<Journal class="Journal" value="EMBO Journal" /> <Page class="#txt" value="3448"> <Page-2 class="#txt" value="55" /> </Page> <Volume class="#txt" value="13" /> <Year class="Year" value="1994" /> </Reference> <Author class="Author" value="Shafferman A" /> <Author class="Author" value="Ordentlich A" /> <Author class="Author" value="Barak D" /> <Author class="Author" value="Kronman C" /> <Author class="Author" value="Ber R" /> <Author class="Author" value="Bino T" /> <Author class="Author" value="Ariel N" /> <Author class="Author" value="Osman R" /> <Author class="Author" value="Velan B" /> <Medline class="Medline" value="8062821" /> <Mutation class="Mutation" value="E84Q_human-ACHE" /> <Mutation class="Mutation" value="E84Q/E292A_human-ACHE" /> <Mutation class="Mutation" value="E84Q/D349N/E358Q_human-ACHE" /> <Mutation class="Mutation" value="E84Q/E292A/D349N/E358Q_human-ACHE" /> <Mutation class="Mutation" value="E84Q/E285A/E292A/D349N/E358Q_human-ACHE" /> <Mutation class="Mutation" value="E84Q/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Mutation class="Mutation" value="E84Q/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Mutation class="Mutation" value="E84Q/E285A/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Mutation class="Mutation" value="E285A_human-ACHE" /> <Mutation class="Mutation" value="E292A_human-ACHE" /> <Mutation class="Mutation" value="E292A/D349N/E358Q_human-ACHE" /> <Mutation class="Mutation" value="E292A/E389Q/D390N_human-ACHE" /> <Mutation class="Mutation" value="E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Mutation class="Mutation" value="D349N_human-ACHE" /> <Mutation class="Mutation" value="D349N/E358Q_human-ACHE" /> <Mutation class="Mutation" value="D349N/E358Q/E389Q/D390N_human-ACHE" /> <Mutation class="Mutation" value="E358Q_human-ACHE" /> <Mutation class="Mutation" value="E389Q_human-ACHE" /> <Mutation class="Mutation" value="E389Q/D390N_human-ACHE" /> <Mutation class="Mutation" value="D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E292A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E285A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_D349N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E389Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q/E292A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E292A/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q/E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q/E285A/E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Acetylthiocholine_E84Q/E285A/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E292A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E285A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_D349N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E389Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q/E292A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E292A/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q/E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q/E285A/E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="3,3-dimethylbutylthioacetate_E84Q/E285A/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_WT_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E292A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E285A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_D349N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E389Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q/E292A_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E292A/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q/E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q/E285A/E292A/D349N/E358Q_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kinetic_parameter class="Kinetic_parameter" value="Edrophonium_E84Q/E285A/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Abstract class="LongText" value="Shafferman_1994_EMBO.J_13_3448" /> <Inhibitor class="Inhibitor" value="Edrophonium" /> <Substrate class="Substrate" value="3,3-dimethylbutylthioacetate" /> <Substrate class="Substrate" value="Acetylthiocholine" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E292A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E285A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_D349N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E389Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q/E292A_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E292A/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q/E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q/E285A/E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Km_Acetylthiocholine_E84Q/E285A/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E292A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E285A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_D349N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E389Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q/E292A_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E292A/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q/E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q/E285A/E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kcat_Acetylthiocholine_E84Q/E285A/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E292A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E285A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_D349N_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E389Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E84Q/E292A_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E84Q/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E292A/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_E84Q/E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Kapp_Acetylthiocholine_D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" 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value="Kapp_3,3-dimethylbutylthioacetate_E84Q/E285A/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_WT_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E292A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E285A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_D349N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E389Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q/E292A_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E292A/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q/E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q/E285A/E292A/D349N/E358Q_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> <Kin_value class="Kin_value" value="Ki_Edrophonium_Acetylthiocholine_E84Q/E285A/E292A/D349N/E358Q/E389Q/D390N_human-ACHE" /> </Paper>