| Title : Coumarin Analogues as Promising Anti-Obesity Agents: In Silico Design, Synthesis, and In Vitro Pancreatic Lipase Inhibitory Activity - Yadav_2025_Chem.Biol.Drug.Des_105_e70046 |
| Author(s) : Yadav N , Paul AT |
| Ref : Chemical Biology Drug Des , 105 :e70046 , 2025 |
| Abstract : |
| PubMedSearch : Yadav_2025_Chem.Biol.Drug.Des_105_e70046 |
| PubMedID: 39865472 |
| Title : Coumarin Analogues as Promising Anti-Obesity Agents: In Silico Design, Synthesis, and In Vitro Pancreatic Lipase Inhibitory Activity - Yadav_2025_Chem.Biol.Drug.Des_105_e70046 |
| Author(s) : Yadav N , Paul AT |
| Ref : Chemical Biology Drug Des , 105 :e70046 , 2025 |
| Abstract : |
| PubMedSearch : Yadav_2025_Chem.Biol.Drug.Des_105_e70046 |
| PubMedID: 39865472 |
| Title : Design, Synthesis, and Pharmacological Evaluation of Prenylated Arylidene-Substituted Thiazolidinedione-Based Pancreatic Lipase Inhibitors as Anti-obesity Agents - Khator_2025_Arch.Pharm.(Weinheim)_358_e70135 |
| Author(s) : Khator R , Jagtap UA , Lavanya B , Paul AT , Monga V |
| Ref : Arch Pharm (Weinheim) , 358 :e70135 , 2025 |
| Abstract : |
| PubMedSearch : Khator_2025_Arch.Pharm.(Weinheim)_358_e70135 |
| PubMedID: 41214857 |
| Title : Synthetic pancreatic lipase inhibitors in obesity treatment: current updates on in silico design, synthesis, bioactivity, and SAR - Jagtap_2025_RSC.Med.Chem__ |
| Author(s) : Jagtap UA , Paul AT |
| Ref : RSC Med Chem , : , 2025 |
| Abstract : |
| PubMedSearch : Jagtap_2025_RSC.Med.Chem__ |
| PubMedID: 41058933 |
| Gene_locus related to this paper: human-PNLIP , pig-1plip |
| Title : Design, Synthesis, and Pharmacological Evaluation of Prenylated Arylidene-Substituted Thiazolidinedione-Based Pancreatic Lipase Inhibitors as Anti-obesity Agents - Khator_2025_Arch.Pharm.(Weinheim)_358_e70135 |
| Author(s) : Khator R , Jagtap UA , Lavanya B , Paul AT , Monga V |
| Ref : Arch Pharm (Weinheim) , 358 :e70135 , 2025 |
| Abstract : |
| PubMedSearch : Khator_2025_Arch.Pharm.(Weinheim)_358_e70135 |
| PubMedID: 41214857 |
| Title : Coumarin Analogues as Promising Anti-Obesity Agents: In Silico Design, Synthesis, and In Vitro Pancreatic Lipase Inhibitory Activity - Yadav_2025_Chem.Biol.Drug.Des_105_e70046 |
| Author(s) : Yadav N , Paul AT |
| Ref : Chemical Biology Drug Des , 105 :e70046 , 2025 |
| Abstract : |
| PubMedSearch : Yadav_2025_Chem.Biol.Drug.Des_105_e70046 |
| PubMedID: 39865472 |
| Title : Synthetic pancreatic lipase inhibitors in obesity treatment: current updates on in silico design, synthesis, bioactivity, and SAR - Jagtap_2025_RSC.Med.Chem__ |
| Author(s) : Jagtap UA , Paul AT |
| Ref : RSC Med Chem , : , 2025 |
| Abstract : |
| PubMedSearch : Jagtap_2025_RSC.Med.Chem__ |
| PubMedID: 41058933 |
| Gene_locus related to this paper: human-PNLIP , pig-1plip |
| Title : Design, Synthesis, and Pharmacological Evaluation of Prenylated Arylidene-Substituted Thiazolidinedione-Based Pancreatic Lipase Inhibitors as Anti-obesity Agents - Khator_2025_Arch.Pharm.(Weinheim)_358_e70135 |
