Title : Optimization of the choline transporter (CHT) inhibitor ML352: Development of VU6001221, an improved in vivo tool compound - Bertron_2016_Bioorg.Med.Chem.Lett_26_4637 |
Author(s) : Bertron JL , Ennis EA , Tarr CJ , Wright J , Dickerson JW , Locuson CW , Blobaum AL , Rook JM , Blakely RD , Lindsley CW |
Ref : Bioorganic & Medicinal Chemistry Lett , 26 :4637 , 2016 |
Abstract : |
PubMedSearch : Bertron_2016_Bioorg.Med.Chem.Lett_26_4637 |
PubMedID: 27575469 |
Title : Identification and Characterization of ML352: A Novel, Noncompetitive Inhibitor of the Presynaptic Choline Transporter - Ennis_2015_ACS.Chem.Neurosci_6_417 |
Author(s) : Ennis EA , Wright J , Retzlaff CL , McManus OB , Lin Z , Huang X , Wu M , Li M , Daniels JS , Lindsley CW , Hopkins CR , Blakely RD |
Ref : ACS Chem Neurosci , 6 :417 , 2015 |
Abstract : |
PubMedSearch : Ennis_2015_ACS.Chem.Neurosci_6_417 |
PubMedID: 25560927 |
Title : Transgenic overexpression of the presynaptic choline transporter elevates acetylcholine levels and augments motor endurance - Holmstrand_2014_Neurochem.Int_73_217 |
Author(s) : Holmstrand EC , Lund D , Cherian AK , Wright J , Martin RF , Ennis EA , Stanwood GD , Sarter M , Blakely RD |
Ref : Neurochem Int , 73 :217 , 2014 |
Abstract : |
PubMedSearch : Holmstrand_2014_Neurochem.Int_73_217 |
PubMedID: 24274995 |
Title : Nonoisotopic assay for the presynaptic choline transporter reveals capacity for allosteric modulation of choline uptake - Ruggiero_2012_ACS.Chem.Neurosci_3_767 |
Author(s) : Ruggiero AM , Wright J , Ferguson SM , Lewis M , Emerson KS , Iwamoto H , Ivy MT , Holmstrand EC , Ennis EA , Weaver CD , Blakely RD |
Ref : ACS Chem Neurosci , 3 :767 , 2012 |
Abstract : |
PubMedSearch : Ruggiero_2012_ACS.Chem.Neurosci_3_767 |
PubMedID: 23077721 |