Title : Prodrugs of gamma-Alkyl-modified Nucleoside Triphosphates - improved Inhibition of HIV Reverse Transcriptase - Meier_2020_Angew.Chem.Int.Ed.Engl__ |
Author(s) : Meier C , Zhao C , Weber S , Schols D , Balzarini J |
Ref : Angew Chem Int Ed Engl , : , 2020 |
Abstract : |
PubMedSearch : Meier_2020_Angew.Chem.Int.Ed.Engl__ |
PubMedID: 32379948 |
Title : Dipeptidyl peptidase IV (DPPIV\/CD26)-based prodrugs of hydroxy-containing drugs - Diez-Torrubia_2012_ChemMedChem_7_618 |
Author(s) : Diez-Torrubia A , Cabrera S , Lambeir AM , Balzarini J , Camarasa MJ , Velazquez S |
Ref : ChemMedChem , 7 :618 , 2012 |
Abstract : |
PubMedSearch : Diez-Torrubia_2012_ChemMedChem_7_618 |
PubMedID: 22307932 |
Title : Application of the dipeptidyl peptidase IV (DPPIV\/CD26) based prodrug approach to different amine-containing drugs - Diez-Torrubia_2010_J.Med.Chem_53_559 |
Author(s) : Diez-Torrubia A , Garcia-Aparicio C , Cabrera S , De Meester I , Balzarini J , Camarasa MJ , Velazquez S |
Ref : Journal of Medicinal Chemistry , 53 :559 , 2010 |
Abstract : |
PubMedSearch : Diez-Torrubia_2010_J.Med.Chem_53_559 |
PubMedID: 20000418 |
Title : Efficient conversion of tetrapeptide-based TSAO prodrugs to the parent drug by dipeptidyl-peptidase IV (DPPIV\/CD26) - Garcia-Aparicio_2007_Antiviral.Res_76_130 |
Author(s) : Garcia-Aparicio C , Diez-Torrubia A , Balzarini J , Lambeir AM , Velazquez S , Camarasa MJ |
Ref : Antiviral Res , 76 :130 , 2007 |
Abstract : |
PubMedSearch : Garcia-Aparicio_2007_Antiviral.Res_76_130 |
PubMedID: 17675255 |
Title : Bis-cycloSal-d4T-monophosphates: drugs that deliver two molecules of bioactive nucleotides - Ducho_2007_J.Med.Chem_50_1335 |
Author(s) : Ducho C , Gorbig U , Jessel S , Gisch N , Balzarini J , Meier C |
Ref : Journal of Medicinal Chemistry , 50 :1335 , 2007 |
Abstract : |
PubMedSearch : Ducho_2007_J.Med.Chem_50_1335 |
PubMedID: 17328534 |
Title : Coexpression and interaction of CXCL10 and CD26 in mesenchymal cells by synergising inflammatory cytokines: CXCL8 and CXCL10 are discriminative markers for autoimmune arthropathies - Proost_2006_Arthritis.Res.Ther_8_R107 |
Author(s) : Proost P , Struyf S , Loos T , Gouwy M , Schutyser E , Conings R , Ronsse I , Parmentier M , Grillet B , Opdenakker G , Balzarini J , Van Damme J |
Ref : Arthritis Res Ther , 8 :R107 , 2006 |
Abstract : |
PubMedSearch : Proost_2006_Arthritis.Res.Ther_8_R107 |
PubMedID: 16846531 |
Title : Design and discovery of a novel dipeptidyl-peptidase IV (CD26)-based prodrug approach - Garcia-Aparicio_2006_J.Med.Chem_49_5339 |
Author(s) : Garcia-Aparicio C , Bonache MC , De Meester I , San-Felix A , Balzarini J , Camarasa MJ , Velazquez S |
Ref : Journal of Medicinal Chemistry , 49 :5339 , 2006 |
Abstract : |
PubMedSearch : Garcia-Aparicio_2006_J.Med.Chem_49_5339 |
