Mutation

Kinetic parameters

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Kinetic parameters for mutation E450A_human-ACHE

Substrate

MoleculeKmKcatExp. conditionsReference

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
HuperzineA 6 & 1 nM - - 50mM Na phosphate pH8 T22C Acetylthiocholine Ariel_1998_Biochem.J_335_95
Tacrine 530 & 50 nM 870 & 70 nM - 50mM Na phosphate pH8 T22C Acetylthiocholine Ariel_1998_Biochem.J_335_95

Send your questions or comments to :
Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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