<Journal class="Journal" value="Journal of Biological Chemistry" /> <Page class="#txt" value="27819"> <Page-2 class="#txt" value="22" /> </Page> <Volume class="#txt" value="269" /> <Year class="Year" value="1994" /> </Reference> <Author class="Author" value="Kronman C" /> <Author class="Author" value="Ordentlich A" /> <Author class="Author" value="Barak D" /> <Author class="Author" value="Velan B" /> <Author class="Author" value="Shafferman A" /> <Medline class="Medline" value="7961709" /> <Mutation class="Mutation" value="E84Q_human-ACHE" /> <Mutation class="Mutation" value="W86A_human-ACHE" /> <Mutation class="Mutation" value="D131N_human-ACHE" /> <Mutation class="Mutation" value="V132A_human-ACHE" /> <Mutation class="Mutation" value="V132K_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_W86A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_D131N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_V132A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_V132K_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_D131N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_V132A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_V132K_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_W86A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_D131N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_V132A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_V132K_human-ACHE" /> <Abstract class="LongText" value="Kronman_1994_J.Biol.Chem_269_27819" /> <Inhibitor class="Inhibitor" value="Edrophonium" /> <Substrate class="Substrate" value="3,3-dimethylbutylthioacetate" /> <Substrate class="Substrate" value="Acetylthiocholine" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_D131N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_V132A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_V132K_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_D131N_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_V132A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_V132K_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_D131N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_V132A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_V132K_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_D131N_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_V132A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_V132K_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_D131N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_V132A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_V132K_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_D131N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_V132A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_V132K_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_D131N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_V132K_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_V132A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_D131N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_V132K_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_V132A_human-ACHE" /> </Paper>