PubMedID: 16913724 |
Title : cycloSal-PMEA and cycloAmb-PMEA: potentially new phosphonate prodrugs based on the cycloSal-pronucleotide approach - Meier_2005_J.Med.Chem_48_8079 |
Author(s) : Meier C , Gorbig U , Muller C , Balzarini J |
Ref : Journal of Medicinal Chemistry , 48 :8079 , 2005 |
Abstract : |
PubMedSearch : Meier_2005_J.Med.Chem_48_8079 |
PubMedID: 16335932 |
Title : Novel cyclosal nucleotides with reduced inhibitory potency toward human butyrylcholinesterase - Ducho_2005_Nucleosides.Nucleotides.Nucleic.Acids_24_519 |
Author(s) : Ducho C , Jessel S , Gisch N , Balzarini J , Meier C |
Ref : Nucleosides Nucleotides Nucleic Acids , 24 :519 , 2005 |
Abstract : |
PubMedSearch : Ducho_2005_Nucleosides.Nucleotides.Nucleic.Acids_24_519 |
PubMedID: 16247982 |
Title : Interaction of cycloSal-pronucleotides with cholinesterases from different origins. A structure-activity relationship - Meier_2004_J.Med.Chem_47_2839 |
Author(s) : Meier C , Ducho C , Gorbig U , Esnouf R , Balzarini J |
Ref : Journal of Medicinal Chemistry , 47 :2839 , 2004 |
Abstract : |
PubMedSearch : Meier_2004_J.Med.Chem_47_2839 |
PubMedID: 15139762 |
Title : Obligatory involvement of CD26\/dipeptidyl peptidase IV in the activation of the antiretroviral tripeptide glycylprolylglycinamide (GPG-NH(2)) - Balzarini_2004_Int.J.Biochem.Cell.Biol_36_1848 |
Author(s) : Balzarini J , Andersson E , Schols D , Proost P , Van Damme J , Svennerholm B , Horal P , Vahlne A |
Ref : International Journal of Biochemistryistry & Cell Biology , 36 :1848 , 2004 |
Abstract : |
PubMedSearch : Balzarini_2004_Int.J.Biochem.Cell.Biol_36_1848 |
PubMedID: 15183349 |
Title : Non-inhibition of acetylcholinesterase by cycloSal nucleotides - Ducho_2003_Nucleosides.Nucleotides.Nucleic.Acids_22_841 |
Author(s) : Ducho C , Balzarini J , Meier C |
Ref : Nucleosides Nucleotides Nucleic Acids , 22 :841 , 2003 |
Abstract : |
PubMedSearch : Ducho_2003_Nucleosides.Nucleotides.Nucleic.Acids_22_841 |
PubMedID: 14565292 |
Title : Intracellular metabolism of CycloSaligenyl 3'-azido-2', 3'-dideoxythymidine monophosphate, a prodrug of 3'-azido-2', 3'-dideoxythymidine (zidovudine) - Balzarini_1999_Mol.Pharmacol_56_1354 |
Author(s) : Balzarini J , Naesens L , Aquaro S , Knispel T , Perno C , De Clercq E , Meier C |
Ref : Molecular Pharmacology , 56 :1354 , 1999 |
Abstract : |
PubMedSearch : Balzarini_1999_Mol.Pharmacol_56_1354 |
PubMedID: 10570065 |
Title : 9-(2-Phosphonylmethoxyethyl)adenine induces tumor cell differentiation or cell death by blocking cell cycle progression through the S phase - Hatse_1999_Cell.Growth.Differ_10_435 |
Author(s) : Hatse S , Schols D , De Clercq E , Balzarini J |
Ref : Cell Growth Differ , 10 :435 , 1999 |
Abstract : |
PubMedSearch : Hatse_1999_Cell.Growth.Differ_10_435 |
PubMedID: 10392905 |