1RWQ

Name : Human Dipeptidyl peptidase IV in complex with 5-aminomethyl-6-(2,4-dichloro-phenyl)-2-(3,5-dimethoxy-phenyl)-pyrimidin-4-amine

Revelation date : 17-Dec-2004

Family : DPP4N_Peptidase_S9

Gene_locus : human-DPP4

PDB file : ESTHER: header of PDB entry RCSB: Full entry

Comment
"Hennig, M., Thoma, R., Stihle, M."

Ligand :

References (1)

Title : Aminomethylpyrimidines as novel DPP-IV inhibitors: a 10(5)-fold activity increase by optimization of aromatic substituents - Peters_2004_Bioorg.Med.Chem.Lett_14_1491
Author(s) : Peters JU , Weber S , Kritter S , Weiss P , Wallier A , Boehringer M , Hennig M , Kuhn B , Loeffler BM
Ref : Bioorganic & Medicinal Chemistry Lett , 14 :1491 , 2004
Abstract : Peters_2004_Bioorg.Med.Chem.Lett_14_1491
ESTHER : Peters_2004_Bioorg.Med.Chem.Lett_14_1491
PubMedSearch : Peters_2004_Bioorg.Med.Chem.Lett_14_1491
PubMedID: 15006388
Gene_locus related to this paper: human-DPP4

Representative scheme of Prolylcarboxypeptidase structure and an image from PDBsum server

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