4JNC
Name : Soluble Epoxide Hydrolase complexed with a carboxamide inhibitor
Revelation date : 05-Jun-2013
Family : Epoxide_hydrolase
Gene_locus : human-EPHX2
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Thalji, R.K., McAtee, J.J., Belyanskaya, S., Brandt, M., Brown, G.D., Costell, M.H., Ding, Y., Dodson, J.W., Eisennagel, S.H., Fries, R.E., Gross, J.W., Harpel, M.R., Holt, D.A., Israel, D.I., Jolivette, L.J., Krosky, D., Li, H., Lu, Q., Mandichak, T., Roethke, T., Schnackenberg, C.G., Schwartz, B., Shewchuk, L.M., Xie, W., Behm, D.J., Douglas, S.A., Shaw, A.L., Marino, J.P.
Ligand :
References (1)
| Title : Discovery of 1-(1,3,5-triazin-2-yl)piperidine-4-carboxamides as inhibitors of soluble epoxide hydrolase - Thalji_2013_Bioorg.Med.Chem.Lett_23_3584 |
| Author(s) : Thalji RK , McAtee JJ , Belyanskaya S , Brandt M , Brown GD , Costell MH , Ding Y , Dodson JW , Eisennagel SH , Fries RE , Gross JW , Harpel MR , Holt DA , Israel DI , Jolivette LJ , Krosky D , Li H , Lu Q , Mandichak T , Roethke T , Schnackenberg CG , Schwartz B , Shewchuk LM , Xie W , Behm DJ , Douglas SA , Shaw AL , Marino JP, Jr. |
| Ref : Bioorganic & Medicinal Chemistry Lett , 23 :3584 , 2013 |
| Abstract : Thalji_2013_Bioorg.Med.Chem.Lett_23_3584 |
| ESTHER : Thalji_2013_Bioorg.Med.Chem.Lett_23_3584 |
| PubMedSearch : Thalji_2013_Bioorg.Med.Chem.Lett_23_3584 |
| PubMedID: 23664879 |
| Gene_locus related to this paper: human-EPHX2 |
Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server
