Kato_2011_Bioorg.Med.Chem_19_7221

Reference

Title : Discovery and pharmacological characterization of N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methyl pyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride (anagliptin hydrochloride salt) as a potent and selective DPP-IV inhibitor - Kato_2011_Bioorg.Med.Chem_19_7221
Author(s) : Kato N , Oka M , Murase T , Yoshida M , Sakairi M , Yamashita S , Yasuda Y , Yoshikawa A , Hayashi Y , Makino M , Takeda M , Mirensha Y , Kakigami T
Ref : Bioorganic & Medicinal Chemistry , 19 :7221 , 2011
Abstract : Kato_2011_Bioorg.Med.Chem_19_7221
ESTHER : Kato_2011_Bioorg.Med.Chem_19_7221
PubMedSearch : Kato_2011_Bioorg.Med.Chem_19_7221
PubMedID: 22019046

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Kato N, Oka M, Murase T, Yoshida M, Sakairi M, Yamashita S, Yasuda Y, Yoshikawa A, Hayashi Y, Makino M, Takeda M, Mirensha Y, Kakigami T (2011)
Discovery and pharmacological characterization of N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methyl pyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride (anagliptin hydrochloride salt) as a potent and selective DPP-IV inhibitor
Bioorganic & Medicinal Chemistry 19 :7221

Kato N, Oka M, Murase T, Yoshida M, Sakairi M, Yamashita S, Yasuda Y, Yoshikawa A, Hayashi Y, Makino M, Takeda M, Mirensha Y, Kakigami T (2011)
Bioorganic & Medicinal Chemistry 19 :7221