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| Title : Discovery of covalent prolyl oligopeptidase boronic ester inhibitors - Plescia_2020_Eur.J.Med.Chem_185_111783 |
| Author(s) : Plescia J , Dufresne C , Janmamode N , Wahba AS , Mittermaier AK , Moitessier N |
| Ref : Eur Journal of Medicinal Chemistry , 185 :111783 , 2020 |
| Abstract : Plescia_2020_Eur.J.Med.Chem_185_111783 |
| ESTHER : Plescia_2020_Eur.J.Med.Chem_185_111783 |
| PubMedSearch : Plescia_2020_Eur.J.Med.Chem_185_111783 |
| PubMedID: 31732257 |
| Gene_locus related to this paper: human-PREP |
| Title : Integrated Synthetic, Biophysical, and Computational Investigations of Covalent Inhibitors of Prolyl Oligopeptidase and Fibroblast Activation Protein alpha - Plescia_2019_J.Med.Chem_62_7874 |
| Author(s) : Plescia J , De Cesco S , Patrascu MB , Kurian J , Di Trani J , Dufresne C , Wahba AS , Janmamode N , Mittermaier AK , Moitessier N |
| Ref : Journal of Medicinal Chemistry , 62 :7874 , 2019 |
| Abstract : Plescia_2019_J.Med.Chem_62_7874 |
| ESTHER : Plescia_2019_J.Med.Chem_62_7874 |
| PubMedSearch : Plescia_2019_J.Med.Chem_62_7874 |
| PubMedID: 31393718 |
| Title : Metabolic Instability of Cyanothiazolidine-Based Prolyl Oligopeptidase Inhibitors: a Structural Assignment Challenge and Potential Medicinal Chemistry Implications - Schiavini_2015_ChemMedChem_10_1174 |
| Author(s) : Schiavini P , Pottel J , Moitessier N , Auclair K |
| Ref : ChemMedChem , 10 :1174 , 2015 |
| Abstract : Schiavini_2015_ChemMedChem_10_1174 |
| ESTHER : Schiavini_2015_ChemMedChem_10_1174 |
| PubMedSearch : Schiavini_2015_ChemMedChem_10_1174 |
| PubMedID: 26018317 |
| Title : Virtual screening and computational optimization for the discovery of covalent prolyl oligopeptidase inhibitors with activity in human cells - De Cesco_2012_J.Med.Chem_55_6306 |
| Author(s) : De Cesco S , Deslandes S , Therrien E , Levan D , Cueto M , Schmidt R , Cantin LD , Mittermaier A , Juillerat-Jeanneret L , Moitessier N |
| Ref : Journal of Medicinal Chemistry , 55 :6306 , 2012 |
| Abstract : De Cesco_2012_J.Med.Chem_55_6306 |
| ESTHER : De Cesco_2012_J.Med.Chem_55_6306 |
| PubMedSearch : De Cesco_2012_J.Med.Chem_55_6306 |
| PubMedID: 22765237 |
| Title : Inhibitors of prolyl oligopeptidases for the therapy of human diseases: defining diseases and inhibitors - |
| Author(s) : Lawandi J , Gerber-Lemaire S , Juillerat-Jeanneret L , Moitessier N |
| Ref : Journal of Medicinal Chemistry , 53 :3423 , 2010 |
| PubMedID: 20058865 |
| Title : Constrained peptidomimetics reveal detailed geometric requirements of covalent prolyl oligopeptidase inhibitors - Lawandi_2009_J.Med.Chem_52_6672 |
| Author(s) : Lawandi J , Toumieux S , Seyer V , Campbell P , Thielges S , Juillerat-Jeanneret L , Moitessier N |
| Ref : Journal of Medicinal Chemistry , 52 :6672 , 2009 |
| Abstract : Lawandi_2009_J.Med.Chem_52_6672 |
| ESTHER : Lawandi_2009_J.Med.Chem_52_6672 |
| PubMedSearch : Lawandi_2009_J.Med.Chem_52_6672 |
| PubMedID: 19888757 |