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Inhibitor Report for: E2030

General
Type Pyridine, Boron compound
Chemical_Nomenclature [2-methoxy-5-[(E)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)ethenyl]pyridin-4-yl]methanamine
Canonical SMILES B1(OC(C(O1)(C)C)(C)C)C=CC2=CN=C(C=C2CN)OC
InChI InChI=1S/C15H23BN2O3/c1-14(2)15(3,4)21-16(20-14)7-6-11-10-18-13(19-5)8-12(11)9-17/h6-8,10H,9,17H2,1-5H3/b7-6+
InChIKey LAGBVTUFYIBFIX-VOTSOKGWSA-N
Other name(s) E-2030 ; 3-(2-(1-(1,3-dioxolan-2-ylmethyl)-4-piperidyl)ethyl)-2H-3,4-dihydro-1,3-benzoxazin-2,4-dione hydrochloride
________________________________________________________________________________________________
MW|290.16
Formula|C15H23BN2O3
CAS_number|
PubChem|74890773
UniChem|LAGBVTUFYIBFIX-VOTSOKGWSA-N
IUPHAR|
Wikipedia|

Target
Families | E2030 ligand of proteins in family: ACHE, BCHE

References:
Search PubMed for references concerning: E2030
    Title: Central and peripheral activity of cholinesterase inhibitors as revealed by yawning and fasciculation in rats
    Ogura H, Kosasa T, Kuriya Y, Yamanishi Y
    Ref: European Journal of Pharmacology, 415:157, 2001 : PubMed