E , Micheletti R , Montagna E , Giachetti A , Vigano MA , Ladinsky H , Melchiorre C
Ref : Journal of Pharmacology & Experimental Therapeutics , 244 :1016 , 1988
Abstract : Giraldo_1988_J.Pharmacol.Exp.Ther_244_1016
ESTHER : Giraldo_1988_J.Pharmacol.Exp.Ther_244_1016
PubMedSearch : Giraldo_1988_J.Pharmacol.Exp.Ther_244_1016
PubMedID: 3252019

Title : Methoctramine selectively blocks cardiac muscarinic M2 receptors in vivo - Wess_1988_Naunyn.Schmiedebergs.Arch.Pharmacol_338_246
Author(s) : Wess J , Angeli P , Melchiorre C , Moser U , Mutschler E , Lambrecht G
Ref : Naunyn Schmiedebergs Arch Pharmacol , 338 :246 , 1988
Abstract : Wess_1988_Naunyn.Schmiedebergs.Arch.Pharmacol_338_246
ESTHER : Wess_1988_Naunyn.Schmiedebergs.Arch.Pharmacol_338_246
PubMedSearch : Wess_1988_Naunyn.Schmiedebergs.Arch.Pharmacol_338_246
PubMedID: 3057387

Title : Selective blockade in vivo of cardiac muscarinic M2 receptors by a polymethylene tetramine, BHC-9C - Wess_1987_Eur.J.Pharmacol_142_475
Author(s) : Wess J , Lambrecht G , Mutschler E , Melchiorre C , Angeli P
Ref : European Journal of Pharmacology , 142 :475 , 1987
Abstract : Wess_1987_Eur.J.Pharmacol_142_475
ESTHER : Wess_1987_Eur.J.Pharmacol_142_475
PubMedSearch : Wess_1987_Eur.J.Pharmacol_142_475
PubMedID: 3428357

Title : Antimuscarinic action of methoctramine, a new cardioselective M-2 muscarinic receptor antagonist, alone and in combination with atropine and gallamine - Melchiorre_1987_Eur.J.Pharmacol_144_117
Author(s) : Melchiorre C , Angeli P , Lambrecht G , Mutschler E , Picchio MT , Wess J
Ref : European Journal of Pharmacology , 144 :117 , 1987
Abstract : Melchiorre_1987_Eur.J.Pharmacol_144_117
ESTHER : Melchiorre_1987_Eur.J.Pharmacol_144_117
PubMedSearch : Melchiorre_1987_Eur.J.Pharmacol_144_117
PubMedID: 3436364

Title : Potentiation and inhibition of nicotinic effects on striated muscle by the tetramine disulfide benextramine - Benfey_1980_Can.J.Physiol.Pharmacol_58_984
Author(s) : Benfey BG , Brasili L , Melchiorre C , Belleau B
Ref : Canadian Journal of Physiology & Pharmacology , 58 :984 , 1980
Abstract : Benfey_1980_Can.J.Physiol.Pharmacol_58_984
ESTHER : Benfey_1980_Can.J.Physiol.Pharmacol_58_984
PubMedSearch : Benfey_1980_Can.J.Physiol.Pharmacol_58_984
PubMedID: 6112056