| Author(s) : Khator R , Jagtap UA , Lavanya B , Paul AT , Monga V |
| Ref : Arch Pharm (Weinheim) , 358 :e70135 , 2025 |
| Abstract : |
| PubMedSearch : Khator_2025_Arch.Pharm.(Weinheim)_358_e70135 |
| PubMedID: 41214857 |
| Title : Synthetic pancreatic lipase inhibitors in obesity treatment: current updates on in silico design, synthesis, bioactivity, and SAR - Jagtap_2025_RSC.Med.Chem__ |
| Author(s) : Jagtap UA , Paul AT |
| Ref : RSC Med Chem , : , 2025 |
| Abstract : |
| PubMedSearch : Jagtap_2025_RSC.Med.Chem__ |
| PubMedID: 41058933 |
| Gene_locus related to this paper: human-PNLIP , pig-1plip |
| Title : Discovery of thiazolidinedione-based pancreatic lipase inhibitors as anti-obesity agents: synthesis, in silico studies and pharmacological investigations - Dhiman_2024_J.Biomol.Struct.Dyn__1 |
| Author(s) : Dhiman P , Yadav N , Auti PS , Jaswal S , Singh G , Mehan S , Ghosh B , Paul AT , Monga V |
| Ref : J Biomol Struct Dyn , :1 , 2024 |
| Abstract : |
| PubMedSearch : Dhiman_2024_J.Biomol.Struct.Dyn__1 |
| PubMedID: 38315459 |
| Title : Discovery of thiazolidinedione-based pancreatic lipase inhibitors as anti-obesity agents: synthesis, in silico studies and pharmacological investigations - Dhiman_2024_J.Biomol.Struct.Dyn__1 |
| Author(s) : Dhiman P , Yadav N , Auti PS , Jaswal S , Singh G , Mehan S , Ghosh B , Paul AT , Monga V |
| Ref : J Biomol Struct Dyn , :1 , 2024 |
| Abstract : |
| PubMedSearch : Dhiman_2024_J.Biomol.Struct.Dyn__1 |
| PubMedID: 38315459 |
| Title : Discovery of thiazolidinedione-based pancreatic lipase inhibitors as anti-obesity agents: synthesis, in silico studies and pharmacological investigations - Dhiman_2024_J.Biomol.Struct.Dyn__1 |
| Author(s) : Dhiman P , Yadav N , Auti PS , Jaswal S , Singh G , Mehan S , Ghosh B , Paul AT , Monga V |
| Ref : J Biomol Struct Dyn , :1 , 2024 |
| Abstract : |
| PubMedSearch : Dhiman_2024_J.Biomol.Struct.Dyn__1 |
| PubMedID: 38315459 |
| Title : Pancreatic lipase and its related proteins: where are we now? - Yadav_2023_Drug.Discov.Today__103855 |
| Author(s) : Yadav N , Paul AT |
| Ref : Drug Discov Today , :103855 , 2023 |
| Abstract : |
| PubMedSearch : Yadav_2023_Drug.Discov.Today__103855 |
| PubMedID: 38081381 |
| Title : Synthesis, molecular modelling and pharmacological evaluation of novel indole-thiazolidinedione based hybrid analogues as potential pancreatic lipase inhibitors - George_2023_J.Biomol.Struct.Dyn__1 |
| Author(s) : George G , Auti PS , Sengupta P , Yadav N , Paul AT |
| Ref : J Biomol Struct Dyn , :1 , 2023 |
| Abstract : |
| PubMedSearch : George_2023_J.Biomol.Struct.Dyn__1 |
| PubMedID: 38095559 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Pancreatic lipase and its related proteins: where are we now? - Yadav_2023_Drug.Discov.Today__103855 |
| Author(s) : Yadav N , Paul AT |
| Ref : Drug Discov Today , :103855 , 2023 |
| Abstract : |
| PubMedSearch : Yadav_2023_Drug.Discov.Today__103855 |
| PubMedID: 38081381 |
