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| Title : Structure-activity relationships and binding mode in the human acetylcholinesterase active site of pseudo-irreversible inhibitors related to xanthostigmine - Rizzo_2009_ChemMedChem_4_670 |
| Author(s) : Rizzo S , Cavalli A , Ceccarini L , Bartolini M , Belluti F , Bisi A , Andrisano V , Recanatini M , Rampa A |
| Ref : ChemMedChem , 4 :670 , 2009 |
| Abstract : Rizzo_2009_ChemMedChem_4_670 |
| ESTHER : Rizzo_2009_ChemMedChem_4_670 |
| PubMedSearch : Rizzo_2009_ChemMedChem_4_670 |
| PubMedID: 19222043 |
| Title : The role of Li+, Na+, and K+ in the ligand binding inside the human acetylcholinesterase gorge - Petraglio_2008_Proteins_70_779 |
| Author(s) : Petraglio G , Bartolini M , Branduardi D , Andrisano V , Recanatini M , Gervasio FL , Cavalli A , Parrinello M |
| Ref : Proteins , 70 :779 , 2008 |
| Abstract : Petraglio_2008_Proteins_70_779 |
| ESTHER : Petraglio_2008_Proteins_70_779 |
| PubMedSearch : Petraglio_2008_Proteins_70_779 |
| PubMedID: 17729290 |
| Title : Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 4. Further investigation on the inner spacer - Tumiatti_2008_J.Med.Chem_51_7308 |
| Author(s) : Tumiatti V , Milelli A , Minarini A , Rosini M , Bolognesi ML , Micco M , Andrisano V , Bartolini M , Mancini F , Recanatini M , Cavalli A , Melchiorre C |
| Ref : Journal of Medicinal Chemistry , 51 :7308 , 2008 |
| Abstract : Tumiatti_2008_J.Med.Chem_51_7308 |
| ESTHER : Tumiatti_2008_J.Med.Chem_51_7308 |
| PubMedSearch : Tumiatti_2008_J.Med.Chem_51_7308 |
| PubMedID: 18954037 |
| Title : Multi-target-directed coumarin derivatives: hAChE and BACE1 inhibitors as potential anti-Alzheimer compounds - Piazzi_2008_Bioorg.Med.Chem.Lett_18_423 |
| Author(s) : Piazzi L , Cavalli A , Colizzi F , Belluti F , Bartolini M , Mancini F , Recanatini M , Andrisano V , Rampa A |
| Ref : Bioorganic & Medicinal Chemistry Lett , 18 :423 , 2008 |
| Abstract : Piazzi_2008_Bioorg.Med.Chem.Lett_18_423 |
| ESTHER : Piazzi_2008_Bioorg.Med.Chem.Lett_18_423 |
| PubMedSearch : Piazzi_2008_Bioorg.Med.Chem.Lett_18_423 |
| PubMedID: 17998161 |
| Title : Synthesis and pharmacological profile of a series of 1-substituted-2-carbonyl derivatives of Diphenidol: novel M4 muscarinic receptor antagonists - Varoli_2008_Med.Chem_4_121 |
| Author(s) : Varoli L , Angeli P , Buccioni M , Burnelli S , Fazio N , Marucci G , Recanatini M , Spampinato S |
| Ref : Med Chem , 4 :121 , 2008 |
| Abstract : Varoli_2008_Med.Chem_4_121 |
| ESTHER : Varoli_2008_Med.Chem_4_121 |
| PubMedSearch : Varoli_2008_Med.Chem_4_121 |
| PubMedID: 18336331 |
| Title : Extensive SAR and computational studies of 3-{4-[(benzylmethylamino)methyl]phenyl}-6,7-dimethoxy-2H-2-chromenone (AP2238) derivatives - Piazzi_2007_J.Med.Chem_50_4250 |
| Author(s) : Piazzi L , Cavalli A , Belluti F , Bisi A , Gobbi S , Rizzo S , Bartolini M , Andrisano V , Recanatini M , Rampa A |
| Ref : Journal of Medicinal Chemistry , 50 :4250 , 2007 |
| Abstract : Piazzi_2007_J.Med.Chem_50_4250 |
| ESTHER : Piazzi_2007_J.Med.Chem_50_4250 |
| PubMedSearch : Piazzi_2007_J.Med.Chem_50_4250 |
| PubMedID: 17655212 |
