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Eur Journal of Medicinal Chemistry 259: 115695
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Discovery of 1-(phenylsulfonyl)-1H-indole-based multifunctional ligands targeting cholinesterases and 5-HT(6) receptor with anti-aggregation properties against amyloid-beta and tau
Eur Journal of Medicinal Chemistry 225: 113783
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Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT6R antagonists with beta-amyloid anti-aggregation properties
Eur Journal of Medicinal Chemistry 225: 113792
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New Dual Small Molecules for Alzheimer's Disease Therapy Combining Histamine H3 Receptor (H3R) Antagonism and Calcium Channels Blockade with Additional Cholinesterase Inhibition
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Novel Multitarget-Directed Ligands Aiming at Symptoms and Causes of Alzheimer's Disease
ACS Chem Neurosci 9: 1195
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Novel multi-target-directed ligands for Alzheimer's disease: Combining cholinesterase inhibitors and 5-HT6 receptor antagonists. Design, synthesis and biological evaluation
Eur Journal of Medicinal Chemistry 124: 63