| Title : Synthesis, molecular modelling and pharmacological evaluation of novel indole-thiazolidinedione based hybrid analogues as potential pancreatic lipase inhibitors - George_2023_J.Biomol.Struct.Dyn__1 |
| Author(s) : George G , Auti PS , Sengupta P , Yadav N , Paul AT |
| Ref : J Biomol Struct Dyn , :1 , 2023 |
| Abstract : |
| PubMedSearch : George_2023_J.Biomol.Struct.Dyn__1 |
| PubMedID: 38095559 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Pancreatic lipase and its related proteins: where are we now? - Yadav_2023_Drug.Discov.Today__103855 |
| Author(s) : Yadav N , Paul AT |
| Ref : Drug Discov Today , :103855 , 2023 |
| Abstract : |
| PubMedSearch : Yadav_2023_Drug.Discov.Today__103855 |
| PubMedID: 38081381 |
| Title : Synthesis, molecular modelling and pharmacological evaluation of novel indole-thiazolidinedione based hybrid analogues as potential pancreatic lipase inhibitors - George_2023_J.Biomol.Struct.Dyn__1 |
| Author(s) : George G , Auti PS , Sengupta P , Yadav N , Paul AT |
| Ref : J Biomol Struct Dyn , :1 , 2023 |
| Abstract : |
| PubMedSearch : George_2023_J.Biomol.Struct.Dyn__1 |
| PubMedID: 38095559 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Synthesis, molecular modelling, in vitro and in vivo evaluation of conophylline inspired novel benzyloxy substituted indole glyoxylamides as potent pancreatic lipase inhibitors - Sridhar_2021_J.Biomol.Struct.Dyn__1 |
| Author(s) : Sridhar SNC , Sengupta P , Palawat S , Dileep PS , Ginson G , Paul AT |
| Ref : J Biomol Struct Dyn , :1 , 2021 |
| Abstract : |
| PubMedSearch : Sridhar_2021_J.Biomol.Struct.Dyn__1 |
| PubMedID: 34032197 |
| Title : Synthesis, molecular modelling, in vitro and in vivo evaluation of conophylline inspired novel benzyloxy substituted indole glyoxylamides as potent pancreatic lipase inhibitors - Sridhar_2021_J.Biomol.Struct.Dyn__1 |
| Author(s) : Sridhar SNC , Sengupta P , Palawat S , Dileep PS , Ginson G , Paul AT |
| Ref : J Biomol Struct Dyn , :1 , 2021 |
| Abstract : |
| PubMedSearch : Sridhar_2021_J.Biomol.Struct.Dyn__1 |
| PubMedID: 34032197 |
| Title : Synthesis, molecular modelling, in vitro and in vivo evaluation of conophylline inspired novel benzyloxy substituted indole glyoxylamides as potent pancreatic lipase inhibitors - Sridhar_2021_J.Biomol.Struct.Dyn__1 |
| Author(s) : Sridhar SNC , Sengupta P , Palawat S , Dileep PS , Ginson G , Paul AT |
| Ref : J Biomol Struct Dyn , :1 , 2021 |
| Abstract : |
| PubMedSearch : Sridhar_2021_J.Biomol.Struct.Dyn__1 |
| PubMedID: 34032197 |
| Title : Design, synthesis, evaluation, and molecular modeling studies of indolyl oxoacetamides as potential pancreatic lipase inhibitors - Sridhar_2020_Arch.Pharm.(Weinheim)_353_e2000048 |
| Author(s) : Sridhar SNC , Palawat S , Paul AT |
| Ref : Arch Pharm (Weinheim) , :e2000048 , 2020 |
| Abstract : |
| PubMedSearch : Sridhar_2020_Arch.Pharm.(Weinheim)_353_e2000048 |
| PubMedID: 32484265 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Design, synthesis, evaluation, and molecular modeling studies of indolyl oxoacetamides as potential pancreatic lipase inhibitors - Sridhar_2020_Arch.Pharm.(Weinheim)_353_e2000048 |
