Full name : Papke Roger Lee
First name : Roger Lee
Mail : Department of Pharmacology and Therapeutics, College of Medicine, University of Florida, PO 100267 1200 Newell Dr., 32610 Gainesville, Florida
Zip Code :
City :
Country : USA
Email : rlpapke@ufl.edu
Phone : 352-392-4712
Fax : 352-392-9696
Website : \/\/pharmacology.med.ufl.edu\/faculty\/primary-faculty-2\/roger-papke-ph-d\/
Directory :
| Title : Cholinergic Receptors and Addiction - Papke_2020_Curr.Top.Behav.Neurosci_45_123 |
| Author(s) : Papke RL , Brunzell DH , De Biasi M |
| Ref : Curr Top Behavioral Neuroscience , 45 :123 , 2020 |
| Abstract : Papke_2020_Curr.Top.Behav.Neurosci_45_123 |
| ESTHER : Papke_2020_Curr.Top.Behav.Neurosci_45_123 |
| PubMedSearch : Papke_2020_Curr.Top.Behav.Neurosci_45_123 |
| PubMedID: 32451953 |
| Title : Heteromeric Neuronal Nicotinic Acetylcholine Receptors with Mutant beta Subunits Acquire Sensitivity to alpha7-Selective Positive Allosteric Modulators - Stokes_2019_J.Pharmacol.Exp.Ther_370_252 |
| Author(s) : Stokes C , Garai S , Kulkarni AR , Cantwell LN , Noviello CM , Hibbs RE , Horenstein NA , Abboud KA , Thakur GA , Papke RL |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 370 :252 , 2019 |
| Abstract : Stokes_2019_J.Pharmacol.Exp.Ther_370_252 |
| ESTHER : Stokes_2019_J.Pharmacol.Exp.Ther_370_252 |
| PubMedSearch : Stokes_2019_J.Pharmacol.Exp.Ther_370_252 |
| PubMedID: 31175218 |
| Title : The alpha7 nicotinic receptor agonist ABT-107 protects against nigrostriatal damage in rats with unilateral 6-hydroxydopamine lesions - Bordia_2015_Exp.Neurol_263_277 |
| Author(s) : Bordia T , McGregor M , Papke RL , Decker MW , McIntosh JM , Quik M |
| Ref : Experimental Neurology , 263 :277 , 2015 |
| Abstract : Bordia_2015_Exp.Neurol_263_277 |
| ESTHER : Bordia_2015_Exp.Neurol_263_277 |
| PubMedSearch : Bordia_2015_Exp.Neurol_263_277 |
| PubMedID: 25261754 |
| Title : Merging old and new perspectives on nicotinic acetylcholine receptors - Papke_2014_Biochem.Pharmacol_89_1 |
| Author(s) : Papke RL |
| Ref : Biochemical Pharmacology , 89 :1 , 2014 |
| Abstract : Papke_2014_Biochem.Pharmacol_89_1 |
| ESTHER : Papke_2014_Biochem.Pharmacol_89_1 |
| PubMedSearch : Papke_2014_Biochem.Pharmacol_89_1 |
| PubMedID: 24486571 |
| Title : Rare Human Nicotinic Acetylcholine Receptor alpha4 Subunit (CHRNA4) Variants Affect Expression and Function of High-Affinity Nicotinic Acetylcholine Receptors - McClure-Begley_2014_J.Pharmacol.Exp.Ther_348_410 |
| Author(s) : McClure-Begley TD , Papke RL , Stone KL , Stokes C , Levy AD , Gelernter J , Xie P , Lindstrom JM , Picciotto MR |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 348 :410 , 2014 |
| Abstract : McClure-Begley_2014_J.Pharmacol.Exp.Ther_348_410 |
| ESTHER : McClure-Begley_2014_J.Pharmacol.Exp.Ther_348_410 |
| PubMedSearch : McClure-Begley_2014_J.Pharmacol.Exp.Ther_348_410 |
| PubMedID: 24385388 |
| Title : The Activity of GAT107, an Allosteric Activator and Positive Modulator of alpha7 Nicotinic Acetylcholine Receptors (nAChR), Is Regulated by Aromatic Amino Acids That Span the Subunit Interface - Papke_2014_J.Biol.Chem_289_4515 |
| Author(s) : Papke RL , Horenstein NA , Kulkarni AR , Stokes C , Corrie LW , Maeng CY , Thakur GA |
| Ref : Journal of Biological Chemistry , 289 :4515 , 2014 |
| Abstract : Papke_2014_J.Biol.Chem_289_4515 |
| ESTHER : Papke_2014_J.Biol.Chem_289_4515 |
| PubMedSearch : Papke_2014_J.Biol.Chem_289_4515 |
| PubMedID: 24362025 |
| Title : The cytisine derivatives, CC4 and CC26, reduce nicotine-induced conditioned place preference in zebrafish by acting on heteromeric neuronal nicotinic acetylcholine receptors - Ponzoni_2014_Psychopharmacology.(Berl)_231_4681 |
