Title : Selective Activation of N,N'-Diacyl Rhodamine Pro-fluorophores Paired with Releasing Enzyme, Porcine Liver Esterase (PLE) - Abney_2018_Chemistry_24_8985 |
Author(s) : Abney KK , Ramos-Hunter SJ , Romaine IM , Goodwin JS , Sulikowski GA , Weaver CD |
Ref : Chemistry , 24 :8985 , 2018 |
Abstract : |
PubMedSearch : Abney_2018_Chemistry_24_8985 |
PubMedID: 29679472 |
Title : Nonoisotopic assay for the presynaptic choline transporter reveals capacity for allosteric modulation of choline uptake - Ruggiero_2012_ACS.Chem.Neurosci_3_767 |
Author(s) : Ruggiero AM , Wright J , Ferguson SM , Lewis M , Emerson KS , Iwamoto H , Ivy MT , Holmstrand EC , Ennis EA , Weaver CD , Blakely RD |
Ref : ACS Chem Neurosci , 3 :767 , 2012 |
Abstract : |
PubMedSearch : Ruggiero_2012_ACS.Chem.Neurosci_3_767 |
PubMedID: 23077721 |
Title : Discovery and optimization of a novel, selective and brain penetrant M1 positive allosteric modulator (PAM): the development of ML169, an MLPCN probe - Reid_2011_Bioorg.Med.Chem.Lett_21_2697 |
Author(s) : Reid PR , Bridges TM , Sheffler DJ , Cho HP , Lewis LM , Days E , Daniels JS , Jones CK , Niswender CM , Weaver CD , Conn PJ , Lindsley CW , Wood MR |
Ref : Bioorganic & Medicinal Chemistry Lett , 21 :2697 , 2011 |
Abstract : |
PubMedSearch : Reid_2011_Bioorg.Med.Chem.Lett_21_2697 |
PubMedID: 21194936 |
Title : Discovery and characterization of novel subtype-selective allosteric agonists for the investigation of M(1) receptor function in the central nervous system - Lebois_2010_ACS.Chem.Neurosci_1_104 |
Author(s) : LeBois EP , Bridges TM , Lewis LM , Dawson ES , Kane AS , Xiang Z , Jadhav SB , Yin H , Kennedy JP , Meiler J , Niswender CM , Jones CK , Conn PJ , Weaver CD , Lindsley CW |
Ref : ACS Chem Neurosci , 1 :104 , 2010 |
Abstract : |
PubMedSearch : Lebois_2010_ACS.Chem.Neurosci_1_104 |
PubMedID: 21961051 |
Title : Discovery and characterization of novel allosteric potentiators of M1 muscarinic receptors reveals multiple modes of activity - Marlo_2009_Mol.Pharmacol_75_577 |
Author(s) : Marlo JE , Niswender CM , Days EL , Bridges TM , Xiang Y , Rodriguez AL , Shirey JK , Brady AE , Nalywajko T , Luo Q , Austin CA , Williams MB , Kim K , Williams R , Orton D , Brown HA , Lindsley CW , Weaver CD , Conn PJ |
Ref : Molecular Pharmacology , 75 :577 , 2009 |
Abstract : |
PubMedSearch : Marlo_2009_Mol.Pharmacol_75_577 |
PubMedID: 19047481 |
Title : A novel selective muscarinic acetylcholine receptor subtype 1 antagonist reduces seizures without impairing hippocampus-dependent learning - Sheffler_2009_Mol.Pharmacol_76_356 |
Author(s) : Sheffler DJ , Williams R , Bridges TM , Xiang Z , Kane AS , Byun NE , Jadhav S , Mock MM , Zheng F , Lewis LM , Jones CK , Niswender CM , Weaver CD , Lindsley CW , Conn PJ |
Ref : Molecular Pharmacology , 76 :356 , 2009 |
Abstract : |
PubMedSearch : Sheffler_2009_Mol.Pharmacol_76_356 |
PubMedID: 19407080 |
Title : Discovery of the first highly M5-preferring muscarinic acetylcholine receptor ligand, an M5 positive allosteric modulator derived from a series of 5-trifluoromethoxy N-benzyl isatins - Bridges_2009_J.Med.Chem_52_3445 |
Author(s) : Bridges TM , Marlo JE , Niswender CM , Jones CK , Jadhav SB , Gentry PR , Plumley HC , Weaver CD , Conn PJ , Lindsley CW |
Ref : Journal of Medicinal Chemistry , 52 :3445 , 2009 |
Abstract : |
PubMedSearch : Bridges_2009_J.Med.Chem_52_3445 |
PubMedID: 19438238 |
Title : Discovery and development of a potent and highly selective small molecule muscarinic acetylcholine receptor subtype I (mAChR 1 or M1) antagonist in vitro and in vivo probe - Weaver_2009_Curr.Top.Med.Chem_9_1217 |
Author(s) : Weaver CD , Sheffler DJ , Lewis LM , Bridges TM , Williams R , Nalywajko NT , Kennedy JP , Mulder MM , Jadhav S , Aldrich LA , Jones CK , Marlo JE , Niswender CM , Mock MM , Zheng F , Conn PJ , Lindsley CW |
Ref : Curr Top Med Chem , 9 :1217 , 2009 |
Abstract : |
PubMedSearch : Weaver_2009_Curr.Top.Med.Chem_9_1217 |
PubMedID: 19807667 |