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Inhibitor Report for: GSK-264220A

Name Class
GSK-264220ATypeUrea derivative
Sulfur Compound
Sulfonamide
Other_Name (5)
Chemical_Nomenclature1-(2-methyl-5-piperidin-1-ylsulfonylfuran-3-yl)-3-phenylurea
FormulaC17H21N3O4S
CAS_number685506-42-7
MW363.43
PaperGoodman_2009_Bioorg.Med.Chem.Lett_19_27
CommentSelective sulfonylfuran urea endothelial lipase inhibitors (human-LIPG)
Gene_locushuman-LIPG
CID2810413
FamilyLipoprotein_Lipase
InChIKeyLVOVQRPAMXCXTM-UHFFFAOYSA-N
CanonicalSMILESCC1=C(C=C(O1)S(=O)(=O)N2CCCCC2)NC(=O)NC3=CC=CC=C3
InChIInChI=1S/C17H21N3O4S/c1-13-15(19-17(21)18-14-8-4-2-5-9-14)12-16(24-13)25(22,23)20-10-6-3-7-11-20/h2,4-5,8-9,12H,3,6-7,10-11H2,1H3,(H2,18,19,21)
IupharLig6697

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