| Author(s) : Ponzoni L , Braida D , Pucci L , Andrea D , Fasoli F , Manfredi I , Papke RL , Stokes C , Cannazza G , Clementi F , Gotti C , Sala M |
| Ref : Psychopharmacology (Berl) , 231 :4681 , 2014 |
| Abstract : Ponzoni_2014_Psychopharmacology.(Berl)_231_4681 |
| ESTHER : Ponzoni_2014_Psychopharmacology.(Berl)_231_4681 |
| PubMedSearch : Ponzoni_2014_Psychopharmacology.(Berl)_231_4681 |
| PubMedID: 24862365 |
| Title : Differential modulation of brain nicotinic acetylcholine receptor function by cytisine, varenicline, and two novel bispidine compounds: emergent properties of a hybrid molecule - Peng_2013_J.Pharmacol.Exp.Ther_347_424 |
| Author(s) : Peng C , Stokes C , Mineur YS , Picciotto MR , Tian C , Eibl C , Tomassoli I , Guendisch D , Papke RL |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 347 :424 , 2013 |
| Abstract : Peng_2013_J.Pharmacol.Exp.Ther_347_424 |
| ESTHER : Peng_2013_J.Pharmacol.Exp.Ther_347_424 |
| PubMedSearch : Peng_2013_J.Pharmacol.Exp.Ther_347_424 |
| PubMedID: 23959137 |
| Title : Expeditious synthesis, enantiomeric resolution, and enantiomer functional characterization of (4-(4-bromophenyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide (4BP-TQS): an allosteric agonist-positive allosteric modulator of alpha7 nicotinic acetylcholine receptors - Thakur_2013_J.Med.Chem_56_8943 |
| Author(s) : Thakur GA , Kulkarni AR , Deschamps JR , Papke RL |
| Ref : Journal of Medicinal Chemistry , 56 :8943 , 2013 |
| Abstract : Thakur_2013_J.Med.Chem_56_8943 |
| ESTHER : Thakur_2013_J.Med.Chem_56_8943 |
| PubMedSearch : Thakur_2013_J.Med.Chem_56_8943 |
| PubMedID: 24090443 |
| Title : Synthesis and evaluation of a conditionally-silent agonist for the alpha7 nicotinic acetylcholine receptor - Chojnacka_2013_Bioorg.Med.Chem.Lett_23_4145 |
| Author(s) : Chojnacka K , Papke RL , Horenstein NA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 23 :4145 , 2013 |
| Abstract : Chojnacka_2013_Bioorg.Med.Chem.Lett_23_4145 |
| ESTHER : Chojnacka_2013_Bioorg.Med.Chem.Lett_23_4145 |
| PubMedSearch : Chojnacka_2013_Bioorg.Med.Chem.Lett_23_4145 |
| PubMedID: 23746476 |
| Title : Point-to-point ligand-receptor interactions across the subunit interface modulate the induction and stabilization of conformational states of alpha7 nAChR by benzylidene anabaseines - Isaacson_2013_Biochem.Pharmacol_85_817 |
| Author(s) : Isaacson MD , Horenstein NA , Stokes C , Kem WR , Papke RL |
| Ref : Biochemical Pharmacology , 85 :817 , 2013 |
| Abstract : Isaacson_2013_Biochem.Pharmacol_85_817 |
| ESTHER : Isaacson_2013_Biochem.Pharmacol_85_817 |
| PubMedSearch : Isaacson_2013_Biochem.Pharmacol_85_817 |
| PubMedID: 23352650 |
| Title : Multiple Modes of alpha7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents - Peng_2013_Mol.Pharmacol_84_459 |
| Author(s) : Peng C , Kimbrell MR , Tian C , Pack TF , Crooks PA , Fifer EK , Papke RL |
| Ref : Molecular Pharmacology , 84 :459 , 2013 |
| Abstract : Peng_2013_Mol.Pharmacol_84_459 |
| ESTHER : Peng_2013_Mol.Pharmacol_84_459 |
| PubMedSearch : Peng_2013_Mol.Pharmacol_84_459 |
| PubMedID: 23839567 |
| Title : Poster: Discovery of Lu AF58801, a novel, selective and brain penetrant positive allosteric modulator of alpha-7 nicotinic acetylcholine receptors: Attenuation of subchronic phencyclidine (PCP)-induced cognitive deficits in rats following oral administration - |
| Author(s) : Bastlund JF , Bundgaard C , Dekermendjian K , Papke RL , Redrobe JP , Frederiksen K , Eskildsen J |
| Ref : Biochemical Pharmacology , 86 :1231 , 2013 |
| PubMedID: |
| Title : alpha7beta2 nicotinic acetylcholine receptors assemble, function, and are activated primarily via their alpha7-alpha7 interfaces - Murray_2012_Mol.Pharmacol_81_175 |
