Title : p-Trifluoromethyldiazirinyl-etomidate: a potent photoreactive general anesthetic derivative of etomidate that is selective for ligand-gated cationic ion channels - Husain_2010_J.Med.Chem_53_6432 |
Author(s) : Husain SS , Stewart D , Desai R , Hamouda AK , Li SG , Kelly E , Dostalova Z , Zhou X , Cotten JF , Raines DE , Olsen RW , Cohen JB , Forman SA , Miller KW |
Ref : Journal of Medicinal Chemistry , 53 :6432 , 2010 |
Abstract : |
PubMedSearch : Husain_2010_J.Med.Chem_53_6432 |
PubMedID: 20704351 |
Title : Time-resolved photolabeling of the nicotinic acetylcholine receptor by [3H]azietomidate, an open-state inhibitor - Chiara_2009_Mol.Pharmacol_75_1084 |
Author(s) : Chiara DC , Hong FH , Arevalo E , Husain SS , Miller KW , Forman SA , Cohen JB |
Ref : Molecular Pharmacology , 75 :1084 , 2009 |
Abstract : |
PubMedSearch : Chiara_2009_Mol.Pharmacol_75_1084 |
PubMedID: 19218367 |
Title : Synthesis of trifluoromethylaryl diazirine and benzophenone derivatives of etomidate that are potent general anesthetics and effective photolabels for probing sites on ligand-gated ion channels - Husain_2006_J.Med.Chem_49_4818 |
Author(s) : Husain SS , Nirthanan S , Ruesch D , Solt K , Cheng Q , Li GD , Arevalo E , Olsen RW , Raines DE , Forman SA , Cohen JB , Miller KW |
Ref : Journal of Medicinal Chemistry , 49 :4818 , 2006 |
Abstract : |
PubMedSearch : Husain_2006_J.Med.Chem_49_4818 |
PubMedID: 16884293 |
Title : Identification of binding sites in the nicotinic acetylcholine receptor for [3H]azietomidate, a photoactivatable general anesthetic - Ziebell_2004_J.Biol.Chem_279_17640 |
Author(s) : Ziebell MR , Nirthanan S , Husain SS , Miller KW , Cohen JB |
Ref : Journal of Biological Chemistry , 279 :17640 , 2004 |
Abstract : |
PubMedSearch : Ziebell_2004_J.Biol.Chem_279_17640 |
PubMedID: 14761946 |
Title : 2-(3-Methyl-3H-diaziren-3-yl)ethyl 1-(1-phenylethyl)-1H-imidazole-5-carboxylate: a derivative of the stereoselective general anesthetic etomidate for photolabeling ligand-gated ion channels - Husain_2003_J.Med.Chem_46_1257 |
Author(s) : Husain SS , Ziebell MR , Ruesch D , Hong F , Arevalo E , Kosterlitz JA , Olsen RW , Forman SA , Cohen JB , Miller KW |
Ref : Journal of Medicinal Chemistry , 46 :1257 , 2003 |
Abstract : |
PubMedSearch : Husain_2003_J.Med.Chem_46_1257 |
PubMedID: 12646036 |
Title : Identification of sites of incorporation in the nicotinic acetylcholine receptor of a photoactivatible general anesthetic - Pratt_2000_J.Biol.Chem_275_29441 |
Author(s) : Pratt MB , Husain SS , Miller KW , Cohen JB |
Ref : Journal of Biological Chemistry , 275 :29441 , 2000 |
Abstract : |
PubMedSearch : Pratt_2000_J.Biol.Chem_275_29441 |
PubMedID: 10859324 |
Title : Synthesis and properties of 3-(2-hydroxyethyl)-3-n-pentyldiazirine, a photoactivable general anesthetic - Husain_1999_J.Med.Chem_42_3300 |
Author(s) : Husain SS , Forman SA , Kloczewiak MA , Addona GH , Olsen RW , Pratt MB , Cohen JB , Miller KW |
Ref : Journal of Medicinal Chemistry , 42 :3300 , 1999 |
Abstract : |
PubMedSearch : Husain_1999_J.Med.Chem_42_3300 |
PubMedID: 10464016 |
Title : Where does cholesterol act during activation of the nicotinic acetylcholine receptor? - Addona_1998_Biochim.Biophys.Acta_1370_299 |
Author(s) : Addona GH , Sandermann H, Jr. , Kloczewiak MA , Husain SS , Miller KW |
Ref : Biochimica & Biophysica Acta , 1370 :299 , 1998 |
Abstract : |
PubMedSearch : Addona_1998_Biochim.Biophys.Acta_1370_299 |
PubMedID: 9545586 |
Title : Probing the agonist binding pocket in the nicotinic acetylcholine receptor: a high-resolution solid-state NMR approach - Williamson_1998_Biochemistry_37_10854 |
Author(s) : Williamson PT , Grobner G , Spooner PJ , Miller KW , Watts A |
Ref : Biochemistry , 37 :10854 , 1998 |
Abstract : |
PubMedSearch : Williamson_1998_Biochemistry_37_10854 |
PubMedID: 9692976 |
Title : Fourier transform infrared difference spectroscopy of the nicotinic acetylcholine receptor: evidence for specific protein structural changes upon desensitization - Baenziger_1993_Biochemistry_32_5448 |
Author(s) : Baenziger JE , Miller KW , Rothschild KJ |
Ref : Biochemistry , 32 :5448 , 1993 |
Abstract : |
PubMedSearch : Baenziger_1993_Biochemistry_32_5448 |
PubMedID: 8499448 |
Title : Probing conformational changes in the nicotinic acetylcholine receptor by Fourier transform infrared difference spectroscopy - Baenziger_1992_Biophys.J_62_64 |
Author(s) : Baenziger JE , Miller KW , McCarthy MP , Rothschild KJ |
Ref : Biophysical Journal , 62 :64 , 1992 |
Abstract : |
PubMedSearch : Baenziger_1992_Biophys.J_62_64 |
PubMedID: 1600101 |
Title : Incorporation of the nicotinic acetylcholine receptor into planar multilamellar films: characterization by fluorescence and Fourier transform infrared difference spectroscopy - Baenziger_1992_Biophys.J_61_983 |
Author(s) : Baenziger JE , Miller KW , Rothschild KJ |
Ref : Biophysical Journal , 61 :983 , 1992 |
Abstract : |
PubMedSearch : Baenziger_1992_Biophys.J_61_983 |
PubMedID: 1581507 |
Title : The modes of binding of ligands to cardiac muscarinic receptors - Birdsall_1989_Trends.Pharmacol.Sci_Suppl_31 |
Author(s) : Birdsall NJ , Chan SC , Eveleigh P , Hulme EC , Miller KW |
Ref : Trends in Pharmacological Sciences , Suppl :31 , 1989 |
Abstract : |
PubMedSearch : Birdsall_1989_Trends.Pharmacol.Sci_Suppl_31 |
PubMedID: 2694519 |