Mutation

Kinetic parameters

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Kinetic parameters for mutation Y124Q_mouse-ACHE

Substrate

MoleculeKmKcatExp. conditionsReference
Acetylthiocholine 120 & 21 uM 110000 & 30000/min 100mM NaP pH7 T22C eq3 sch3 Radic_1993_Biochemistry_32_12074

Inhibitor

MoleculeKiKsiIc50Exp. conditionsSubstrateReference
BW284C51 16 & 2 nM 60 & 31 nM - 100mM NaP pH7.0 T22C eq3.gif sch3.gif Acetylthiocholine Radic_1993_Biochemistry_32_12074
Decamethonium 26 & 6 uM 68 & 2 uM - 100mM NaP pH7.0 T22C eq3.gif sch3.gif Acetylthiocholine Radic_1993_Biochemistry_32_12074
Propidium 13 & 6 uM 66 & 18 uM - 100mM NaP pH7.0 T22C eq3.gif sch3.gif Acetylthiocholine Radic_1993_Biochemistry_32_12074
WT-fasciculin2 - 590 pM - 100mM NaP pH7.0 T37C eq4 sch4 meth5 Acetylthiocholine Radic_1994_J.Biol.Chem_269_11233

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Mail to: Nicolas Lenfant, Thierry Hotelier, Yves Bourne, Pascale Marchot and Arnaud Chatonnet.
Please cite: Lenfant 2013 Nucleic.Acids.Res. or Marchot Chatonnet 2012 Prot.Pept Lett.
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