| Author(s) : Murray TA , Bertrand D , Papke RL , George AA , Pantoja R , Srinivasan R , Liu Q , Wu J , Whiteaker P , Lester HA , Lukas RJ |
| Ref : Molecular Pharmacology , 81 :175 , 2012 |
| Abstract : Murray_2012_Mol.Pharmacol_81_175 |
| ESTHER : Murray_2012_Mol.Pharmacol_81_175 |
| PubMedSearch : Murray_2012_Mol.Pharmacol_81_175 |
| PubMedID: 22039094 |
| Title : Use of an alpha3beta4 nicotinic acetylcholine receptor subunit concatamer to characterize ganglionic receptor subtypes with specific subunit composition reveals species-specific pharmacologic properties - Stokes_2012_Neuropharmacol_63_538 |
| Author(s) : Stokes C , Papke RL |
| Ref : Neuropharmacology , 63 :538 , 2012 |
| Abstract : Stokes_2012_Neuropharmacol_63_538 |
| ESTHER : Stokes_2012_Neuropharmacol_63_538 |
| PubMedSearch : Stokes_2012_Neuropharmacol_63_538 |
| PubMedID: 22580377 |
| Title : The nicotinic acetylcholine receptors of zebrafish and an evaluation of pharmacological tools used for their study - Papke_2012_Biochem.Pharmacol_84_352 |
| Author(s) : Papke RL , Ono F , Stokes C , Urban JM , Boyd RT |
| Ref : Biochemical Pharmacology , 84 :352 , 2012 |
| Abstract : Papke_2012_Biochem.Pharmacol_84_352 |
| ESTHER : Papke_2012_Biochem.Pharmacol_84_352 |
| PubMedSearch : Papke_2012_Biochem.Pharmacol_84_352 |
| PubMedID: 22580045 |
| Title : Potential state-selective hydrogen bond formation can modulate activation and desensitization of the alpha7 nicotinic acetylcholine receptor - Wang_2012_J.Biol.Chem_287_21957 |
| Author(s) : Wang J , Papke RL , Stokes C , Horenstein NA |
| Ref : Journal of Biological Chemistry , 287 :21957 , 2012 |
| Abstract : Wang_2012_J.Biol.Chem_287_21957 |
| ESTHER : Wang_2012_J.Biol.Chem_287_21957 |
| PubMedSearch : Wang_2012_J.Biol.Chem_287_21957 |
| PubMedID: 22556416 |
| Title : Intrinsically low open probability of alpha7 nicotinic acetylcholine receptors can be overcome by positive allosteric modulation and serum factors leading to the generation of excitotoxic currents at physiological temperatures - Williams_2012_Mol.Pharmacol_82_746 |
| Author(s) : Williams DK , Peng C , Kimbrell MR , Papke RL |
| Ref : Molecular Pharmacology , 82 :746 , 2012 |
| Abstract : Williams_2012_Mol.Pharmacol_82_746 |
| ESTHER : Williams_2012_Mol.Pharmacol_82_746 |
| PubMedSearch : Williams_2012_Mol.Pharmacol_82_746 |
| PubMedID: 22828799 |
| Title : Positive allosteric modulators as an approach to nicotinic acetylcholine receptor-targeted therapeutics: advantages and limitations - Williams_2011_Biochem.Pharmacol_82(8)_915 |
| Author(s) : Williams DK , Wang J , Papke RL |
| Ref : Biochemical Pharmacology , 82 :915 , 2011 |
| Abstract : Williams_2011_Biochem.Pharmacol_82(8)_915 |
| ESTHER : Williams_2011_Biochem.Pharmacol_82(8)_915 |
| PubMedSearch : Williams_2011_Biochem.Pharmacol_82(8)_915 |
| PubMedID: 21575610 |
| Title : Cysteine accessibility analysis of the human alpha7 nicotinic acetylcholine receptor ligand-binding domain identifies L119 as a gatekeeper - Papke_2011_Neuropharmacol_60_159 |
| Author(s) : Papke RL , Stokes C , Williams DK , Wang J , Horenstein NA |
| Ref : Neuropharmacology , 60 :159 , 2011 |
| Abstract : Papke_2011_Neuropharmacol_60_159 |
| ESTHER : Papke_2011_Neuropharmacol_60_159 |
| PubMedSearch : Papke_2011_Neuropharmacol_60_159 |
| PubMedID: 20650284 |
| Title : Electrophysiological perspectives on the therapeutic use of nicotinic acetylcholine receptor partial agonists - Papke_2011_J.Pharmacol.Exp.Ther_337_367 |
| Author(s) : Papke RL , Trocme-Thibierge C , Guendisch D , Al Rubaiy SA , Bloom SA |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 337 :367 , 2011 |
| Abstract : Papke_2011_J.Pharmacol.Exp.Ther_337_367 |
| ESTHER : Papke_2011_J.Pharmacol.Exp.Ther_337_367 |
| PubMedSearch : Papke_2011_J.Pharmacol.Exp.Ther_337_367 |