| Title : Multi-target-directed drug design strategy: from a dual binding site acetylcholinesterase inhibitor to a trifunctional compound against Alzheimer's disease - Bolognesi_2007_J.Med.Chem_50_6446 |
| Author(s) : Bolognesi ML , Cavalli A , Valgimigli L , Bartolini M , Rosini M , Andrisano V , Recanatini M , Melchiorre C |
| Ref : Journal of Medicinal Chemistry , 50 :6446 , 2007 |
| Abstract : Bolognesi_2007_J.Med.Chem_50_6446 |
| ESTHER : Bolognesi_2007_J.Med.Chem_50_6446 |
| PubMedSearch : Bolognesi_2007_J.Med.Chem_50_6446 |
| PubMedID: 18047264 |
| Title : Cholinesterase inhibitors: SAR and enzyme inhibitory activity of 3-[omega-(benzylmethylamino)alkoxy]xanthen-9-ones - Piazzi_2007_Bioorg.Med.Chem_15_575 |
| Author(s) : Piazzi L , Belluti F , Bisi A , Gobbi S , Rizzo S , Bartolini M , Andrisano V , Recanatini M , Rampa A |
| Ref : Bioorganic & Medicinal Chemistry , 15 :575 , 2007 |
| Abstract : Piazzi_2007_Bioorg.Med.Chem_15_575 |
| ESTHER : Piazzi_2007_Bioorg.Med.Chem_15_575 |
| PubMedSearch : Piazzi_2007_Bioorg.Med.Chem_15_575 |
| PubMedID: 17008100 |
| Title : Cholinesterase inhibitors: xanthostigmine derivatives blocking the acetylcholinesterase-induced beta-amyloid aggregation - Belluti_2005_J.Med.Chem_48_4444 |
| Author(s) : Belluti F , Rampa A , Piazzi L , Bisi A , Gobbi S , Bartolini M , Andrisano V , Cavalli A , Recanatini M , Valenti P |
| Ref : Journal of Medicinal Chemistry , 48 :4444 , 2005 |
| Abstract : Belluti_2005_J.Med.Chem_48_4444 |
| ESTHER : Belluti_2005_J.Med.Chem_48_4444 |
| PubMedSearch : Belluti_2005_J.Med.Chem_48_4444 |
| PubMedID: 15974596 |
| Title : Heterocyclic inhibitors of AChE acylation and peripheral sites - Bolognesi_2005_Farmaco_60_465 |
| Author(s) : Bolognesi ML , Andrisano V , Bartolini M , Cavalli A , Minarini A , Recanatini M , Rosini M , Tumiatti V , Melchiorre C |
| Ref : Farmaco , 60 :465 , 2005 |
| Abstract : Bolognesi_2005_Farmaco_60_465 |
| ESTHER : Bolognesi_2005_Farmaco_60_465 |
| PubMedSearch : Bolognesi_2005_Farmaco_60_465 |
| PubMedID: 15878569 |
| Title : Acetylcholinesterase inhibitors as a starting point towards improved Alzheimer's disease therapeutics - Recanatini_2004_Curr.Pharm.Des_10_3157 |
| Author(s) : Recanatini M , Valenti P |
| Ref : Curr Pharm Des , 10 :3157 , 2004 |
| Abstract : Recanatini_2004_Curr.Pharm.Des_10_3157 |
| ESTHER : Recanatini_2004_Curr.Pharm.Des_10_3157 |
| PubMedSearch : Recanatini_2004_Curr.Pharm.Des_10_3157 |
| PubMedID: 15544505 |
| Title : A computational study of the binding of propidium to the peripheral anionic site of human acetylcholinesterase - Cavalli_2004_J.Med.Chem_47_3991 |
| Author(s) : Cavalli A , Bottegoni G , Raco C , De Vivo M , Recanatini M |
| Ref : Journal of Medicinal Chemistry , 47 :3991 , 2004 |
| Abstract : Cavalli_2004_J.Med.Chem_47_3991 |
| ESTHER : Cavalli_2004_J.Med.Chem_47_3991 |
| PubMedSearch : Cavalli_2004_J.Med.Chem_47_3991 |
| PubMedID: 15267237 |
| Title : Structure-activity relationships of acetylcholinesterase noncovalent inhibitors based on a polyamine backbone. 2. Role of the substituents on the phenyl ring and nitrogen atoms of caproctamine - Tumiatti_2003_J.Med.Chem_46_954 |