| Author(s) : Sridhar SNC , Palawat S , Paul AT |
| Ref : Arch Pharm (Weinheim) , :e2000048 , 2020 |
| Abstract : |
| PubMedSearch : Sridhar_2020_Arch.Pharm.(Weinheim)_353_e2000048 |
| PubMedID: 32484265 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Design, synthesis, evaluation, and molecular modeling studies of indolyl oxoacetamides as potential pancreatic lipase inhibitors - Sridhar_2020_Arch.Pharm.(Weinheim)_353_e2000048 |
| Author(s) : Sridhar SNC , Palawat S , Paul AT |
| Ref : Arch Pharm (Weinheim) , :e2000048 , 2020 |
| Abstract : |
| PubMedSearch : Sridhar_2020_Arch.Pharm.(Weinheim)_353_e2000048 |
| PubMedID: 32484265 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Design, synthesis, biological evaluation, and molecular modeling studies of rhodanine derivatives as pancreatic lipase inhibitors - Chauhan_2019_Arch.Pharm.(Weinheim)__e1900029 |
| Author(s) : Chauhan D , George G , Sridhar SNC , Bhatia R , Paul AT , Monga V |
| Ref : Arch Pharm (Weinheim) , :e1900029 , 2019 |
| Abstract : |
| PubMedSearch : Chauhan_2019_Arch.Pharm.(Weinheim)__e1900029 |
| PubMedID: 31407389 |
| Title : Design, synthesis, biological evaluation, and molecular modeling studies of rhodanine derivatives as pancreatic lipase inhibitors - Chauhan_2019_Arch.Pharm.(Weinheim)__e1900029 |
| Author(s) : Chauhan D , George G , Sridhar SNC , Bhatia R , Paul AT , Monga V |
| Ref : Arch Pharm (Weinheim) , :e1900029 , 2019 |
| Abstract : |
| PubMedSearch : Chauhan_2019_Arch.Pharm.(Weinheim)__e1900029 |
| PubMedID: 31407389 |
| Title : Design, synthesis, biological evaluation and molecular modelling studies of indole glyoxylamides as a new class of potential pancreatic lipase inhibitors - Sridhar_2019_Bioorg.Chem_85_373 |
| Author(s) : Sridhar SNC , Palawat S , Paul AT |
| Ref : Bioorg Chem , 85 :373 , 2019 |
| Abstract : |
| PubMedSearch : Sridhar_2019_Bioorg.Chem_85_373 |
| PubMedID: 30658237 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Design, synthesis, biological evaluation, and molecular modeling studies of rhodanine derivatives as pancreatic lipase inhibitors - Chauhan_2019_Arch.Pharm.(Weinheim)__e1900029 |
| Author(s) : Chauhan D , George G , Sridhar SNC , Bhatia R , Paul AT , Monga V |
| Ref : Arch Pharm (Weinheim) , :e1900029 , 2019 |
| Abstract : |
| PubMedSearch : Chauhan_2019_Arch.Pharm.(Weinheim)__e1900029 |
| PubMedID: 31407389 |
| Title : Design, synthesis, biological evaluation and molecular modelling studies of indole glyoxylamides as a new class of potential pancreatic lipase inhibitors - Sridhar_2019_Bioorg.Chem_85_373 |
| Author(s) : Sridhar SNC , Palawat S , Paul AT |
| Ref : Bioorg Chem , 85 :373 , 2019 |
| Abstract : |
| PubMedSearch : Sridhar_2019_Bioorg.Chem_85_373 |
| PubMedID: 30658237 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Design, synthesis, biological evaluation and molecular modelling studies of indole glyoxylamides as a new class of potential pancreatic lipase inhibitors - Sridhar_2019_Bioorg.Chem_85_373 |