| PubMedID: 21285282 |
| Title : The effective opening of nicotinic acetylcholine receptors with single agonist binding sites - Williams_2011_J.Gen.Physiol_137_369 |
| Author(s) : Williams DK , Stokes C , Horenstein NA , Papke RL |
| Ref : Journal of General Physiology , 137 :369 , 2011 |
| Abstract : Williams_2011_J.Gen.Physiol_137_369 |
| ESTHER : Williams_2011_J.Gen.Physiol_137_369 |
| PubMedSearch : Williams_2011_J.Gen.Physiol_137_369 |
| PubMedID: 21444659 |
| Title : Investigation of the molecular mechanism of the alpha7 nicotinic acetylcholine receptor positive allosteric modulator PNU-120596 provides evidence for two distinct desensitized states - Williams_2011_Mol.Pharmacol_80_1013 |
| Author(s) : Williams DK , Wang J , Papke RL |
| Ref : Molecular Pharmacology , 80 :1013 , 2011 |
| Abstract : Williams_2011_Mol.Pharmacol_80_1013 |
| ESTHER : Williams_2011_Mol.Pharmacol_80_1013 |
| PubMedSearch : Williams_2011_Mol.Pharmacol_80_1013 |
| PubMedID: 21885620 |
| Title : Poster: Positive and negative cooperativity of agonist and allosteric modulator binding in alpha7 nAChR: Looking for the therapeutic window - |
| Author(s) : Papke RL , Williams DK , Wang J , Horenstein NA |
| Ref : Biochemical Pharmacology , 82 :1031 , 2011 |
| PubMedID: |
| Title : Poster: The twin drug approach for novel nicotinic acetylcholine receptor (nAChR) ligands: Synthesis and structure-affinity relationships - |
| Author(s) : Tomassoli I , Eibl C , Wulf M , Papke RL , Picciotto MR , Gndisch D |
| Ref : Biochemical Pharmacology , 82 :1028 , 2011 |
| PubMedID: |
| Title : Tricks of perspective: insights and limitations to the study of macroscopic currents for the analysis of nAChR activation and desensitization - Papke_2010_J.Mol.Neurosci_40_77 |
| Author(s) : Papke RL |
| Ref : Journal of Molecular Neuroscience , 40 :77 , 2010 |
| Abstract : Papke_2010_J.Mol.Neurosci_40_77 |
| ESTHER : Papke_2010_J.Mol.Neurosci_40_77 |
| PubMedSearch : Papke_2010_J.Mol.Neurosci_40_77 |
| PubMedID: 19672724 |
| Title : alpha4beta2 Nicotinic acetylcholine receptors, willing if able - Papke_2010_Br.J.Pharmacol_160_1903 |
| Author(s) : Papke RL |
| Ref : British Journal of Pharmacology , 160 :1903 , 2010 |
| Abstract : Papke_2010_Br.J.Pharmacol_160_1903 |
| ESTHER : Papke_2010_Br.J.Pharmacol_160_1903 |
| PubMedSearch : Papke_2010_Br.J.Pharmacol_160_1903 |
| PubMedID: 20649588 |
| Title : Discovery of novel alpha7 nicotinic receptor antagonists - Peng_2010_Bioorg.Med.Chem.Lett_20_4825 |
| Author(s) : Peng Y , Zhang Q , Snyder GL , Zhu H , Yao W , Tomesch J , Papke RL , O'Callaghan JP , Welsh WJ , Wennogle LP |
| Ref : Bioorganic & Medicinal Chemistry Lett , 20 :4825 , 2010 |
| Abstract : Peng_2010_Bioorg.Med.Chem.Lett_20_4825 |
| ESTHER : Peng_2010_Bioorg.Med.Chem.Lett_20_4825 |
| PubMedSearch : Peng_2010_Bioorg.Med.Chem.Lett_20_4825 |
| PubMedID: 20638843 |
| Title : Activation and inhibition of mouse muscle and neuronal nicotinic acetylcholine receptors expressed in Xenopus oocytes - Papke_2010_J.Pharmacol.Exp.Ther_333_501 |
| Author(s) : Papke RL , Wecker L , Stitzel JA |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 333 :501 , 2010 |
| Abstract : Papke_2010_J.Pharmacol.Exp.Ther_333_501 |
| ESTHER : Papke_2010_J.Pharmacol.Exp.Ther_333_501 |
| PubMedSearch : Papke_2010_J.Pharmacol.Exp.Ther_333_501 |
| PubMedID: 20100906 |
| Title : Tethered agonist analogs as site-specific probes for domains of the human alpha7 nicotinic acetylcholine receptor that differentially regulate activation and desensitization - Wang_2010_Mol.Pharmacol_78_1012 |
| Author(s) : Wang J , Horenstein NA , Stokes C , Papke RL |
| Ref : Molecular Pharmacology , 78 :1012 , 2010 |
| Abstract : Wang_2010_Mol.Pharmacol_78_1012 |
