2OQI
Name : Human Dipeptidyl Peptidase IV (DPP4) with Piperidinone-constrained phenethylamine
Revelation date : 03-Apr-2007
Family : DPP4N_Peptidase_S9
Gene_locus : human-DPP4
PDB file : ESTHER: header of PDB entry RCSB: Full entry
Comment
Pei, Z., Li, X., von Geldern, T. W., Longenecker, K.L., Pireh, D., Stewart, K.D., Backes, B.J., Lai, C., Lubben, T.H., Ballaron, S.J., Beno, D.W., Kempf-Grote, A.J., Sham, H.L., Trevillyan, J.M.
Ligand :
References (1)
| Title : Discovery and structure-activity relationships of piperidinone- and piperidine-constrained phenethylamines as novel, potent, and selective dipeptidyl peptidase IV inhibitors - Pei_2007_J.Med.Chem_50_1983 |
| Author(s) : Pei Z , Li X , von Geldern TW , Longenecker K , Pireh D , Stewart KD , Backes BJ , Lai C , Lubben TH , Ballaron SJ , Beno DW , Kempf-Grote AJ , Sham HL , Trevillyan JM |
| Ref : Journal of Medicinal Chemistry , 50 :1983 , 2007 |
| Abstract : Pei_2007_J.Med.Chem_50_1983 |
| ESTHER : Pei_2007_J.Med.Chem_50_1983 |
| PubMedSearch : Pei_2007_J.Med.Chem_50_1983 |
| PubMedID: 17367123 |
| Gene_locus related to this paper: human-DPP4 |
Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server
