Title : Discovery of novel cholinesterase inhibitors easily crossing the blood-brain barrier via structure-property relationship investigation: Methylenedioxy-cinnamicamides containing tertiary amine side chain - Liu_2024_Chem.Biodivers__e202400557 |
Author(s) : Liu HR , Shi Q , Yang ZY , Wang YH , Yi BX , Gao XH , Ding YJ , Peng D , Chen YL |
Ref : Chem Biodivers , :e202400557 , 2024 |
Abstract : |
PubMedSearch : Liu_2024_Chem.Biodivers__e202400557 |
PubMedID: 38701359 |
Title : Design, synthesis and the evaluation of cholinesterase inhibition and blood-brain permeability of daidzein derivatives or analogs - Wang_2023_Chem.Biol.Drug.Des__ |
Author(s) : Wang YH , Gao XH , Li X , Ding YJ , Shi Q , Yang ZY , Peng D , Liu HR |
Ref : Chemical Biology Drug Des , : , 2023 |
Abstract : |
PubMedSearch : Wang_2023_Chem.Biol.Drug.Des__ |
PubMedID: 37291745 |
Title : Nitrogen-containing flavonoid and their analogs with diverse B-ring in acetylcholinesterase and butyrylcholinesterase inhibition - Lu_2020_Drug.Dev.Res__ |
Author(s) : Lu QQ , Chen YM , Liu HR , Yan JY , Cui PW , Zhang QF , Gao XH , Feng X , Liu YZ |
Ref : Drug Dev Res , : , 2020 |
Abstract : |
PubMedSearch : Lu_2020_Drug.Dev.Res__ |
PubMedID: 32754990 |
Title : Structure-activity study of fluorine or chlorine-substituted cinnamic acid derivatives with tertiary amine side chain in acetylcholinesterase and butyrylcholinesterase inhibition - Gao_2019_Drug.Dev.Res_80_438 |
Author(s) : Gao XH , Tang JJ , Liu HR , Liu LB , Liu YZ |
Ref : Drug Dev Res , 80 :438 , 2019 |
Abstract : |
PubMedSearch : Gao_2019_Drug.Dev.Res_80_438 |
PubMedID: 30680760 |
Title : Structure-activity relationship investigation of benzamide and picolinamide derivatives containing dimethylamine side chain as acetylcholinesterase inhibitors - Gao_2018_J.Enzyme.Inhib.Med.Chem_33_110 |
Author(s) : Gao XH , Liu LB , Liu HR , Tang JJ , Kang L , Wu H , Cui P , Yan J |
Ref : J Enzyme Inhib Med Chem , 33 :110 , 2018 |
Abstract : |
PubMedSearch : Gao_2018_J.Enzyme.Inhib.Med.Chem_33_110 |
PubMedID: 29166796 |
Title : Structure-activity relationship investigation of coumarin-chalcone hybrids with diverse side-chains as acetylcholinesterase and butyrylcholinesterase inhibitors - Kang_2018_Mol.Divers_22_893 |
Author(s) : Kang L , Gao XH , Liu HR , Men X , Wu HN , Cui PW , Oldfield E , Yan JY |
Ref : Mol Divers , 22 :893 , 2018 |
Abstract : |
PubMedSearch : Kang_2018_Mol.Divers_22_893 |
PubMedID: 29934672 |
Title : Discovery of potent and selective acetylcholinesterase (AChE) inhibitors: acacetin 7-O-methyl ether Mannich base derivatives synthesised from easy access natural product naringin - Liu_2017_Nat.Prod.Res__1 |
Author(s) : Liu HR , Men X , Gao XH , Liu LB , Fan HQ , Xia XH , Wang QA |
Ref : Nat Prod Res , :1 , 2017 |
Abstract : |
PubMedSearch : Liu_2017_Nat.Prod.Res__1 |
PubMedID: 28617100 |
Title : Tertiary amine derivatives of chlorochalcone as acetylcholinesterase (AChE) and buthylcholinesterase (BuChE) inhibitors: the influence of chlorine, alkyl amine side chain and alpha,beta-unsaturated ketone group - Gao_2016_J.Enzyme.Inhib.Med.Chem__1 |
Author(s) : Gao XH , Zhou C , Liu HR , Liu LB , Tang JJ , Xia XH |
Ref : J Enzyme Inhib Med Chem , :1 , 2016 |
Abstract : |
PubMedSearch : Gao_2016_J.Enzyme.Inhib.Med.Chem__1 |
PubMedID: 27801600 |
Title : Novel Potent and Selective Acetylcholinesterase Inhibitors as Potential Drugs for the Treatment of Alzheimer's Disease: Synthesis, Pharmacological Evaluation, and Molecular Modeling of Amino-Alkyl-Substituted Fluoro-Chalcones Derivatives - Liu_2015_Chem.Biol.Drug.Des_86_517 |
Author(s) : Liu HR , Zhou C , Fan HQ , Tang JJ , Liu LB , Gao XH , Wang QA , Liu WK |
Ref : Chemical Biology Drug Des , 86 :517 , 2015 |
Abstract : |
PubMedSearch : Liu_2015_Chem.Biol.Drug.Des_86_517 |
PubMedID: 25588967 |
Title : Design, synthesis and pharmacological evaluation of chalcone derivatives as acetylcholinesterase inhibitors - Liu_2014_Bioorg.Med.Chem_22_6124 |
Author(s) : Liu HR , Liu XJ , Fan HQ , Tang JJ , Gao XH , Liu WK |
Ref : Bioorganic & Medicinal Chemistry , 22 :6124 , 2014 |
Abstract : |
PubMedSearch : Liu_2014_Bioorg.Med.Chem_22_6124 |
PubMedID: 25260958 |
Title : Synthesis and acetylcholinesterase inhibitory activity of Mannich base derivatives flavokawain B - Liu_2014_Bioorg.Med.Chem.Lett_24_4749 |
Author(s) : Liu HR , Huang XQ , Lou DH , Liu XJ , Liu WK , Wang QA |
Ref : Bioorganic & Medicinal Chemistry Lett , 24 :4749 , 2014 |
Abstract : |
PubMedSearch : Liu_2014_Bioorg.Med.Chem.Lett_24_4749 |
PubMedID: 25205193 |