| ESTHER : Wang_2010_Mol.Pharmacol_78_1012 |
| PubMedSearch : Wang_2010_Mol.Pharmacol_78_1012 |
| PubMedID: 20823218 |
| Title : Biochemical and functional properties of distinct nicotinic acetylcholine receptors in the superior cervical ganglion of mice with targeted deletions of nAChR subunit genes - David_2010_Eur.J.Neurosci_31_978 |
| Author(s) : David R , Ciuraszkiewicz A , Simeone X , Orr-Urtreger A , Papke RL , McIntosh JM , Huck S , Scholze P |
| Ref : European Journal of Neuroscience , 31 :978 , 2010 |
| Abstract : David_2010_Eur.J.Neurosci_31_978 |
| ESTHER : David_2010_Eur.J.Neurosci_31_978 |
| PubMedSearch : David_2010_Eur.J.Neurosci_31_978 |
| PubMedID: 20377613 |
| Title : Activation and desensitization of nicotinic alpha7-type acetylcholine receptors by benzylidene anabaseines and nicotine - Papke_2009_J.Pharmacol.Exp.Ther_329_791 |
| Author(s) : Papke RL , Kem WR , Soti F , Lopez-Hernandez GY , Horenstein NA |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 329 :791 , 2009 |
| Abstract : Papke_2009_J.Pharmacol.Exp.Ther_329_791 |
| ESTHER : Papke_2009_J.Pharmacol.Exp.Ther_329_791 |
| PubMedSearch : Papke_2009_J.Pharmacol.Exp.Ther_329_791 |
| PubMedID: 19223664 |
| Title : Cytisine-based nicotinic partial agonists as novel antidepressant compounds - Mineur_2009_J.Pharmacol.Exp.Ther_329_377 |
| Author(s) : Mineur YS , Eibl C , Young G , Kochevar C , Papke RL , Gundisch D , Picciotto MR |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 329 :377 , 2009 |
| Abstract : Mineur_2009_J.Pharmacol.Exp.Ther_329_377 |
| ESTHER : Mineur_2009_J.Pharmacol.Exp.Ther_329_377 |
| PubMedSearch : Mineur_2009_J.Pharmacol.Exp.Ther_329_377 |
| PubMedID: 19164465 |
| Title : Positive modulation of alpha7 nAChR responses in rat hippocampal interneurons to full agonists and the alpha7-selective partial agonists, 4OH-GTS-21 and S 24795 - Lopez-Hernandez_2009_Neuropharmacol_56_821 |
| Author(s) : Lopez-Hernandez GY , Thinschmidt JS , Morain P , Trocme-Thibierge C , Kem WR , Soti F , Papke RL |
| Ref : Neuropharmacology , 56 :821 , 2009 |
| Abstract : Lopez-Hernandez_2009_Neuropharmacol_56_821 |
| ESTHER : Lopez-Hernandez_2009_Neuropharmacol_56_821 |
| PubMedSearch : Lopez-Hernandez_2009_Neuropharmacol_56_821 |
| PubMedID: 19705574 |
| Title : Selective inhibition of acetylcholine-evoked responses of alpha7 neuronal nicotinic acetylcholine receptors by novel tris- and tetrakis-azaaromatic quaternary ammonium antagonists - Lopez-Hernandez_2009_Mol.Pharmacol_76_652 |
| Author(s) : Lopez-Hernandez GY , Thinschmidt JS , Zheng G , Zhang Z , Crooks PA , Dwoskin LP , Papke RL |
| Ref : Molecular Pharmacology , 76 :652 , 2009 |
| Abstract : Lopez-Hernandez_2009_Mol.Pharmacol_76_652 |
| ESTHER : Lopez-Hernandez_2009_Mol.Pharmacol_76_652 |
| PubMedSearch : Lopez-Hernandez_2009_Mol.Pharmacol_76_652 |
| PubMedID: 19556356 |
| Title : TC-5619: an alpha7 neuronal nicotinic receptor-selective agonist that demonstrates efficacy in animal models of the positive and negative symptoms and cognitive dysfunction of schizophrenia - Hauser_2009_Biochem.Pharmacol_78(7)_803 |
| Author(s) : Hauser TA , Kucinski A , Jordan KG , Gatto GJ , Wersinger SR , Hesse RA , Stachowiak EK , Stachowiak MK , Papke RL , Lippiello PM , Bencherif M |
| Ref : Biochemical Pharmacology , 78 :803 , 2009 |
| Abstract : Hauser_2009_Biochem.Pharmacol_78(7)_803 |
| ESTHER : Hauser_2009_Biochem.Pharmacol_78(7)_803 |
| PubMedSearch : Hauser_2009_Biochem.Pharmacol_78(7)_803 |
| PubMedID: 19482012 |
| Title : Extending the analysis of nicotinic receptor antagonists with the study of alpha6 nicotinic receptor subunit chimeras - Papke_2008_Neuropharmacol_54_1189 |
| Author(s) : Papke RL , Dwoskin LP , Crooks PA , Zheng G , Zhang Z , McIntosh JM , Stokes C |
