Zhao N, Darby CM, Small J, Bachovchin DA, Jiang X, Burns-Huang KE, Botella H, Ehrt S, Boger DL, Anderson ED, Cravatt BF, Speers AE, Fernandez-Vega V, Hodder PS, Eberhart C, Rosen H, Spicer TP, Nathan CF (2015)
Target-Based Screen Against a Periplasmic Serine Protease That Regulates Intrabacterial pH Homeostasis in Mycobacterium tuberculosis
ACS Chemical Biology 10: 364
Adibekian A, Martin BR, Chang JW, Hsu KL, Tsuboi K, Bachovchin DA, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Cravatt BF, Hodder P, Rosen H (2013)
Characterization of a Selective, Reversible Inhibitor of Lysophospholipase 1 (LYPLA1)
Probe Report
Adibekian A, Martin BR, Chang JW, Hsu KL, Tsuboi K, Bachovchin DA, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Cravatt BF, Hodder P, Rosen H (2013)
Characterization of a Selective, Reversible Inhibitor of Lysophospholipase 2 (LYPLA2)
Probe Report
Hsu KL, Tsuboi K, Chang JW, Whitby LR, Speers AE, Pugh H, Cravatt BF (2013)
Discovery and optimization of piperidyl-1,2,3-triazole ureas as potent, selective, and in vivo-active inhibitors of alpha/beta-hydrolase domain containing 6 (ABHD6)
Journal of Medicinal Chemistry 56: 8270
Hsu KL, Tsuboi K, Whitby LR, Speers AE, Pugh H, Inloes J, Cravatt BF (2013)
Development and optimization of piperidyl-1,2,3-triazole ureas as selective chemical probes of endocannabinoid biosynthesis
Journal of Medicinal Chemistry 56: 8257
Nagano JM, Hsu KL, Whitby LR, Niphakis MJ, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Hodder P, Srinivasan P, Gonzalez TD, Rosen H, Bahnson BJ, Cravatt BF (2013)
Selective inhibitors and tailored activity probes for lipoprotein-associated phospholipase A(2)
Bioorganic & Medicinal Chemistry Lett 23: 839
Adibekian A, Martin BR, Chang JW, Hsu KL, Tsuboi K, Bachovchin DA, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Hodder PS, Rosen H, Cravatt BF (2012)
Confirming target engagement for reversible inhibitors in vivo by kinetically tuned activity-based probes
J Am Chem Soc 134: 10345
Hsu KL, Tsuboi K, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Cravatt BF, Hodder P, Rosen H (2012)
Optimization and characterization of a triazole urea inhibitor for diacylglycerol lipase beta (DAGL-beta)
Probe Report
Liu X, Dix M, Speers AE, Bachovchin DA, Zuhl AM, Cravatt BF, Kodadek TJ (2012)
Rapid development of a potent photo-triggered inhibitor of the serine hydrolase RBBP9
Chembiochem 13: 2082
Adibekian A, Hsu KL, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Cravatt BF, Hodder P, Rosen H (2011)
Optimization and characterization of a triazole urea inhibitor for alpha/beta hydrolase domain-containing protein 11 (ABHD11): anti-probe for LYPLA1/LYPLA2 dual inhibitor ML211
Probe Report
Adibekian A, Hsu KL, Speers AE, Monillas ES, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Bahnson BJ, Cravatt BF, Hodder P, Rosen H (2011)
Optimization and characterization of a triazole urea inhibitor for platelet-activating factor acetylhydrolase type 2 (PAFAH2)
Probe Report
Adibekian A, Martin BR, Speers AE, Brown SJ, Spicer T, Fernandez-Vega V, Ferguson J, Cravatt BF, Hodder P, Rosen H (2011)
Optimization and characterization of a triazole urea dual inhibitor for lysophospholipase 1 (LYPLA1) and lysophospholipase 2 (LYPLA2)
Probe Report
Lone AM, Bachovchin DA, Westwood DB, Speers AE, Spicer TP, Fernandez-Vega V, Chase P, Hodder PS, Rosen H, Cravatt BF, Saghatelian A (2011)
A substrate-free activity-based protein profiling screen for the discovery of selective PREPL inhibitors
Journal of the American Chemical Society 133: 11665
Bachovchin DA, Speers AE, Brown SJ, Spicer TP, Fernandez V, Ferguson J, Mohr JT, Murphy J, Fu GC, Cravatt BF, Hodder PS, Rosen H (2010)
Probe Development Efforts to Identify Novel Inhibitors of Protein Phosphatase Methylesterase-1 (PME-1)
Probe Report
Bachovchin DA, Speers AE, Brown SJ, Cravatt BF, Spicer T, Mercer BA, Ferguson J, Hodder P, Rosen HR (2010)
Probe Report for RBBP9 Inhibitors - Probe 2
Probe Report
Bachovchin DA, Speers AE, Zuhl AM, Brown SJ, Cravatt BF, Fernandez V, Spicer T, Mercer BA, Ferguson J, Hodder P, Rosen HR (2010)
Probe Report for PME-1 Inhibitors
Probe Report