Okondo MC, Rao SD, Taabazuing CY, Chui AJ, Poplawski SE, Johnson DC, Bachovchin DA (2018)
Inhibition of Dpp8/9 Activates the Nlrp1b Inflammasome
Cell Chemical Biology 25: 262
Okondo MC, Johnson DC, Sridharan R, Go EB, Chui AJ, Wang MS, Poplawski SE, Wu W, Liu Y, Lai JH, Sanford DG, Arciprete MO, Golub TR, Bachovchin WW, Bachovchin DA (2017)
DPP8 and DPP9 inhibition induces pro-caspase-1-dependent monocyte and macrophage pyroptosis
Nat Chemical Biology 13: 46
Bachovchin DA, Koblan LW, Wu W, Liu Y, Li Y, Zhao P, Woznica I, Shu Y, Lai JH, Poplawski SE, Kiritsy CP, Healey SE, DiMare M, Sanford DG, Munford RS, Bachovchin WW, Golub TR (2014)
A high-throughput, multiplexed assay for superfamily-wide profiling of enzyme activity
Nat Chemical Biology 10: 656
Keane FM, Yao TW, Seelk S, Gall MG, Chowdhury S, Poplawski SE, Lai JH, Li Y, Wu W, Farrell P, Vieira de Ribeiro AJ, Osborne B, Yu DM, Seth D, Rahman K, Haber P, Topaloglu AK, Wang C, Thomson S, Hennessy A, Prins J, Twigg SM, McLennan SV, McCaughan GW, Bachovchin WW, Gorrell MD (2013)
Quantitation of fibroblast activation protein (FAP)-specific protease activity in mouse, baboon and human fluids and organs
FEBS Open Bio 4: 43
Poplawski SE, Lai JH, Li Y, Jin Z, Liu Y, Wu W, Wu Y, Zhou Y, Sudmeier JL, Sanford DG, Bachovchin WW (2013)
Identification of selective and potent inhibitors of fibroblast activation protein and prolyl oligopeptidase
Journal of Medicinal Chemistry 56: 3467
Wu W, Liu Y, Milo LJ, Jr., Shu Y, Zhao P, Li Y, Woznica I, Yu G, Sanford DG, Zhou Y, Poplawski SE, Connolly BA, Sudmeier JL, Bachovchin WW, Lai JH (2012)
4-Substituted boro-proline dipeptides: synthesis, characterization, and dipeptidyl peptidase IV, 8, and 9 activities
Bioorganic & Medicinal Chemistry Lett 22: 5536
Poplawski SE, Lai JH, Sanford DG, Sudmeier JL, Wu W, Bachovchin WW (2011)
Pro-soft Val-boroPro: a strategy for enhancing in vivo performance of boronic acid inhibitors of serine proteases
Journal of Medicinal Chemistry 54: 2022
Lai JH, Wu W, Zhou Y, Maw HH, Liu Y, Milo LJ, Jr., Poplawski SE, Henry GD, Sudmeier JL, Sanford DG, Bachovchin WW (2007)
Synthesis and characterization of constrained peptidomimetic dipeptidyl peptidase IV inhibitors: amino-lactam boroalanines
Journal of Medicinal Chemistry 50: 2391