| Ref : Neuropharmacology , 54 :1189 , 2008 |
| Abstract : Papke_2008_Neuropharmacol_54_1189 |
| ESTHER : Papke_2008_Neuropharmacol_54_1189 |
| PubMedSearch : Papke_2008_Neuropharmacol_54_1189 |
| PubMedID: 18448138 |
| Title : Modeling binding modes of alpha7 nicotinic acetylcholine receptor with ligands: the roles of Gln117 and other residues of the receptor in agonist binding - Huang_2008_J.Med.Chem_51_6293 |
| Author(s) : Huang X , Zheng F , Stokes C , Papke RL , Zhan CG |
| Ref : Journal of Medicinal Chemistry , 51 :6293 , 2008 |
| Abstract : Huang_2008_J.Med.Chem_51_6293 |
| ESTHER : Huang_2008_J.Med.Chem_51_6293 |
| PubMedSearch : Huang_2008_J.Med.Chem_51_6293 |
| PubMedID: 18826295 |
| Title : Multiple pharmacophores for the selective activation of nicotinic alpha7-type acetylcholine receptors - Horenstein_2008_Mol.Pharmacol_74_1496 |
| Author(s) : Horenstein NA , Leonik FM , Papke RL |
| Ref : Molecular Pharmacology , 74 :1496 , 2008 |
| Abstract : Horenstein_2008_Mol.Pharmacol_74_1496 |
| ESTHER : Horenstein_2008_Mol.Pharmacol_74_1496 |
| PubMedSearch : Horenstein_2008_Mol.Pharmacol_74_1496 |
| PubMedID: 18768388 |
| Title : Neuronal nicotinic receptors as brain targets for pharmacotherapy of drug addiction - Rahman_2008_CNS.Neurol.Disord.Drug.Targets_7_422 |
| Author(s) : Rahman S , Lopez-Hernandez GY , Corrigall WA , Papke RL |
| Ref : CNS Neurol Disord Drug Targets , 7 :422 , 2008 |
| Abstract : Rahman_2008_CNS.Neurol.Disord.Drug.Targets_7_422 |
| ESTHER : Rahman_2008_CNS.Neurol.Disord.Drug.Targets_7_422 |
| PubMedSearch : Rahman_2008_CNS.Neurol.Disord.Drug.Targets_7_422 |
| PubMedID: 19128201 |
| Title : Region-specific effects of N,N'-dodecane-1,12-diyl-bis-3-picolinium dibromide on nicotine-induced increase in extracellular dopamine in vivo - Rahman_2008_Br.J.Pharmacol_153_792 |
| Author(s) : Rahman S , Zhang Z , Papke RL , Crooks PA , Dwoskin LP , Bardo MT |
| Ref : British Journal of Pharmacology , 153 :792 , 2008 |
| Abstract : Rahman_2008_Br.J.Pharmacol_153_792 |
| ESTHER : Rahman_2008_Br.J.Pharmacol_153_792 |
| PubMedSearch : Rahman_2008_Br.J.Pharmacol_153_792 |
| PubMedID: 18059317 |
| Title : The pharmacological activity of nicotine and nornicotine on nAChRs subtypes: relevance to nicotine dependence and drug discovery - Papke_2007_J.Neurochem_101_160 |
| Author(s) : Papke RL , Dwoskin LP , Crooks PA |
| Ref : Journal of Neurochemistry , 101 :160 , 2007 |
| Abstract : Papke_2007_J.Neurochem_101_160 |
| ESTHER : Papke_2007_J.Neurochem_101_160 |
| PubMedSearch : Papke_2007_J.Neurochem_101_160 |
| PubMedID: 17241116 |
| Title : Discovery of a novel nicotinic receptor antagonist for the treatment of nicotine addiction: 1-(3-Picolinium)-12-triethylammonium-dodecane dibromide (TMPD) - Dwoskin_2007_Biochem.Pharmacol_74(8)_1271 |
| Author(s) : Dwoskin LP , Joyce BM , Zheng G , Neugebauer NM , Manda VK , Lockman P , Papke RL , Bardo MT , Crooks PA |
| Ref : Biochemical Pharmacology , 74 :1271 , 2007 |
| Abstract : Dwoskin_2007_Biochem.Pharmacol_74(8)_1271 |
| ESTHER : Dwoskin_2007_Biochem.Pharmacol_74(8)_1271 |
| PubMedSearch : Dwoskin_2007_Biochem.Pharmacol_74(8)_1271 |
| PubMedID: 17727820 |
| Title : The characterization of a novel rigid nicotine analog with alpha7-selective nAChR agonist activity and modulation of agonist properties by boron inclusion - Papke_2005_Bioorg.Med.Chem.Lett_15_3874 |
| Author(s) : Papke RL , Zheng G , Horenstein NA , Dwoskin LP , Crooks PA |
| Ref : Bioorganic & Medicinal Chemistry Lett , 15 :3874 , 2005 |
| Abstract : Papke_2005_Bioorg.Med.Chem.Lett_15_3874 |
| ESTHER : Papke_2005_Bioorg.Med.Chem.Lett_15_3874 |
| PubMedSearch : Papke_2005_Bioorg.Med.Chem.Lett_15_3874 |
| PubMedID: 16005216 |
