Mutation

Kinetic parameters

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Kinetic parameters for mutation F297I_mouse-ACHE

Substrate

MoleculeKmKcatExp. conditionsReference
Acetylthiocholine 170 uM 15000 /min 100mM NaPhosphate Ph7.0 T22C Hosea_1995_Biochemistry_34_11528
Acetylthiocholine 172 & 64 uM 15000 & 2000/min 100mM NaP pH7 T22C eq3 sch3 Radic_1993_Biochemistry_32_12074
Benzoylthiocholine 19 uM 450 /min 100mM NaPhosphate Ph7.0 T22C Hosea_1995_Biochemistry_34_11528
Butyrylthiocholine 82 uM 60000 /min 100mM NaPhosphate Ph7.0 T22C Hosea_1995_Biochemistry_34_11528

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
WT-fasciculin2 - 19 pM - 100mM NaP pH7.0 T37C eq4 sch4 meth5 Acetylthiocholine Radic_1994_J.Biol.Chem_269_11233

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Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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