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| Title : DPP8 and DPP9 inhibition induces pro-caspase-1-dependent monocyte and macrophage pyroptosis - Okondo_2017_Nat.Chem.Biol_13_46 |
| Author(s) : Okondo MC , Johnson DC , Sridharan R , Go EB , Chui AJ , Wang MS , Poplawski SE , Wu W , Liu Y , Lai JH , Sanford DG , Arciprete MO , Golub TR , Bachovchin WW , Bachovchin DA |
| Ref : Nat Chemical Biology , 13 :46 , 2017 |
| Abstract : Okondo_2017_Nat.Chem.Biol_13_46 |
| ESTHER : Okondo_2017_Nat.Chem.Biol_13_46 |
| PubMedSearch : Okondo_2017_Nat.Chem.Biol_13_46 |
| PubMedID: 27820798 |
| Gene_locus related to this paper: human-DPP8 , human-DPP9 |
| Title : A high-throughput, multiplexed assay for superfamily-wide profiling of enzyme activity - Bachovchin_2014_Nat.Chem.Biol_10_656 |
| Author(s) : Bachovchin DA , Koblan LW , Wu W , Liu Y , Li Y , Zhao P , Woznica I , Shu Y , Lai JH , Poplawski SE , Kiritsy CP , Healey SE , DiMare M , Sanford DG , Munford RS , Bachovchin WW , Golub TR |
| Ref : Nat Chemical Biology , 10 :656 , 2014 |
| Abstract : Bachovchin_2014_Nat.Chem.Biol_10_656 |
| ESTHER : Bachovchin_2014_Nat.Chem.Biol_10_656 |
| PubMedSearch : Bachovchin_2014_Nat.Chem.Biol_10_656 |
| PubMedID: 24997602 |
| Gene_locus related to this paper: human-PPME1 |
| Title : Identification of selective and potent inhibitors of fibroblast activation protein and prolyl oligopeptidase - Poplawski_2013_J.Med.Chem_56_3467 |
| Author(s) : Poplawski SE , Lai JH , Li Y , Jin Z , Liu Y , Wu W , Wu Y , Zhou Y , Sudmeier JL , Sanford DG , Bachovchin WW |
| Ref : Journal of Medicinal Chemistry , 56 :3467 , 2013 |
| Abstract : Poplawski_2013_J.Med.Chem_56_3467 |
| ESTHER : Poplawski_2013_J.Med.Chem_56_3467 |
| PubMedSearch : Poplawski_2013_J.Med.Chem_56_3467 |
| PubMedID: 23594271 |
| Title : 4-Substituted boro-proline dipeptides: synthesis, characterization, and dipeptidyl peptidase IV, 8, and 9 activities - Wu_2012_Bioorg.Med.Chem.Lett_22_5536 |
| Author(s) : Wu W , Liu Y , Milo LJ, Jr. , Shu Y , Zhao P , Li Y , Woznica I , Yu G , Sanford DG , Zhou Y , Poplawski SE , Connolly BA , Sudmeier JL , Bachovchin WW , Lai JH |
| Ref : Bioorganic & Medicinal Chemistry Lett , 22 :5536 , 2012 |
| Abstract : Wu_2012_Bioorg.Med.Chem.Lett_22_5536 |
| ESTHER : Wu_2012_Bioorg.Med.Chem.Lett_22_5536 |
| PubMedSearch : Wu_2012_Bioorg.Med.Chem.Lett_22_5536 |
| PubMedID: 22853995 |
| Title : Pro-soft Val-boroPro: a strategy for enhancing in vivo performance of boronic acid inhibitors of serine proteases - Poplawski_2011_J.Med.Chem_54_2022 |
| Author(s) : Poplawski SE , Lai JH , Sanford DG , Sudmeier JL , Wu W , Bachovchin WW |
| Ref : Journal of Medicinal Chemistry , 54 :2022 , 2011 |
| Abstract : Poplawski_2011_J.Med.Chem_54_2022 |
| ESTHER : Poplawski_2011_J.Med.Chem_54_2022 |
| PubMedSearch : Poplawski_2011_J.Med.Chem_54_2022 |
| PubMedID: 21388136 |
| Title : Dipeptide boronic acid inhibitors of dipeptidyl peptidase IV: determinants of potency and in vivo efficacy and safety - Connolly_2008_J.Med.Chem_51_6005 |
| Author(s) : Connolly BA , Sanford DG , Chiluwal AK , Healey SE , Peters DE , Dimare MT , Wu W , Liu Y , Maw H , Zhou Y , Li Y , Jin Z , Sudmeier JL , Lai JH , Bachovchin WW |
| Ref : Journal of Medicinal Chemistry , 51 :6005 , 2008 |
| Abstract : Connolly_2008_J.Med.Chem_51_6005 |
| ESTHER : Connolly_2008_J.Med.Chem_51_6005 |
| PubMedSearch : Connolly_2008_J.Med.Chem_51_6005 |
| PubMedID: 18783201 |
| Title : Synthesis and characterization of constrained peptidomimetic dipeptidyl peptidase IV inhibitors: amino-lactam boroalanines - Lai_2007_J.Med.Chem_50_2391 |
| Author(s) : Lai JH , Wu W , Zhou Y , Maw HH , Liu Y , Milo LJ, Jr. , Poplawski SE , Henry GD , Sudmeier JL , Sanford DG , Bachovchin WW |
| Ref : Journal of Medicinal Chemistry , 50 :2391 , 2007 |
| Abstract : Lai_2007_J.Med.Chem_50_2391 |
| ESTHER : Lai_2007_J.Med.Chem_50_2391 |
| PubMedSearch : Lai_2007_J.Med.Chem_50_2391 |
| PubMedID: 17458948 |