| Author(s) : Tumiatti V , Rosini M , Bartolini M , Cavalli A , Marucci G , Andrisano V , Angeli P , Banzi R , Minarini A , Recanatini M , Melchiorre C |
| Ref : Journal of Medicinal Chemistry , 46 :954 , 2003 |
| Abstract : Tumiatti_2003_J.Med.Chem_46_954 |
| ESTHER : Tumiatti_2003_J.Med.Chem_46_954 |
| PubMedSearch : Tumiatti_2003_J.Med.Chem_46_954 |
| PubMedID: 12620072 |
| Title : Synthesis and antagonistic activity at muscarinic receptor subtypes of some derivatives of diphenidol - Varoli_2003_Farmaco_58_651 |
| Author(s) : Varoli L , Angeli P , Buccioni M , Burnelli S , Cavalli A , Marucci G , Recanatini M |
| Ref : Farmaco , 58 :651 , 2003 |
| Abstract : Varoli_2003_Farmaco_58_651 |
| ESTHER : Varoli_2003_Farmaco_58_651 |
| PubMedSearch : Varoli_2003_Farmaco_58_651 |
| PubMedID: 13679157 |
| Title : 3-(4-[[Benzyl(methyl)amino]methyl]phenyl)-6,7-dimethoxy-2H-2-chromenone (AP2238) inhibits both acetylcholinesterase and acetylcholinesterase-induced beta-amyloid aggregation: a dual function lead for Alzheimer's disease therapy - Piazzi_2003_J.Med.Chem_46_2279 |
| Author(s) : Piazzi L , Rampa A , Bisi A , Gobbi S , Belluti F , Cavalli A , Bartolini M , Andrisano V , Valenti P , Recanatini M |
| Ref : Journal of Medicinal Chemistry , 46 :2279 , 2003 |
| Abstract : Piazzi_2003_J.Med.Chem_46_2279 |
| ESTHER : Piazzi_2003_J.Med.Chem_46_2279 |
| PubMedSearch : Piazzi_2003_J.Med.Chem_46_2279 |
| PubMedID: 12773032 |
| Title : Determination of the dissociation constants (pKa) of basic acetylcholinesterase inhibitors by reversed-phase liquid chromatography - Bartolini_2002_J.Chromatogr.A_958_59 |
| Author(s) : Bartolini M , Bertucci C , Gotti R , Tumiatti V , Cavalli A , Recanatini M , Andrisano V |
| Ref : Journal of Chromatography A , 958 :59 , 2002 |
| Abstract : Bartolini_2002_J.Chromatogr.A_958_59 |
| ESTHER : Bartolini_2002_J.Chromatogr.A_958_59 |
| PubMedSearch : Bartolini_2002_J.Chromatogr.A_958_59 |
| PubMedID: 12134831 |
| Title : Acetylcholinesterase Inhibitors: SAR and Kinetic Studies on omega-[N-Methyl-N-(3-alkylcarbamoyloxyphenyl)methyl]aminoalkoxyaryl Derivatives - Rampa_2001_J.Med.Chem_44_3810 |
| Author(s) : Rampa A , Piazzi L , Belluti F , Gobbi S , Bisi A , Bartolini M , Andrisano V , Cavrini V , Cavalli A , Recanatini M , Valenti P |
| Ref : Journal of Medicinal Chemistry , 44 :3810 , 2001 |
| Abstract : Rampa_2001_J.Med.Chem_44_3810 |
| ESTHER : Rampa_2001_J.Med.Chem_44_3810 |
| PubMedSearch : Rampa_2001_J.Med.Chem_44_3810 |
| PubMedID: 11689067 |
| Title : Synthesis and Screening for Antiacetylcholinesterase Activity of (1-Benzyl-4-oxopiperidin-3-ylidene)methylindoles and -pyrroles Related to Donepezil - Andreani_2001_J.Med.Chem_44_4011 |
| Author(s) : Andreani A , Cavalli A , Granaiola M , Guardigli M , Leoni A , Locatelli A , Morigi R , Rambaldi M , Recanatini M , Roda A |
| Ref : Journal of Medicinal Chemistry , 44 :4011 , 2001 |
| Abstract : Andreani_2001_J.Med.Chem_44_4011 |
| ESTHER : Andreani_2001_J.Med.Chem_44_4011 |
| PubMedSearch : Andreani_2001_J.Med.Chem_44_4011 |
| PubMedID: 11689088 |
