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Paper Report for: Woolford_2016_J.Med.Chem_59_10738

Reference
Title: Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2)
Woolford AJ, Day PJ, Beneton V, Berdini V, Coyle JE, Dudit Y, Grondin P, Huet P, Lee LY and Zhang X <11 more author(s)>
Ref: Journal of Medicinal Chemistry, 59:10738, 2016 : PubMed

        


Related information
Gene_Locus : human-PLA2G7
Structure in RCSB-PDB : 5LYY, 5LZ2, 5LZ4, 5LZ5, 5LZ7, 5LZ8, 5LZ9
Structure in ESTHER : 5LYY, 5LZ2, 5LZ4, 5LZ5, 5LZ7, 5LZ8, 5LZ9
Inhibitor : 7BP-5LZ8, CHEMBL3924430, CHEMBL3983270, CHEMBL3975283, 3-cyano-N-cyclopropylbenzenesulfonamide, CHEMBL3908555, 5LZ9-7BR,

Citations formats
Woolford AJ, Day PJ, Beneton V, Berdini V, Coyle JE, Dudit Y, Grondin P, Huet P, Lee LY, Manas ES, McMenamin RL, Murray CW, Page LW, Patel VK, Potvain F, Rich SJ, Sang Y, Somers DO, Trottet L, Wan Z, Zhang X (2016)
Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2)
Journal of Medicinal Chemistry 59: 10738-10749

Woolford AJ, Day PJ, Beneton V, Berdini V, Coyle JE, Dudit Y, Grondin P, Huet P, Lee LY, Manas ES, McMenamin RL, Murray CW, Page LW, Patel VK, Potvain F, Rich SJ, Sang Y, Somers DO, Trottet L, Wan Z, Zhang X (2016)
Journal of Medicinal Chemistry 59: 10738-10749


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