| Title : In vivo characterization of a novel inhibitor of CNS nicotinic receptors - Damaj_2005_Eur.J.Pharmacol_521_43 |
| Author(s) : Damaj MI , Wiley JL , Martin BR , Papke RL |
| Ref : European Journal of Pharmacology , 521 :43 , 2005 |
| Abstract : Damaj_2005_Eur.J.Pharmacol_521_43 |
| ESTHER : Damaj_2005_Eur.J.Pharmacol_521_43 |
| PubMedSearch : Damaj_2005_Eur.J.Pharmacol_521_43 |
| PubMedID: 16181622 |
| Title : The effects of subunit composition on the inhibition of nicotinic receptors by the amphipathic blocker 2,2,6,6-tetramethylpiperidin-4-yl heptanoate - Papke_2005_Mol.Pharmacol_67_1977 |
| Author(s) : Papke RL , Buhr JD , Francis MM , Choi KI , Thinschmidt JS , Horenstein NA |
| Ref : Molecular Pharmacology , 67 :1977 , 2005 |
| Abstract : Papke_2005_Mol.Pharmacol_67_1977 |
| ESTHER : Papke_2005_Mol.Pharmacol_67_1977 |
| PubMedSearch : Papke_2005_Mol.Pharmacol_67_1977 |
| PubMedID: 15761116 |
| Title : Rhesus monkey alpha7 nicotinic acetylcholine receptors: comparisons to human alpha7 receptors expressed in Xenopus oocytes - Papke_2005_Eur.J.Pharmacol_524_11 |
| Author(s) : Papke RL , McCormack TJ , Jack BA , Wang D , Bugaj-Gaweda B , Schiff HC , Buhr JD , Waber AJ , Stokes C |
| Ref : European Journal of Pharmacology , 524 :11 , 2005 |
| Abstract : Papke_2005_Eur.J.Pharmacol_524_11 |
| ESTHER : Papke_2005_Eur.J.Pharmacol_524_11 |
| PubMedSearch : Papke_2005_Eur.J.Pharmacol_524_11 |
| PubMedID: 16266703 |
| Title : An alpha7 nicotinic acetylcholine receptor gain-of-function mutant that retains pharmacological fidelity - Placzek_2005_Mol.Pharmacol_68_1863 |
| Author(s) : Placzek AN , Grassi F , Meyer EM , Papke RL |
| Ref : Molecular Pharmacology , 68 :1863 , 2005 |
| Abstract : Placzek_2005_Mol.Pharmacol_68_1863 |
| ESTHER : Placzek_2005_Mol.Pharmacol_68_1863 |
| PubMedSearch : Placzek_2005_Mol.Pharmacol_68_1863 |
| PubMedID: 16186249 |
| Title : The structural basis for GTS-21 selectivity between human and rat nicotinic alpha7 receptors - Stokes_2004_Mol.Pharmacol_66_14 |
| Author(s) : Stokes C , Papke JK , Horenstein NA , Kem WR , McCormack TJ , Papke RL |
| Ref : Molecular Pharmacology , 66 :14 , 2004 |
| Abstract : Stokes_2004_Mol.Pharmacol_66_14 |
| ESTHER : Stokes_2004_Mol.Pharmacol_66_14 |
| PubMedSearch : Stokes_2004_Mol.Pharmacol_66_14 |
| PubMedID: 15213292 |
| Title : A single point mutation confers properties of the muscle-type nicotinic acetylcholine receptor to homomeric alpha7 receptors - Placzek_2004_Mol.Pharmacol_66_169 |
| Author(s) : Placzek AN , Grassi F , Papke T , Meyer EM , Papke RL |
| Ref : Molecular Pharmacology , 66 :169 , 2004 |
| Abstract : Placzek_2004_Mol.Pharmacol_66_169 |
| ESTHER : Placzek_2004_Mol.Pharmacol_66_169 |
| PubMedSearch : Placzek_2004_Mol.Pharmacol_66_169 |
| PubMedID: 15213309 |
| Title : Inhibition of wild-type and mutant neuronal nicotinic acetylcholine receptors by local anesthetics - Papke_2001_Mol.Pharmacol_60_1365 |
| Author(s) : Papke RL , Horenstein BA , Placzek AN |
| Ref : Molecular Pharmacology , 60 :1365 , 2001 |
| Abstract : Papke_2001_Mol.Pharmacol_60_1365 |
| ESTHER : Papke_2001_Mol.Pharmacol_60_1365 |
| PubMedSearch : Papke_2001_Mol.Pharmacol_60_1365 |
| PubMedID: 11723244 |
| Title : alpha7 receptor-selective agonists and modes of alpha7 receptor activation - Papke_2000_Eur.J.Pharmacol_393_179 |
| Author(s) : Papke RL , Meyer E , Nutter T , Uteshev VV |
| Ref : European Journal of Pharmacology , 393 :179 , 2000 |
| Abstract : Papke_2000_Eur.J.Pharmacol_393_179 |
| ESTHER : Papke_2000_Eur.J.Pharmacol_393_179 |
| PubMedSearch : Papke_2000_Eur.J.Pharmacol_393_179 |
| PubMedID: 10771012 |
| Title : Subtype-selective inhibition of neuronal nicotinic acetylcholine receptors by cocaine is determined by the alpha4 and beta4 subunits - Francis_2000_Mol.Pharmacol_58_109 |
