| Title : Discovery of a Novel Acetylcholinesterase Inhibitor by Fragment-Based Design and Virtual Screening - Stavrakov_2021_Molecules_26_ |
| Author(s) : Stavrakov G , Philipova I , Lukarski A , Atanasova M , Georgiev B , Atanasova T , Konstantinov S , Doytchinova I |
| Ref : Molecules , 26 : , 2021 |
| Abstract : |
| PubMedSearch : Stavrakov_2021_Molecules_26_ |
| PubMedID: 33916760 |
| Title : Galantamine-Curcumin Hybrids as Dual-Site Binding Acetylcholinesterase Inhibitors - Stavrakov_2020_Molecules_25_ |
| Author(s) : Stavrakov G , Philipova I , Lukarski A , Atanasova M , Zheleva D , Zhivkova ZD , Ivanov S , Atanasova T , Konstantinov S , Doytchinova I |
| Ref : Molecules , 25 : , 2020 |
| Abstract : |
| PubMedSearch : Stavrakov_2020_Molecules_25_ |
| PubMedID: 32717861 |
| Title : Novel hits for acetylcholinesterase inhibition derived by docking-based screening on ZINC database - Doytchinova_2018_J.Enzyme.Inhib.Med.Chem_33_768 |
| Author(s) : Doytchinova I , Atanasova M , Valkova I , Stavrakov G , Philipova I , Zhivkova Z , Zheleva-Dimitrova D , Konstantinov S , Dimitrov I |
| Ref : J Enzyme Inhib Med Chem , 33 :768 , 2018 |
| Abstract : |
| PubMedSearch : Doytchinova_2018_J.Enzyme.Inhib.Med.Chem_33_768 |
| PubMedID: 29651876 |
| Title : Docking-based design and synthesis of galantamine-camphane hybrids as inhibitors of acetylcholinesterase - Stavrakov_2017_Chem.Biol.Drug.Des_90_709 |
| Author(s) : Stavrakov G , Philipova I , Zheleva-Dimitrova D , Valkova I , Salamanova E , Konstantinov S , Doytchinova I |
| Ref : Chemical Biology Drug Des , 90 :709 , 2017 |
| Abstract : |
| PubMedSearch : Stavrakov_2017_Chem.Biol.Drug.Des_90_709 |
| PubMedID: 28374576 |
| Title : Docking-based Design of Galantamine Derivatives with Dual-site Binding to Acetylcholinesterase - Stavrakov_2016_Mol.Inform_35_278 |
| Author(s) : Stavrakov G , Philipova I , Zheleva D , Atanasova M , Konstantinov S , Doytchinova I |
| Ref : Mol Inform , 35 :278 , 2016 |
| Abstract : |
| PubMedSearch : Stavrakov_2016_Mol.Inform_35_278 |
| PubMedID: 27492242 |