| Author(s) : Sridhar SNC , Palawat S , Paul AT |
| Ref : Bioorg Chem , 85 :373 , 2019 |
| Abstract : |
| PubMedSearch : Sridhar_2019_Bioorg.Chem_85_373 |
| PubMedID: 30658237 |
| Gene_locus related to this paper: human-PNLIP |
| Title : Design, synthesis, biological evaluation and molecular modelling studies of novel diaryl substituted pyrazolyl thiazolidinediones as potent pancreatic lipase inhibitors - Sridhar_2017_Bioorg.Med.Chem.Lett_27_3749 |
| Author(s) : Sridhar NCS , Bhurta D , Kantiwal D , George G , Monga V , Paul AT |
| Ref : Bioorganic & Medicinal Chemistry Lett , 27 :3749 , 2017 |
| Abstract : |
| PubMedSearch : Sridhar_2017_Bioorg.Med.Chem.Lett_27_3749 |
| PubMedID: 28705641 |
| Title : Synthesis, evaluation and molecular modelling studies of 2-(carbazol-3-yl)-2-oxoacetamide analogues as a new class of potential pancreatic lipase inhibitors - Sridhar_2017_Bioorg.Med.Chem_25_609 |
| Author(s) : Sridhar SN , Ginson G , Venkataramana Reddy PO , Tantak MP , Kumar D , Paul AT |
| Ref : Bioorganic & Medicinal Chemistry , 25 :609 , 2017 |
| Abstract : |
| PubMedSearch : Sridhar_2017_Bioorg.Med.Chem_25_609 |
| PubMedID: 27908755 |
| Title : Design, synthesis, biological evaluation and molecular modelling studies of novel diaryl substituted pyrazolyl thiazolidinediones as potent pancreatic lipase inhibitors - Sridhar_2017_Bioorg.Med.Chem.Lett_27_3749 |
| Author(s) : Sridhar NCS , Bhurta D , Kantiwal D , George G , Monga V , Paul AT |
| Ref : Bioorganic & Medicinal Chemistry Lett , 27 :3749 , 2017 |
| Abstract : |
| PubMedSearch : Sridhar_2017_Bioorg.Med.Chem.Lett_27_3749 |
| PubMedID: 28705641 |
| Title : Synthesis, evaluation and molecular modelling studies of 2-(carbazol-3-yl)-2-oxoacetamide analogues as a new class of potential pancreatic lipase inhibitors - Sridhar_2017_Bioorg.Med.Chem_25_609 |
| Author(s) : Sridhar SN , Ginson G , Venkataramana Reddy PO , Tantak MP , Kumar D , Paul AT |
| Ref : Bioorganic & Medicinal Chemistry , 25 :609 , 2017 |
| Abstract : |
| PubMedSearch : Sridhar_2017_Bioorg.Med.Chem_25_609 |
| PubMedID: 27908755 |
| Title : Design, synthesis, biological evaluation and molecular modelling studies of novel diaryl substituted pyrazolyl thiazolidinediones as potent pancreatic lipase inhibitors - Sridhar_2017_Bioorg.Med.Chem.Lett_27_3749 |
| Author(s) : Sridhar NCS , Bhurta D , Kantiwal D , George G , Monga V , Paul AT |
| Ref : Bioorganic & Medicinal Chemistry Lett , 27 :3749 , 2017 |
| Abstract : |
| PubMedSearch : Sridhar_2017_Bioorg.Med.Chem.Lett_27_3749 |
| PubMedID: 28705641 |
| Title : Synthesis, evaluation and molecular modelling studies of 2-(carbazol-3-yl)-2-oxoacetamide analogues as a new class of potential pancreatic lipase inhibitors - Sridhar_2017_Bioorg.Med.Chem_25_609 |
| Author(s) : Sridhar SN , Ginson G , Venkataramana Reddy PO , Tantak MP , Kumar D , Paul AT |
| Ref : Bioorganic & Medicinal Chemistry , 25 :609 , 2017 |
| Abstract : |
| PubMedSearch : Sridhar_2017_Bioorg.Med.Chem_25_609 |
| PubMedID: 27908755 |