| Title : SAR of 9-amino-1,2,3,4-tetrahydroacridine-based acetylcholinesterase inhibitors: synthesis, enzyme inhibitory activity, QSAR, and structure-based CoMFA of tacrine analogues - Recanatini_2000_J.Med.Chem_43_2007 |
| Author(s) : Recanatini M , Cavalli A , Belluti F , Piazzi L , Rampa A , Bisi A , Gobbi S , Valenti P , Andrisano V , Bartolini M , Cavrini V |
| Ref : Journal of Medicinal Chemistry , 43 :2007 , 2000 |
| Abstract : Recanatini_2000_J.Med.Chem_43_2007 |
| ESTHER : Recanatini_2000_J.Med.Chem_43_2007 |
| PubMedSearch : Recanatini_2000_J.Med.Chem_43_2007 |
| PubMedID: 10821713 |
| Title : [4-[[N-(3-chlorophenyl)carbamoyl]oxy]-2-butynyl]-trimethylammonium (McN-A-343)-related compounds. Effect of the butynyl chain inclusion into an aromatic unit on the potency for muscarinic receptors - Tumiatti_2000_Bioorg.Med.Chem_8_681 |
| Author(s) : Tumiatti V , Angeli P , Andrisano V , Bolognesi ML , Cavalli A , Marucci G , Minarini A , Recanatini M , Rosini M , Melchiorre C |
| Ref : Bioorganic & Medicinal Chemistry , 8 :681 , 2000 |
| Abstract : Tumiatti_2000_Bioorg.Med.Chem_8_681 |
| ESTHER : Tumiatti_2000_Bioorg.Med.Chem_8_681 |
| PubMedSearch : Tumiatti_2000_Bioorg.Med.Chem_8_681 |
| PubMedID: 10819156 |
| Title : Acetylcholinesterase inhibitors for potential use in Alzheimer's disease: molecular modeling, synthesis and kinetic evaluation of 11H-indeno-[1,2-b]-quinolin-10-ylamine derivatives - Rampa_2000_Bioorg.Med.Chem_8_497 |
| Author(s) : Rampa A , Bisi A , Belluti F , Gobbi S , Valenti P , Andrisano V , Cavrini V , Cavalli A , Recanatini M |
| Ref : Bioorganic & Medicinal Chemistry , 8 :497 , 2000 |
| Abstract : Rampa_2000_Bioorg.Med.Chem_8_497 |
| ESTHER : Rampa_2000_Bioorg.Med.Chem_8_497 |
| PubMedSearch : Rampa_2000_Bioorg.Med.Chem_8_497 |
| PubMedID: 10732965 |
| Title : Synthesis and antagonistic activity at muscarinic receptor subtypes of some 2-carbonyl derivatives of diphenidol - Varoli_1999_Bioorg.Med.Chem_7_1837 |
| Author(s) : Varoli L , Angeli P , Burnelli S , Marucci G , Recanatini M |
| Ref : Bioorganic & Medicinal Chemistry , 7 :1837 , 1999 |
| Abstract : Varoli_1999_Bioorg.Med.Chem_7_1837 |
| ESTHER : Varoli_1999_Bioorg.Med.Chem_7_1837 |
| PubMedSearch : Varoli_1999_Bioorg.Med.Chem_7_1837 |
| PubMedID: 10530931 |
| Title : Acetylcholinesterase Inhibitors: Synthesis and Structure-Activity Relationships of omega-[N-Methyl-N-(3-alkylcarbamoyloxyphenyl)- methyl]aminoalkoxyheteroaryl Derivatives - Rampa_1998_J.Med.Chem_41_3976 |
| Author(s) : Rampa A , Bisi A , Valenti P , Recanatini M , Cavalli A , Andrisano V , Cavrini V , Fin L , Buriani A , Giusti P |
| Ref : Journal of Medicinal Chemistry , 41 :3976 , 1998 |
| Abstract : Rampa_1998_J.Med.Chem_41_3976 |
| ESTHER : Rampa_1998_J.Med.Chem_41_3976 |
| PubMedSearch : Rampa_1998_J.Med.Chem_41_3976 |
| PubMedID: 9767635 |
| Title : Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone for Potential Use against Alzheimer's Disease - |
| Author(s) : Melchiorre C , Andrisano V , Bolognesi ML , Budriesi R , Cavalli A , Cavrini V , Rosini M , Tumiatti V , Recanatini M |
| Ref : Journal of Medicinal Chemistry , 41 :4186 , 1998 |
| PubMedID: 9784091 |