6AX1

Name : Structure of human monoacylglycerol lipase bound to a covalent inhibitor

Revelation date : 27-Dec-2017

Family : Monoglyceridelipase_lysophospholip

Gene_locus : human-MGLL

PDB file : ESTHER: header of PDB entry RCSB: Full entry

Comment
Pandit, J.

Ligand :

References (1)

Title : Azetidine and Piperidine Carbamates as Efficient, Covalent Inhibitors of Monoacylglycerol Lipase - Butler_2017_J.Med.Chem_60_9860
Author(s) : Butler CR , Beck EM , Harris A , Huang Z , McAllister LA , Am Ende CW , Fennell K , Foley TL , Fonseca K , Hawrylik SJ , Johnson DS , Knafels JD , Mente S , Noell GS , Pandit J , Phillips TB , Piro JR , Rogers BN , Samad TA , Wang J , Wan S , Brodney MA
Ref : Journal of Medicinal Chemistry , 60 :9860 , 2017
Abstract : Butler_2017_J.Med.Chem_60_9860
ESTHER : Butler_2017_J.Med.Chem_60_9860
PubMedSearch : Butler_2017_J.Med.Chem_60_9860
PubMedID: 29148769
Gene_locus related to this paper: human-MGLL

Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server

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