Grimshaw CE, Jennings A, Kamran R, Ueno H, Nishigaki N, Kosaka T, Tani A, Sano H, Kinugawa Y, Koumura E, Shi L, Takeuchi K (2016) <br />Trelagliptin (SYR-472, Zafatek), Novel Once-Weekly Treatment for Type 2 Diabetes, Inhibits Dipeptidyl Peptidase-4 (DPP-4) via a Non-Covalent Mechanism<br /><i>PLoS ONE</i> <b>11</b>: e0157509<br /><br />Zhang Z, Wallace MB, Feng J, Stafford JA, Skene RJ, Shi L, Lee B, Aertgeerts K, Jennings A, Xu R, Kassel DB, Kaldor SW, Navre M, Webb DR, Gwaltney SL (2011) <br />Design and synthesis of pyrimidinone and pyrimidinedione inhibitors of dipeptidyl peptidase IV<br /><i>Journal of Medicinal Chemistry</i> <b>54</b>: 510<br /><br />Aertgeerts K, Levin I, Shi L, Snell GP, Jennings A, Prasad GS, Zhang Y, Kraus ML, Salakian S, Sridhar V, Wijnands R, Tennant MG (2005) <br />Structural and kinetic analysis of the substrate specificity of human fibroblast activation protein alpha<br /><i>Journal of Biological Chemistry</i> <b>280</b>: 19441<br /><br />