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Title : Chemical Proteomics Maps Brain Region Specific Activity of Endocannabinoid Hydrolases - Baggelaar_2017_ACS.Chem.Biol_12_852 |
Author(s) : Baggelaar MP , van Esbroeck AC , van Rooden EJ , Florea BI , Overkleeft HS , Marsicano G , Chaouloff F , van der Stelt M |
Ref : ACS Chemical Biology , 12 :852 , 2017 |
Abstract : Baggelaar_2017_ACS.Chem.Biol_12_852 |
ESTHER : Baggelaar_2017_ACS.Chem.Biol_12_852 |
PubMedSearch : Baggelaar_2017_ACS.Chem.Biol_12_852 |
PubMedID: 28106377 |
Gene_locus related to this paper: human-ABHD4 , human-ABHD6 , human-ABHD12 , human-DAGLA , human-MGLL |
Title : Discovery of Glycine Sulfonamides as Dual Inhibitors of sn-1-Diacylglycerol Lipase alpha and alpha\/beta-Hydrolase Domain 6 - Janssen_2014_J.Med.Chem_57_6610 |
Author(s) : Janssen FJ , Deng H , Baggelaar MP , Allara M , van der Wel T , den Dulk H , Ligresti A , van Esbroeck AC , McGuire R , Di Marzo V , Overkleeft HS , van der Stelt M |
Ref : Journal of Medicinal Chemistry , 57 :6610 , 2014 |
Abstract : Janssen_2014_J.Med.Chem_57_6610 |
ESTHER : Janssen_2014_J.Med.Chem_57_6610 |
PubMedSearch : Janssen_2014_J.Med.Chem_57_6610 |
PubMedID: 24988361 |
Title : Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-alpha in brain - |
Author(s) : Baggelaar MP , Janssen FJ , van Esbroeck AC , den Dulk H , Allara M , Hoogendoorn S , McGuire R , Florea BI , Meeuwenoord N , van den Elst H , van der Marel GA , Brouwer J , Di Marzo V , Overkleeft HS , van der Stelt M |
Ref : Angew Chem Int Ed Engl , 52 :12081 , 2013 |
PubMedID: 24173880 |
Gene_locus related to this paper: human-DAGLA |