<Journal class="Journal" value="Journal of Biological Chemistry" /> <Page class="#txt" value="17083"> <Page-2 class="#txt" value="95" /> </Page> <Volume class="#txt" value="268" /> <Year class="Year" value="1993" /> </Reference> <Author class="Author" value="Ordentlich A" /> <Author class="Author" value="Barak D" /> <Author class="Author" value="Kronman C" /> <Author class="Author" value="Flashner Y" /> <Author class="Author" value="Leitner M" /> <Author class="Author" value="Segall Y" /> <Author class="Author" value="Ariel N" /> <Author class="Author" value="Cohen S" /> <Author class="Author" value="Velan B" /> <Author class="Author" value="Shafferman A" /> <Medline class="Medline" value="8349597" /> <Mutation class="Mutation" value="F297V_human-ACHE" /> <Mutation class="Mutation" value="F295L/F297V_human-ACHE" /> <Mutation class="Mutation" value="W86A_human-ACHE" /> <Mutation class="Mutation" value="E202Q_human-ACHE" /> <Mutation class="Mutation" value="W286A_human-ACHE" /> <Mutation class="Mutation" value="F295A_human-ACHE" /> <Mutation class="Mutation" value="F295L_human-ACHE" /> <Mutation class="Mutation" value="F297A_human-ACHE" /> <Mutation class="Mutation" value="Y337F_human-ACHE" /> <Mutation class="Mutation" value="F338A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_W286A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_Y337A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_F338A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_W86A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_W286A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_Y337A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_F338A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="S-N-Propylthioacetate_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="S-N-Propylthioacetate_W286A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="S-N-Propylthioacetate_Y337A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="S-N-Propylthioacetate_F338A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="S-N-Propylthioacetate_W86A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Paranitrophenylacetate_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Paranitrophenylacetate_W286A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Paranitrophenylacetate_Y337A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Paranitrophenylacetate_F338A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Paranitrophenylacetate_W86A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_W286A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_Y337A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_F338A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_W86A_human-ACHE" /> <Abstract class="LongText" value="Ordentlich_1993_J.Biol.Chem_268_17083" /> <Inhibitor class="Inhibitor" value="Edrophonium" /> <Substrate class="Substrate" value="3,3-dimethylbutylthioacetate" /> <Substrate class="Substrate" value="Paranitrophenylacetate" /> <Substrate class="Substrate" value="S-N-Propylthioacetate" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_S-N-Propylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Km_S-N-Propylthioacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_S-N-Propylthioacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_S-N-Propylthioacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_S-N-Propylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Paranitrophenylacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Paranitrophenylacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Paranitrophenylacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Paranitrophenylacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Paranitrophenylacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_S-N-Propylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_S-N-Propylthioacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_S-N-Propylthioacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_S-N-Propylthioacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Paranitrophenylacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Paranitrophenylacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Paranitrophenylacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Paranitrophenylacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Paranitrophenylacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_S-N-Propylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_S-N-Propylthioacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_S-N-Propylthioacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_S-N-Propylthioacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_S-N-Propylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Paranitrophenylacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Paranitrophenylacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Paranitrophenylacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Paranitrophenylacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Paranitrophenylacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethybutylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_3,3-dimethylbutylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_S-N-Propylthioacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_S-N-Propylthioacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_S-N-Propylthioacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_S-N-Propylthioacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_S-N-Propylthioacetate_W86A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Paranitrophenylacetate_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Paranitrophenylacetate_W286A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Paranitrophenylacetate_Y337A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Paranitrophenylacetate_F338A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Paranitrophenylacetate_W86A_human-ACHE" /> </Paper>