Full name : Thakur Ganeshsingh A
First name : Ganeshsingh A
Mail : Dept. of Pharmaceutical Sciences and Center for Drug Discovery, Northeastern University, Boston, MA 02115
Zip Code :
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Country : USA
Email : g.thakur@neu.edu
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Directory :
| Title : Heteromeric Neuronal Nicotinic Acetylcholine Receptors with Mutant beta Subunits Acquire Sensitivity to alpha7-Selective Positive Allosteric Modulators - Stokes_2019_J.Pharmacol.Exp.Ther_370_252 |
| Author(s) : Stokes C , Garai S , Kulkarni AR , Cantwell LN , Noviello CM , Hibbs RE , Horenstein NA , Abboud KA , Thakur GA , Papke RL |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 370 :252 , 2019 |
| Abstract : Stokes_2019_J.Pharmacol.Exp.Ther_370_252 |
| ESTHER : Stokes_2019_J.Pharmacol.Exp.Ther_370_252 |
| PubMedSearch : Stokes_2019_J.Pharmacol.Exp.Ther_370_252 |
| PubMedID: 31175218 |
| Title : The Activity of GAT107, an Allosteric Activator and Positive Modulator of alpha7 Nicotinic Acetylcholine Receptors (nAChR), Is Regulated by Aromatic Amino Acids That Span the Subunit Interface - Papke_2014_J.Biol.Chem_289_4515 |
| Author(s) : Papke RL , Horenstein NA , Kulkarni AR , Stokes C , Corrie LW , Maeng CY , Thakur GA |
| Ref : Journal of Biological Chemistry , 289 :4515 , 2014 |
| Abstract : Papke_2014_J.Biol.Chem_289_4515 |
| ESTHER : Papke_2014_J.Biol.Chem_289_4515 |
| PubMedSearch : Papke_2014_J.Biol.Chem_289_4515 |
| PubMedID: 24362025 |
| Title : Novel adamantyl cannabinoids as CB1 receptor probes - Thakur_2013_J.Med.Chem_56_3904 |
| Author(s) : Thakur GA , Bajaj S , Paronis C , Peng Y , Bowman AL , Barak LS , Caron MG , Parrish D , Deschamps JR , Makriyannis A |
| Ref : Journal of Medicinal Chemistry , 56 :3904 , 2013 |
| Abstract : Thakur_2013_J.Med.Chem_56_3904 |
| ESTHER : Thakur_2013_J.Med.Chem_56_3904 |
| PubMedSearch : Thakur_2013_J.Med.Chem_56_3904 |
| PubMedID: 23621789 |
| Title : Expeditious synthesis, enantiomeric resolution, and enantiomer functional characterization of (4-(4-bromophenyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide (4BP-TQS): an allosteric agonist-positive allosteric modulator of alpha7 nicotinic acetylcholine receptors - Thakur_2013_J.Med.Chem_56_8943 |
| Author(s) : Thakur GA , Kulkarni AR , Deschamps JR , Papke RL |
| Ref : Journal of Medicinal Chemistry , 56 :8943 , 2013 |
| Abstract : Thakur_2013_J.Med.Chem_56_8943 |
| ESTHER : Thakur_2013_J.Med.Chem_56_8943 |
| PubMedSearch : Thakur_2013_J.Med.Chem_56_8943 |
| PubMedID: 24090443 |
| Title : Analysis of tolerance and behavioral\/physical dependence during chronic CB1 agonist treatment: effects of CB1 agonists, antagonists, and noncannabinoid drugs - Desai_2013_J.Pharmacol.Exp.Ther_344_319 |
| Author(s) : Desai RI , Thakur GA , Vemuri VK , Bajaj S , Makriyannis A , Bergman J |
| Ref : Journal of Pharmacology & Experimental Therapeutics , 344 :319 , 2013 |
| Abstract : Desai_2013_J.Pharmacol.Exp.Ther_344_319 |
| ESTHER : Desai_2013_J.Pharmacol.Exp.Ther_344_319 |
| PubMedSearch : Desai_2013_J.Pharmacol.Exp.Ther_344_319 |
| PubMedID: 23197773 |
| Title : The novel cannabinoid CB1 receptor neutral antagonist AM4113 suppresses food intake and food-reinforced behavior but does not induce signs of nausea in rats - Sink_2008_Neuropsychopharmacology_33_946 |
| Author(s) : Sink KS , McLaughlin PJ , Wood JA , Brown C , Fan P , Vemuri VK , Peng Y , Olszewska T , Thakur GA , Makriyannis A , Parker LA , Salamone JD |
| Ref : Neuropsychopharmacology , 33 :946 , 2008 |
| Abstract : Sink_2008_Neuropsychopharmacology_33_946 |
| ESTHER : Sink_2008_Neuropsychopharmacology_33_946 |
| PubMedSearch : Sink_2008_Neuropsychopharmacology_33_946 |
| PubMedID: 17581535 |
| Title : Cannabilactones: a novel class of CB2 selective agonists with peripheral analgesic activity - Khanolkar_2007_J.Med.Chem_50_6493 |
| Author(s) : Khanolkar AD , Lu D , Ibrahim M , Duclos RI, Jr. , Thakur GA , Malan TP, Jr. , Porreca F , Veerappan V , Tian X , George C , Parrish DA , Papahatjis DP , Makriyannis A |
| Ref : Journal of Medicinal Chemistry , 50 :6493 , 2007 |
| Abstract : Khanolkar_2007_J.Med.Chem_50_6493 |
| ESTHER : Khanolkar_2007_J.Med.Chem_50_6493 |
| PubMedSearch : Khanolkar_2007_J.Med.Chem_50_6493 |
| PubMedID: 18038967 |
| Title : Adamantyl cannabinoids: a novel class of cannabinergic ligands - Lu_2005_J.Med.Chem_48_4576 |
| Author(s) : Lu D , Meng Z , Thakur GA , Fan P , Steed J , Tartal CL , Hurst DP , Reggio PH , Deschamps JR , Parrish DA , George C , Jarbe TU , Lamb RJ , Makriyannis A |
| Ref : Journal of Medicinal Chemistry , 48 :4576 , 2005 |
| Abstract : Lu_2005_J.Med.Chem_48_4576 |
| ESTHER : Lu_2005_J.Med.Chem_48_4576 |
| PubMedSearch : Lu_2005_J.Med.Chem_48_4576 |
| PubMedID: 15999995 |