| Author(s) : Francis MM , Vazquez RW , Papke RL , Oswald RE |
| Ref : Molecular Pharmacology , 58 :109 , 2000 |
| Abstract : Francis_2000_Mol.Pharmacol_58_109 |
| ESTHER : Francis_2000_Mol.Pharmacol_58_109 |
| PubMedSearch : Francis_2000_Mol.Pharmacol_58_109 |
| PubMedID: 10860932 |
| Title : The Functional Diversity of Nicotinic Receptors in the Nervous System: Perspectives on Receptor Subtypes and Receptor Specialization - |
| Author(s) : Francis MM , Papke RL |
| Ref : Handbook of Experimental Pharmacology , 144 :301 , 2000 |
| PubMedID: |
| Title : Partial agonist properties of cytisine on neuronal nicotinic receptors containing the beta 2 subunit - Papke_1994_Mol.Pharmacol_45_142 |
| Author(s) : Papke RL , Heinemann SF |
| Ref : Molecular Pharmacology , 45 :142 , 1994 |
| Abstract : Papke_1994_Mol.Pharmacol_45_142 |
| ESTHER : Papke_1994_Mol.Pharmacol_45_142 |
| PubMedSearch : Papke_1994_Mol.Pharmacol_45_142 |
| PubMedID: 8302273 |
| Title : The amino terminal half of the nicotinic beta-subunit extracellular domain regulates the kinetics of inhibition by neuronal bungarotoxin - Papke_1993_Proc.Biol.Sci_252_141 |
| Author(s) : Papke RL , Duvoisin RM , Heinemann SF |
| Ref : Proc Biol Sci , 252 :141 , 1993 |
| Abstract : Papke_1993_Proc.Biol.Sci_252_141 |
| ESTHER : Papke_1993_Proc.Biol.Sci_252_141 |
| PubMedSearch : Papke_1993_Proc.Biol.Sci_252_141 |
| PubMedID: 8391703 |
| Title : The role of the beta 4-subunit in determining the kinetic properties of rat neuronal nicotinic acetylcholine alpha 3-receptors - Papke_1991_J.Physiol_440_95 |
| Author(s) : Papke RL , Heinemann SF |
| Ref : The Journal of Physiology , 440 :95 , 1991 |
| Abstract : Papke_1991_J.Physiol_440_95 |
| ESTHER : Papke_1991_J.Physiol_440_95 |
| PubMedSearch : Papke_1991_J.Physiol_440_95 |
| PubMedID: 1725184 |
| Title : The nicotinic receptor genes - Heinemann_1991_Clin.Neuropharmacol_14 Suppl 1_S45 |
| Author(s) : Heinemann S , Boulter J , Connolly J , Deneris E , Duvoisin R , Hartley M , Hermans-Borgmeyer I , Hollmann M , O'Shea-Greenfield A , Papke RL , Rogers SW , Patrick J |
| Ref : Clinical Neuropharmacology , 14 Suppl 1 :S45 , 1991 |
| Abstract : Heinemann_1991_Clin.Neuropharmacol_14 Suppl 1_S45 |
| ESTHER : Heinemann_1991_Clin.Neuropharmacol_14 Suppl 1_S45 |
| PubMedSearch : Heinemann_1991_Clin.Neuropharmacol_14 Suppl 1_S45 |
| PubMedID: 1913709 |
| Title : Brain nicotinic receptor genes - |
| Author(s) : Heinemann SF , Boulter J , Connolly J , Deneris E , Duvoisin R , Hartley M , Hermans-Borgmeyer I , Hollmann M , O'Shea-Greenfield A , Papke RL , Rogers SW , Patrick J |
| Ref : NIDA Res Monogr , 111 :3 , 1991 |
| PubMedID: 1775184 |
| Title : The brain nicotinic acetylcholine receptor gene family - |
| Author(s) : Heinemann S , Boulter J , Deneris E , Conolly J , Duvoisin R , Papke RL , Patrick J |
| Ref : Prog Brain Res , 86 :195 , 1990 |
| PubMedID: 2087557 |
| Title : Characterization of nicotinic acetylcholine receptor channels of the TE671 human medulloblastoma clonal line - Oswald_1989_Neurosci.Lett_96_207 |
| Author(s) : Oswald RE , Papke RL , Lukas RJ |
| Ref : Neuroscience Letters , 96 :207 , 1989 |
| Abstract : Oswald_1989_Neurosci.Lett_96_207 |
| ESTHER : Oswald_1989_Neurosci.Lett_96_207 |
| PubMedSearch : Oswald_1989_Neurosci.Lett_96_207 |
| PubMedID: 2467233 |
| Title : Single-channel currents of rat neuronal nicotinic acetylcholine receptors expressed in Xenopus oocytes - Papke_1989_Neuron_3_589 |
| Author(s) : Papke RL , Boulter J , Patrick J , Heinemann S |
| Ref : Neuron , 3 :589 , 1989 |
| Abstract : Papke_1989_Neuron_3_589 |
| ESTHER : Papke_1989_Neuron_3_589 |
| PubMedSearch : Papke_1989_Neuron_3_589 |
| PubMedID: 2484342 |