| Title : Aminomethylpyridines as DPP-IV inhibitors - Peters_2004_Bioorg.Med.Chem.Lett_14_3579 |
| Author(s) : Peters JU , Weber S , Kritter S , Weiss P , Wallier A , Zimmerli D , Boehringer M , Steger M , Loeffler BM |
| Ref : Bioorganic & Medicinal Chemistry Lett , 14 :3579 , 2004 |
|
Abstract :
In a novel series of DPP-IV inhibitors, a large increase of inhibitory activity was achieved by optimisation of aromatic substituents and conformational restriction. |
| PubMedSearch : Peters_2004_Bioorg.Med.Chem.Lett_14_3579 |
| PubMedID: 15177478 |
Peters JU, Weber S, Kritter S, Weiss P, Wallier A, Zimmerli D, Boehringer M, Steger M, Loeffler BM (2004)
Aminomethylpyridines as DPP-IV inhibitors
Bioorganic & Medicinal Chemistry Lett
14 :3579
Peters JU, Weber S, Kritter S, Weiss P, Wallier A, Zimmerli D, Boehringer M, Steger M, Loeffler BM (2004)
Bioorganic & Medicinal Chemistry Lett
14 :3579