Title : Novel oxazolidinone calcitonin gene-related peptide (CGRP) receptor antagonists for the acute treatment of migraine - Crowley_2015_Bioorg.Med.Chem.Lett_25_4777 |
Author(s) : Crowley BM , Stump CA , Nguyen DN , Potteiger CM , McWherter MA , Paone DV , Quigley AG , Bruno JG , Cui D , Culberson JC , Danziger A , Fandozzi C , Gauvreau D , Kemmerer AL , Menzel K , Moore EL , Mosser SD , Reddy V , White RB , Salvatore CA , Kane SA , Bell IM , Selnick HG , Fraley ME , Burgey CS |
Ref : Bioorganic & Medicinal Chemistry Lett , 25 :4777 , 2015 |
Abstract : |
PubMedSearch : Crowley_2015_Bioorg.Med.Chem.Lett_25_4777 |
PubMedID: 26231160 |
Title : Identification of potent, highly constrained CGRP receptor antagonists - Stump_2010_Bioorg.Med.Chem.Lett_20_2572 |
Author(s) : Stump CA , Bell IM , Bednar RA , Fay JF , Gallicchio SN , Hershey JC , Jelley R , Kreatsoulas C , Moore EL , Mosser SD , Quigley AG , Roller SA , Salvatore CA , Sharik SS , Theberge CR , Zartman CB , Kane SA , Graham SL , Selnick HG , Vacca JP , Williams TM |
Ref : Bioorganic & Medicinal Chemistry Lett , 20 :2572 , 2010 |
Abstract : |
PubMedSearch : Stump_2010_Bioorg.Med.Chem.Lett_20_2572 |
PubMedID: 20299218 |
Title : The discovery of highly potent CGRP receptor antagonists - Stump_2009_Bioorg.Med.Chem.Lett_19_214 |
Author(s) : Stump CA , Bell IM , Bednar RA , Bruno JG , Fay JF , Gallicchio SN , Johnston VK , Moore EL , Mosser SD , Quigley AG , Salvatore CA , Theberge CR , Blair Zartman C , Zhang XF , Kane SA , Graham SL , Vacca JP , Williams TM |
Ref : Bioorganic & Medicinal Chemistry Lett , 19 :214 , 2009 |
Abstract : |
PubMedSearch : Stump_2009_Bioorg.Med.Chem.Lett_19_214 |
PubMedID: 19010673 |
Title : Novel CGRP receptor antagonists through a design strategy of target simplification with addition of molecular flexibility - Wood_2009_Bioorg.Med.Chem.Lett_19_5787 |
Author(s) : Wood MR , Schirripa KM , Kim JJ , Quigley AG , Stump CA , Bell IM , Bednar RA , Fay JF , Bruno JG , Moore EL , Mosser SD , Roller S , Salvatore CA , Kane SA , Vacca JP , Selnick HG |
Ref : Bioorganic & Medicinal Chemistry Lett , 19 :5787 , 2009 |
Abstract : |
PubMedSearch : Wood_2009_Bioorg.Med.Chem.Lett_19_5787 |
PubMedID: 19703767 |
Title : Benzodiazepine calcitonin gene-related peptide (CGRP) receptor antagonists: optimization of the 4-substituted piperidine - Burgey_2006_Bioorg.Med.Chem.Lett_16_5052 |
Author(s) : Burgey CS , Stump CA , Nguyen DN , Deng JZ , Quigley AG , Norton BR , Bell IM , Mosser SD , Salvatore CA , Rutledge RZ , Kane SA , Koblan KS , Vacca JP , Graham SL , Williams TM |
Ref : Bioorganic & Medicinal Chemistry Lett , 16 :5052 , 2006 |
Abstract : |
PubMedSearch : Burgey_2006_Bioorg.Med.Chem.Lett_16_5052 |
PubMedID: 16889959 |